Palladium-Catalyzed Intramolecular Oxidative Coupling Involving Double C(sp2)–H Bonds for the Synthesis of Annulated Biaryl Sultams JK Laha, KP Jethava, N Dayal The Journal of Organic Chemistry 79 (17), 8010-8019, 2014 | 115 | 2014 |
Spectral deep learning for prediction and prospective validation of functional groups JA Fine, AA Rajasekar, KP Jethava, G Chopra Chemical science 11 (18), 4618-4630, 2020 | 95 | 2020 |
Access to Biaryl Sulfonamides by Palladium-Catalyzed Intramolecular Oxidative Coupling and Subsequent Nucleophilic Ring Opening of Heterobiaryl Sultams with Amines JK Laha, N Dayal, KP Jethava, DV Prajapati Organic letters 17 (5), 1296-1299, 2015 | 72 | 2015 |
Scope of successive C–H functionalizations of the methyl group in 3-picolines: intramolecular carbonylation of arenes to the metal-free synthesis of 4-azafluorenones JK Laha, KP Jethava, S Patel Organic letters 17 (23), 5890-5893, 2015 | 50 | 2015 |
Intramolecular Minisci acylation under silver-free neutral conditions for the synthesis of azafluorenones and fluorenones JK Laha, KV Patel, G Dubey, KP Jethava Organic & Biomolecular Chemistry 15 (10), 2199-2210, 2017 | 42 | 2017 |
Implications of dynamic imine chemistry for the sustainable synthesis of nitrogen heterocycles via transimination followed by intramolecular cyclisation JK Laha, KSS Tummalapalli, KP Jethava Organic & Biomolecular Chemistry 14 (8), 2473-2479, 2016 | 39 | 2016 |
Palladium-catalyzed regio-and chemoselective ortho-benzylation of C–H bond using a functionalizable primary amide directing group: a concise synthesis of dibenzo [b, e] azepin … JK Laha, PU Shah, KP Jethava Chemical Communications 49 (69), 7623-7625, 2013 | 39 | 2013 |
Intramolecular acylation of unactivated pyridines or arenes via multiple C–H functionalizations: Synthesis of all four azafluorenones and fluorenones JK Laha, KP Jethava, S Patel, KV Patel The Journal of Organic Chemistry 82 (1), 76-85, 2017 | 35 | 2017 |
Monitoring phagocytic uptake of amyloid β into glial cell lysosomes in real time P Prakash, KP Jethava, N Korte, P Izquierdo, E Favuzzi, IVL Rose, ... Chemical Science 12 (32), 10901-10918, 2021 | 25 | 2021 |
Accelerated Reactivity Mechanism and Interpretable Machine Learning Model of N-Sulfonylimines toward Fast Multicomponent Reactions KP Jethava, J Fine, Y Chen, A Hossain, G Chopra Organic Letters 22 (21), 8480-8486, 2020 | 23 | 2020 |
Access to imidazolidine-fused sulfamidates and sulfamides bearing a quaternary center via 1, 3-dipolar cycloaddition of nonstabilized azomethine ylides JK Laha, KP Jethava The Journal of Organic Chemistry 82 (7), 3597-3604, 2017 | 23 | 2017 |
Rapid, refined, and robust method for expression, purification, and characterization of recombinant human amyloid beta 1-42 P Prakash, TC Lantz, KP Jethava, G Chopra Methods and protocols 2 (2), 48, 2019 | 11 | 2019 |
Synthesis of Mono‐N‐sulfonylimidazolidines by a 1,3‐Dipolar Cycloaddition Strategy, as an Alternative to Selective N‐Sulfonylation, and Their Ring Cleavage To … JK Laha, KP Jethava, KSS Tummalapalli, S Sharma European Journal of Organic Chemistry 2017 (31), 4617-4624, 2017 | 11 | 2017 |
Combined molecular graph neural network and structural docking selects potent programmable cell death protein 1/programmable death-ligand 1 (PD-1/PD-L1) small molecule inhibitors PR Wijewardhane, KP Jethava, JA Fine, G Chopra | 8 | 2020 |
Palladium-Catalyzed Oxidative Annulation of Pyrrolylalkyl-1H-azoles: Towards the Synthesis of Polyheterocyclic Arenes KN Tripathi, AH Bansode, RP Singh Synthesis 52 (05), 719-726, 2020 | 5 | 2020 |
One Scaffold, Different Organelle Sensors: pH‐Activable Fluorescent Probes for Targeting Live Microglial Cell Organelles KP Jethava, P Prakash, P Manchanda, H Arora, G Chopra ChemBioChem 23 (9), e202100378, 2022 | 2 | 2022 |
Graph Neural Networks Bootstrapped for Synthetic Selection and Validation of Small Molecule Immunomodulators PR Wijewardhane, KP Jethava, JA Fine, G Chopra | 2 | 2021 |
Compounds with immunomodulatory activity and therapeutic uses thereof G Chopra, P Wijewardhane, KP Jethava, J Fine US Patent App. 17/908,530, 2023 | 1 | 2023 |
Front Cover: One Scaffold, Different Organelle Sensors: pH‐Activable Fluorescent Probes for Targeting Live Microglial Cell Organelles (ChemBioChem 9/2022) KP Jethava, P Prakash, P Manchanda, H Arora, G Chopra ChemBioChem 23 (9), e202100667, 2022 | 1 | 2022 |
Ph-activable fluorescent probes for targeting cell organelles G Chopra, K Jethava, P Prakash US Patent App. 18/281,188, 2024 | | 2024 |