关注
Elma Mons
Elma Mons
在 biology.leidenuniv.nl 的电子邮件经过验证
标题
引用次数
引用次数
年份
The alkyne moiety as a latent electrophile in irreversible covalent small molecule inhibitors of cathepsin K
E Mons, IDC Jansen, J Loboda, BR van Doodewaerd, J Hermans, ...
Journal of the American Chemical Society 141 (8), 3507-3514, 2019
952019
Organocatalytic enantioselective Pictet–Spengler reactions for the syntheses of 1-substituted 1, 2, 3, 4-tetrahydroisoquinolines
E Mons, MJ Wanner, S Ingemann, JH van Maarseveen, H Hiemstra
The Journal of Organic Chemistry 79 (16), 7380-7390, 2014
842014
A comprehensive guide for assessing covalent inhibition in enzymatic assays illustrated with kinetic simulations
E Mons, S Roet, RQ Kim, MPC Mulder
Current Protocols 2 (6), e419, 2022
462022
Exploring the versatility of the covalent thiol–alkyne reaction with substituted propargyl warheads: a deciding role for the cysteine protease
E Mons, RQ Kim, BR van Doodewaerd, PA van Veelen, MPC Mulder, ...
Journal of the American Chemical Society 143 (17), 6423-6433, 2021
452021
Profiling withanolide A for therapeutic targets in neurodegenerative diseases
EA Crane, W Heydenreuter, KR Beck, P Strajhar, J Vomacka, M Smiesko, ...
Bioorganic & medicinal chemistry 27 (12), 2508-2520, 2019
122019
Technologies for Direct Detection of Covalent Protein–Drug Adducts
E Mons, RQ Kim, MPC Mulder
Pharmaceuticals 16 (4), 547, 2023
72023
Cathepsin Inhibitors
H Ovaa, MWE Mons, S van Boeckel
WO2019112426A1, 2019
32019
Alkynes in covalent enzyme inhibitors: down the kinetic rabbit hole
E Mons
Leiden University, 2024
2024
系统目前无法执行此操作,请稍后再试。
文章 1–8