Physicochemical characterization and in vitro dissolution studies of solid dispersions of ketoprofen with PVP K30 and D-mannitol PS Yadav, V Kumar, UP Singh, HR Bhat, B Mazumder Saudi Pharmaceutical Journal 21 (1), 77-84, 2013 | 132 | 2013 |
Antifungal activity, SAR and physicochemical correlation of some clubbed thiazole-1,3,5-triazine derivatives. UP Singh, HR Bhat, P Gahtori Journal de Mycologie Médicale / Journal of Medical Mycology 22 (2), 134-141, 2012 | 86* | 2012 |
Antimalarial evaluation and docking studies of hybrid phenylthiazolyl-1, 3, 5-triazine derivatives: A novel and potential antifolate lead for< i> Pf-</i> DHFR-TS inhibition P Gahtori, SK Ghosh, P Parida, A Prakash, K Gogoi, HR Bhat, UP Singh Experimental Parasitology 130 (3), 292-299, 2012 | 77 | 2012 |
1, 3, 5‐Triazine: A versatile pharmacophore with diverse biological activities S Singh, MK Mandal, A Masih, A Saha, SK Ghosh, HR Bhat, UP Singh Archiv der Pharmazie 354 (6), 2000363, 2021 | 76 | 2021 |
Design and discovery of novel monastrol-1,3,5-triazines as potent anti-breast cancer agent via attenuating Epidermal Growth Factor Receptor tyrosine kinase JK Srivastava, GG Pillai, HR Bhat, A Verma, UP Singh Scientific Reports 7 (1), 5851, 2017 | 76 | 2017 |
4-Aminoquinoline-1, 3, 5-triazine: Design, synthesis, in vitro antimalarial activity and docking studies HR Bhat, UP Singh, P Gahtori, SK Ghosh, K Gogoi, A Prakash, RK Singh New Journal of Chemistry 37 (9), 2654-2662, 2013 | 69 | 2013 |
Structure-guided discovery of 1, 3, 5-triazine–pyrazole conjugates as antibacterial and antibiofilm agent against pathogens causing human diseases with favorable metabolic fate B Singh, HR Bhat, MK Kumawat, UP Singh Bioorganic & medicinal chemistry letters 24 (15), 3321-3325, 2014 | 66 | 2014 |
Antimalarial activity and docking studies of novel bi-functional hybrids derived from 4-aminoquinoline and 1, 3, 5-triazine against wild and mutant malaria parasites as pf-DHFR … HR Bhat, UP Singh, P Gahtori, SK Ghosh, K Gogoi, A Prakash, RK Singh RSC Advances 3 (9), 2942-2952, 2013 | 59 | 2013 |
Design, Facile Synthesis, and Antibacterial Activity of Hybrid 1, 3, 4‐thiadiazole‐1, 3, 5‐triazine Derivatives Tethered via–S–Bridge V Dubey, M Pathak, HR Bhat, UP Singh Chemical Biology & Drug Design 80 (4), 598-604, 2012 | 55 | 2012 |
Design, Synthesis, Antibacterial Activity, and Molecular Docking Studies of Novel Hybrid 1, 3‐Thiazine‐1, 3, 5‐Triazine Derivatives as Potential Bacterial Translation Inhibitor UP Singh, M Pathak, V Dubey, HR Bhat, P Gahtori, RK Singh Chemical biology & drug design 80 (4), 572-583, 2012 | 55 | 2012 |
Review on Synthetic Chemistry and Antibacterial Importance of Thiazole Derivatives A Kashyap, N Adhikari, A Das, A Shakya, SK Ghosh, UP Singh, HR Bhat Current drug discovery technologies 15 (3), 214-228, 2018 | 50 | 2018 |
Design, synthesis, anticancer, antibacterial, and antifungal evaluation of 4‐aminoquinoline‐1, 3, 5‐triazine derivatives HR Bhat, A Masih, A Shakya, SK Ghosh, UP Singh Journal of Heterocyclic Chemistry 57 (1), 390-399, 2020 | 49 | 2020 |
Synthesis and antibacterial evaluation of series of novel tri-substituted-s-triazine derivatives UP Singh, RK Singh, HR Bhat, YP Subhashchandra, V Kumar, ... Medicinal Chemistry Research 20 (9), 1603-1610, 2010 | 49 | 2010 |
Discovery of novel 1, 3, 5-triazine-thiazolidine-2, 4-diones as dipeptidyl peptidase-4 inhibitors with antibacterial activity targeting the S1 pocket for the treatment of type … JK Srivastava, P Dubey, S Singh, HR Bhat, MK Kumawat, UP Singh RSC Advances 5 (19), 14095-14102, 2015 | 47 | 2015 |
Synthesis, characterization and antimalarial activity of hybrid 4-aminoquinoline-1, 3, 5-triazine derivatives HR Bhat, UP Singh, PS Yadav, V Kumar, P Gahtori, A Das, D Chetia, ... Arabian Journal of Chemistry 9, S625-S631, 2016 | 46 | 2016 |
In silico ADMET study, docking, synthesis and antimalarial evaluation of thiazole-1, 3, 5-triazine derivatives as Pf-DHFR inhibitor S Sahu, SK Ghosh, P Gahtori, UP Singh, DR Bhattacharyya, HR Bhat Pharmacological Reports 71 (5), 762-767, 2019 | 44 | 2019 |
Synthesis, SAR and antibacterial activity of hybrid chloro, dichloro-phenylthiazolyl-s-triazines P Gahtori, SK Ghosh, B Singh, UP Singh, HR Bhat, A Uppal Saudi Pharmaceutical Journal 20 (1), 35-43, 2012 | 42 | 2012 |
Synthesis, antimalarial activity and molecular docking of hybrid 4-aminoquinoline-1, 3, 5-triazine derivatives HR Bhat, UP Singh, A Thakur, SK Ghosh, K Gogoi, A Prakash, RK Singh Experimental parasitology 157, 59-67, 2015 | 41 | 2015 |
Discovery of potent, novel antibacterial hybrid conjugates from 4-aminoquinoline and 1, 3, 5-triazine: design, synthesis and antibacterial evaluation HR Bhat, SK Gupta, UP Singh RSC Advances 2 (33), 12690-12695, 2012 | 40 | 2012 |
Discovery of novel pyrazole derivatives as a potent anti‐inflammatory agent in RAW264. 7 cells via inhibition of NF‐ĸB for possible benefit against SARS‐CoV‐2 A Masih, AK Agnihotri, JK Srivastava, N Pandey, HR Bhat, UP Singh Journal of biochemical and molecular toxicology 35 (3), e22656, 2021 | 39 | 2021 |