| Comparison between steroid binding to membrane progesterone receptor α (mPRα) and to nuclear progesterone receptor: Correlation with physicochemical properties assessed by … J Kelder, R Azevedo, Y Pang, J de Vlieg, J Dong, P Thomas Steroids 75 (4-5), 314-322, 2010 | 95 | 2010 |
| OpenClinica M Cavelaars, J Rousseau, C Parlayan, S de Ridder, A Verburg, R Ross, ... Journal of clinical bioinformatics 5 (S1), S2, 2015 | 53 | 2015 |
| X-ray structure of p38α bound to TAK-715: comparison with three classic inhibitors R Azevedo, M van Zeeland, H Raaijmakers, B Kazemier, J de Vlieg, ... Acta Crystallographica Section D: Biological Crystallography 68 (8), 1041-1050, 2012 | 43 | 2012 |
| Discovery of pyrazolo [1, 5-a] pyrimidine-based Pim inhibitors: a template-based approach MP Dwyer, K Keertikar, K Paruch, C Alvarez, M Labroli, C Poker, ... Bioorganic & medicinal chemistry letters 23 (22), 6178-6182, 2013 | 42 | 2013 |
| X-ray structures of progesterone receptor ligand binding domain in its agonist state reveal differing mechanisms for mixed profiles of 11β-substituted steroids SJ Lusher, HCA Raaijmakers, D Vu-Pham, B Kazemier, R Bosch, ... Journal of Biological Chemistry 287 (24), 20333-20343, 2012 | 38 | 2012 |
| RORgammaT inhibitors WFJ Karstens, M Van Der Stelt, J Cals, RCRG Azevedo, KJ Barr, H Zhang, ... US Patent 9,095,583, 2015 | 23 | 2015 |
| Multidimensional profiling of CSF1R screening hits and inhibitors: assessing cellular activity, target residence time, and selectivity in a higher throughput way JCM Uitdehaag, CM Sünnen, AM van Doornmalen, N de Rouw, A Oubrie, ... Journal of biomolecular screening 16 (9), 1007-1017, 2011 | 23 | 2011 |
| A molecular informatics view on best practice in multi-parameter compound optimization SJ Lusher, R McGuire, R Azevedo, JW Boiten, RC van Schaik, J de Vlieg Drug discovery today 16 (13-14), 555-568, 2011 | 23 | 2011 |
| RORgammaT inhibitors WFJ Karstens, M Van Der Stelt, J Cals, RCRG Azevedo, KJ Barr, H Zhang, ... US Patent 9,603,838, 2017 | 20 | 2017 |
| Systematically linking tranSMART, Galaxy and EGA for reusing human translational research data C Zhang, J Bijlard, C Staiger, S Scollen, D van Enckevort, Y Hoogstrate, ... F1000Research 6, 2017 | 11 | 2017 |
| TranSMART M Bierkens, W van der Linden, K van Bochove, W Weistra, RJA Fijneman, ... Journal of clinical bioinformatics 5 (1), S9, 2015 | 9 | 2015 |
| Comparison between steroid binding to progesterone membrane receptor α (mPRα) and to progesterone nuclear receptor: correlation with physicochemical properties assessed by … J Kelder, R Azevedo, Y Pang, J de Vlieg, J Dong, P Thomas Steroids 75 (4-5), 314, 2010 | 8 | 2010 |
| RORgammaT inhibitors WFJ Karstens, M Van Der Stelt, J Cals, RCRG Azevedo, KJ Barr, H Zhang, ... US Patent 9,884,043, 2018 | 4 | 2018 |
| Substituted thieno [2, 3-b] pyrazine compounds as modulators of B-Raf kinase activity BJB Folmer, ES Gernette, RCRG Azevedo, H Ibrahim US Patent 8,669,256, 2014 | 4 | 2014 |
| Identification of Novel Bacterial M. SssI DNA Methyltransferase Inhibitors M Hupkes, R Azevedo, H Jansen, EJ van Zoelen, KJ Dechering Journal of biomolecular screening 18 (3), 348-355, 2013 | 3 | 2013 |
| Querying, viewing and analyzing colorectal cancer translational research studies in tranSMART M Bierkens, W van der Linden, W Weistra, K Van Bochove, JAM Beliën, ... Cancer Research 76 (14 Supplement), 3166-3166, 2016 | 2 | 2016 |
| Informatics Solutions for Biomarker Discovery and JW Boiten, R Azevedo, M Cavelaars, JAM Maas, GA Meijer Handbook of Biomarkers and Precision Medicine, 135, 2019 | | 2019 |
