Molecular Iodine Promoted Divergent Synthesis of Benzimidazoles, Benzothiazoles, and 2-Benzyl-3-phenyl-3,4-dihydro-2H-benzo[e][1,2,4]thiadiazines G Naresh, R Kant, T Narender The Journal of Organic Chemistry 79 (9), 3821-3829, 2014 | 88 | 2014 |
Silver (I)-Catalyzed regioselective construction of highly substituted α-naphthols and its application toward expeditious synthesis of lignan natural products G Naresh, R Kant, T Narender Organic letters 17 (14), 3446-3449, 2015 | 70 | 2015 |
Insights into current tropomyosin receptor kinase (TRK) inhibitors: development and clinical application W Yan, NR Lakkaniga, F Carlomagno, M Santoro, NQ McDonald, F Lv, ... Journal of medicinal chemistry 62 (4), 1731-1760, 2018 | 62 | 2018 |
Copper (II) catalyzed expeditious synthesis of furoquinoxalines through a one-pot three-component coupling strategy G Naresh, R Kant, T Narender Organic letters 16 (17), 4528-4531, 2014 | 51 | 2014 |
Catalyst free, C-3 functionalization of imidazo [1, 2-a] pyridines to rapidly access new chemical space for drug discovery efforts N Gunaganti, A Kharbanda, NR Lakkaniga, L Zhang, R Cooper, H Li, ... Chemical Communications 54 (92), 12954-12957, 2018 | 34 | 2018 |
Glucose uptake stimulatory effect of 4-hydroxypipecolic acid by increased GLUT 4 translocation in skeletal muscle cells G Naresh, N Jaiswal, P Sukanya, AK Srivastava, AK Tamrakar, ... Bioorganic & medicinal chemistry letters 22 (17), 5648-5651, 2012 | 32 | 2012 |
Discovery of SP-96, the first non-ATP-competitive Aurora Kinase B inhibitor, for reduced myelosuppression NR Lakkaniga, L Zhang, B Belachew, N Gunaganti, B Frett, H Li European Journal of Medicinal Chemistry 203, 112589, 2020 | 28 | 2020 |
Molecular iodine mediated synthesis of polysubstituted oxazoles by oxidative domino cyclization in water G Naresh, T Narender RSC Advances 4 (23), 11862-11866, 2014 | 27 | 2014 |
Pyrrolo [2, 3-d] pyrimidine derivatives as inhibitors of RET: Design, synthesis and biological evaluation NR Lakkaniga, N Gunaganti, L Zhang, B Belachew, B Frett, YK Leung, ... European journal of medicinal chemistry 206, 112691, 2020 | 23 | 2020 |
Use of Imidazo[1,2‐a]pyridine as a Carbonyl Surrogate in a Mannich‐Like, Catalyst Free, One‐Pot Reaction G Naresh, NR Lakkaniga, A Kharbanda, W Yan, B Frett, H Li European Journal of Organic Chemistry 2019 (4), 770-777, 2019 | 16 | 2019 |
Selective, C-3 Friedel-Crafts acylation to generate functionally diverse, acetylated Imidazo [1, 2-a] pyridine derivatives B Frett, N McConnell, A Kharbanda, G Naresh, B Rounseville, C Warner, ... Tetrahedron 74 (35), 4592-4600, 2018 | 16 | 2018 |
Rational Design, Synthesis and Biological Evaluation of Pyrimidine-4, 6-diamine derivatives as Type-II inhibitors of FLT3 Selective Against c-KIT JB Bharate, N McConnell, G Naresh, L Zhang, NR Lakkaniga, L Ding, ... Scientific reports 8 (1), 1-18, 2018 | 15 | 2018 |
Free fatty acid induced impairment of insulin signaling is prevented by the diastereomeric mixture of calophyllic acid and isocalophyllic acid in skeletal muscle cells N Jaiswal, N Gunaganti, CK Maurya, T Narender, AK Tamrakar European Journal of Pharmacology 746, 70-77, 2015 | 13 | 2015 |
Medicinal Chemistry Optimization of a Diaminopurine Chemotype: Toward a Lead for Trypanosoma brucei Inhibitors B Singh, R Diaz-Gonzalez, G Ceballos-Perez, DI Rojas-Barros, ... Journal of medicinal chemistry 63 (17), 9912-9927, 2020 | 7 | 2020 |
Antifilarial Activity of Constituents of Calophyllum inophyllum and their Derivatives Jankiprasad, G Naresh, J Gupta, SM Bhattacharya, SM Rajendran, ... Natural Product Communications 8 (6), 1934578X1300800630, 2013 | 6 | 2013 |
An imidazo [1, 2-a] pyridine-pyridine derivative potently inhibits FLT3-ITD and FLT3-ITD secondary mutants, including gilteritinib-resistant FLT3-ITD/F691L X Wang, RA DeFilippis, T Weldemichael, N Gunaganti, P Tran, YK Leung, ... European Journal of Medicinal Chemistry 264, 115977, 2024 | 5 | 2024 |
Chemical optimization of Cbl0137 for human African trypanosomiasis Lead drug discovery B Singh, A Sharma, N Gunaganti, M Rivers, PK Gadekar, B Greene, ... Journal of Medicinal Chemistry 66 (3), 1972-1989, 2023 | 4 | 2023 |
β-Amino acid derivatives as mitochondrial complex III inhibitors of L. donovani: a promising chemotype targeting visceral leishmaniasis P Chandrakar, N Gunaganti, N Parmar, A Kumar, SK Singh, M Rashid, ... European Journal of Medicinal Chemistry 182, 111632, 2019 | 4 | 2019 |
Targeting Aurora-kinase B with the novel Aurora Kinase B inhibitor MK7 in multiple myeloma J Contreras, E Caldas-Lopes, D Jayabalan, J Monge, N Lombardi, H Li, ... Clinical Lymphoma, Myeloma and Leukemia 19 (10), e128, 2019 | 1 | 2019 |
KINASE INHIBITOR REPURPOSING FOR NEGLECTED TROPICAL DISEASES. R Díaz-González, C Bosch-Navarrete, G Pérez-Moreno, C Cordon-Obras, ... | | 2022 |