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Gabriele La Monica
Gabriele La Monica
Research Fellow, University of Palermo (Italy), "STEBICEF" Department
在 unipa.it 的电子邮件经过验证 - 首页
标题
引用次数
引用次数
年份
Targeting SARS-CoV-2 Main Protease for Treatment of COVID-19: Covalent Inhibitors Structure–Activity Relationship Insights and Evolution Perspectives
G La Monica, A Bono, A Lauria, A Martorana
Journal of Medicinal Chemistry 65 (19), 12500-12534, 2022
722022
Quinoline anticancer agents active on DNA and DNA-interacting proteins: From classical to emerging therapeutic targets
A Lauria, G La Monica, A Bono, A Martorana
European Journal of Medicinal Chemistry 220, 113555, 2021
522021
Quinoline-Based Molecules Targeting c-Met, EGF, and VEGF Receptors and the Proteins Involved in Related Carcinogenic Pathways
A Martorana, G La Monica, A Lauria
Molecules 25 (18), 4279, 2020
392020
In Silico Identification of Small Molecules as New Cdc25 Inhibitors through the Correlation between Chemosensitivity and Protein Expression Pattern
A Lauria, A Martorana, G La Monica, S Mannino, G Mannino, D Peri, ...
International Journal of Molecular Sciences 22 (7), 3714, 2021
132021
Off-Target-Based Design of Selective HIV-1 PROTEASE Inhibitors
G La Monica, A Lauria, A Bono, A Martorana
International journal of molecular sciences 22 (11), 6070, 2021
62021
Antiproliferative Activity Predictor: A New Reliable In Silico Tool for Drug Response Prediction against NCI60 Panel
A Martorana, G La Monica, A Bono, S Mannino, S Buscemi, ...
International Journal of Molecular Sciences 23 (22), 14374, 2022
52022
In Silico Design of New Dual Inhibitors of SARS-CoV-2 MPRO through Ligand-and Structure-Based Methods
A Bono, A Lauria, G La Monica, F Alamia, F Mingoia, A Martorana
International Journal of Molecular Sciences 24 (9), 8377, 2023
42023
Synthesis of new antiproliferative 1, 3, 4-substituted-pyrrolo [3, 2-c] quinoline derivatives, biological and in silico insights
F Mingoia, C Di Sano, C D'Anna, M Fazzari, L Minafra, A Bono, ...
European Journal of Medicinal Chemistry 258, 115537, 2023
22023
One pot-like regiospecific access to 1-aryl-1H-pyrazol-3 (2H)-one derivatives and evaluation of the anticancer activity
F Mingoia, G Panzeca, MC Vitale, G La Monica, A Bono, A Lauria, ...
Arkivoc 2022, 191-203, 2022
22022
Antiproliferative Properties and G-Quadruplex-Binding of Symmetrical Naphtho [1, 2-b: 8, 7-b’] dithiophene Derivatives
A Lauria, G La Monica, A Terenzi, G Mannino, R Bonsignore, A Bono, ...
Molecules 26 (14), 4309, 2021
22021
Identification of biological targets through the correlation between cell line chemosensitivity and protein expression pattern
A Lauria, G La Monica, C Gentile, G Mannino, A Martorana, D Peri
Drug Discovery Today 26 (10), 2431-2438, 2021
12021
Scaffold-Hopping Strategies in Aurone Optimization: A Comprehensive Review of Synthetic Procedures and Biological Activities of Nitrogen and Sulfur Analogues
G La Monica, F Alamia, A Bono, A Lauria, A Martorana
Molecules 29 (12), 2813, 2024
2024
Bioisosteric heterocyclic analogues of natural bioactive flavonoids by scaffold-hopping approaches: State-of-the-art and perspectives in medicinal chemistry
G La Monica, A Bono, F Alamia, A Lauria, A Martorana
Bioorganic & Medicinal Chemistry, 117791, 2024
2024
Development of an inhibitor of the mutagenic SOS response that suppresses the evolution of quinolone antibiotic resistance
JD Bradbury, T Hodgkinson, AM Thomas, O Tanwar, G La Monica, ...
Chemical Science, 2024
2024
In silico lead optimization and synthesis of a new series of thieno [3, 2-c] quinoline with antiproliferative activity on RET-dependent medullary thyroid cancer cells
G LA MONICA, G Pizzolanti, C Baiamonte, A Bono, F Alamia, G Siragusa, ...
Convegno Congiunto delle Sezioni Sicilia e Calabria della Società Chimica …, 2023
2023
Correction to “Design and Synthesis of Novel Thieno[3,2-c]quinoline Compounds with Antiproliferative Activity on RET-Dependent Medullary Thyroid Cancer Cells”
G La Monica, G Pizzolanti, C Baiamonte, A Bono, F Alamia, F Mingoia, ...
ACS omega 8 (50), 48582-48582, 2023
2023
Design and Synthesis of Novel Thieno[3,2-c]quinoline Compounds with Antiproliferative Activity on RET-Dependent Medullary Thyroid Cancer Cells
G La Monica, G Pizzolanti, C Baiamonte, A Bono, F Alamia, F Mingoia, ...
ACS omega 8 (38), 34640-34649, 2023
2023
In Silico Mixed Ligand/Structure-Based Design of New CDK-1/PARP-1 Dual Inhibitors as Anti-Breast Cancer Agents
A Bono, G La Monica, F Alamia, F Mingoia, C Gentile, D Peri, A Lauria, ...
International Journal of Molecular Sciences 24 (18), 13769, 2023
2023
Antiproliferative Activity Predictor: un nuovo tool in silico per predire l’attività antiproliferativa nei confronti del pannello NCI60
G LA MONICA, A Martorana, A Bono, S Mannino, S Buscemi, ...
Convegno Congiunto Sezioni Calabria e Sicilia Società Chimica Italiana …, 2022
2022
Correlation between cell line chemosensitivity and protein expression pattern as new approach for the design of targeted anticancer small molecules
G LA MONICA
Università degli Studi di Palermo, 2022
2022
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