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Rolando Cannalire
Rolando Cannalire
在 unina.it 的电子邮件经过验证
标题
引用次数
引用次数
年份
Visible light photocatalysis in the late-stage functionalization of pharmaceutically relevant compounds
R Cannalire, S Pelliccia, L Sancineto, E Novellino, GC Tron, ...
Chemical Society Reviews 50 (2), 766-897, 2021
2562021
Targeting SARS-CoV-2 proteases and polymerase for COVID-19 treatment: state of the art and future opportunities
R Cannalire, C Cerchia, AR Beccari, FS Di Leva, V Summa
Journal of medicinal chemistry 65 (4), 2716-2746, 2020
1842020
Identification of inhibitors of SARS-CoV-2 3CL-pro enzymatic activity using a small molecule in vitro repurposing screen
M Kuzikov, E Costanzi, J Reinshagen, F Esposito, L Vangeel, M Wolf, ...
ACS pharmacology & translational science 4 (3), 1096-1110, 2021
1172021
SARS-CoV-2 entry inhibitors: Small molecules and peptides targeting virus or host cells
R Cannalire, I Stefanelli, C Cerchia, AR Beccari, S Pelliccia, V Summa
International journal of molecular sciences 21 (16), 5707, 2020
772020
Targeting flavivirus RNA dependent RNA polymerase through a pyridobenzothiazole inhibitor
D Tarantino, R Cannalire, E Mastrangelo, R Croci, G Querat, ML Barreca, ...
Antiviral research 134, 226-235, 2016
582016
A journey around the medicinal chemistry of hepatitis C virus inhibitors targeting NS4B: from target to preclinical drug candidates
R Cannalire, ML Barreca, G Manfroni, V Cecchetti
Journal of medicinal chemistry 59 (1), 16-41, 2016
562016
The versatile nature of the 6-aminoquinolone scaffold: identification of submicromolar hepatitis C virus NS5B inhibitors
G Manfroni, R Cannalire, ML Barreca, N Kaushik-Basu, P Leyssen, ...
Journal of medicinal chemistry 57 (5), 1952-1963, 2014
522014
Natural compounds inhibit SARS-CoV-2 nsp13 unwinding and ATPase enzyme activities
A Corona, K Wycisk, C Talarico, C Manelfi, J Milia, R Cannalire, ...
ACS pharmacology & translational science 5 (4), 226-239, 2022
502022
2-Phenylquinoline S. aureus NorA Efflux Pump Inhibitors: Evaluation of the Importance of Methoxy Group Introduction
T Felicetti, R Cannalire, D Pietrella, G Latacz, A Lubelska, G Manfroni, ...
Journal of medicinal chemistry 61 (17), 7827-7848, 2018
492018
Mode of action of the 2-phenylquinoline efflux inhibitor PQQ4R against Escherichia coli
D Machado, L Fernandes, SS Costa, R Cannalire, G Manfroni, O Tabarrini, ...
PeerJ 5, e3168, 2017
382017
New pyrazolobenzothiazine derivatives as hepatitis C virus NS5B polymerase palm site I inhibitors
G Manfroni, D Manvar, ML Barreca, N Kaushik-Basu, P Leyssen, ...
Journal of medicinal chemistry 57 (8), 3247-3262, 2014
372014
Searching for Novel Inhibitors of the S. aureus NorA Efflux Pump: Synthesis and Biological Evaluation of the 3‐Phenyl‐1,4‐benzothiazine Analogues
T Felicetti, R Cannalire, MS Burali, S Massari, G Manfroni, ML Barreca, ...
ChemMedChem 12 (16), 1293-1302, 2017
352017
Functionalized 2, 1-benzothiazine 2, 2-dioxides as new inhibitors of Dengue NS5 RNA-dependent RNA polymerase
R Cannalire, D Tarantino, A Astolfi, ML Barreca, S Sabatini, S Massari, ...
European journal of medicinal chemistry 143, 1667-1676, 2018
322018
Natural isoflavone biochanin A as a template for the design of new and potent 3-phenylquinolone efflux inhibitors against Mycobacterium avium
R Cannalire, D Machado, T Felicetti, SS Costa, S Massari, G Manfroni, ...
European Journal of Medicinal Chemistry 140, 321-330, 2017
322017
Pyridobenzothiazolones exert potent anti-dengue activity by hampering multiple functions of NS5 polymerase
R Cannalire, KW Ki Chan, MS Burali, CP Gwee, S Wang, A Astolfi, ...
ACS Medicinal Chemistry Letters 11 (5), 773-782, 2020
272020
Boosting Effect of 2-Phenylquinoline Efflux Inhibitors in Combination with Macrolides against Mycobacterium smegmatis and Mycobacterium avium
D Machado, R Cannalire, S Santos Costa, G Manfroni, O Tabarrini, ...
ACS Infectious Diseases 1 (12), 593-603, 2015
252015
Broad spectrum anti-flavivirus pyridobenzothiazolones leading to less infective virions
R Cannalire, D Tarantino, G Piorkowski, T Carletti, S Massari, T Felicetti, ...
Antiviral Research 167, 6-12, 2019
242019
Broad‐spectrum flavivirus inhibitors: a medicinal chemistry point of view
T Felicetti, G Manfroni, V Cecchetti, R Cannalire
ChemMedChem 15 (24), 2391-2419, 2020
222020
Studies on 2-phenylquinoline Staphylococcus aureus NorA efflux pump inhibitors: New insights on the C-6 position
T Felicetti, R Cannalire, MG Nizi, O Tabarrini, S Massari, ML Barreca, ...
European Journal of Medicinal Chemistry 155, 428-433, 2018
212018
Discovery of potent p38α MAPK inhibitors through a funnel like workflow combining in silico screening and in vitro validation
A Astolfi, M Kudolo, J Brea, G Manni, G Manfroni, D Palazzotti, S Sabatini, ...
European Journal of Medicinal Chemistry 182, 111624, 2019
202019
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