A new, substituted palladacycle for ppm level Pd-catalyzed Suzuki–Miyaura cross couplings in water BS Takale, RR Thakore, S Handa, F Gallou, J Reilly, BH Lipshutz Chemical science 10 (38), 8825-8831, 2019 | 75 | 2019 |
N,C-Disubstituted Biarylpalladacycles as Precatalysts for ppm Pd-Catalyzed Cross Couplings in Water under Mild Conditions RR Thakore, BS Takale, F Gallou, J Reilly, BH Lipshutz ACS Catalysis 9 (12), 11647-11657, 2019 | 51 | 2019 |
A Sustainable 1-pot, 3-step synthesis of Boscalid using part per Million level Pd catalysis in water BS Takale, RR Thakore, R Mallarapu, F Gallou, BH Lipshutz Organic process research & development 24 (1), 101-105, 2019 | 50 | 2019 |
N 2 Phos–an easily made, highly effective ligand designed for ppm level Pd-catalyzed Suzuki–Miyaura cross couplings in water N Akporji, RR Thakore, M Cortes-Clerget, J Andersen, E Landstrom, ... Chemical science 11 (20), 5205-5212, 2020 | 42 | 2020 |
An environmentally responsible 3-pot, 5-step synthesis of the antitumor agent sonidegib using ppm levels of Pd catalysis in water BS Takale, RR Thakore, FY Kong, BH Lipshutz Green Chemistry 21 (23), 6258-6262, 2019 | 42 | 2019 |
Mild and Robust Stille Reactions in Water using Parts Per Million Levels of a Triphenylphosphine‐Based Palladacycle BS Takale, RR Thakore, G Casotti, X Li, F Gallou, BH Lipshutz Angewandte Chemie International Edition 60 (8), 4158-4163, 2021 | 41 | 2021 |
Chemoselective reductive aminations in aqueous nanoreactors using parts per million level Pd/C catalysis RR Thakore, BS Takale, G Casotti, ES Gao, HS Jin, BH Lipshutz Organic Letters 22 (16), 6324-6329, 2020 | 39 | 2020 |
Environmentally responsible, safe, and chemoselective catalytic hydrogenation of olefins: ppm level Pd catalysis in recyclable water at room temperature BS Takale, RR Thakore, ES Gao, F Gallou, BH Lipshutz Green Chemistry 22 (18), 6055-6061, 2020 | 37 | 2020 |
Sustainable and cost-effective Suzuki–Miyaura couplings toward the key biaryl subunits of Arylex and Rinskor active BS Takale, RR Thakore, NM Irvine, AD Schuitman, X Li, BH Lipshutz Organic Letters 22 (12), 4823-4827, 2020 | 31 | 2020 |
High turnover Pd/C catalyst for nitro group reductions in water. One-pot sequences and syntheses of pharmaceutical intermediates X Li, RR Thakore, BS Takale, F Gallou, BH Lipshutz Organic Letters 23 (20), 8114-8118, 2021 | 28 | 2021 |
“TPG-lite”: A new, simplified “designer” surfactant for general use in synthesis under micellar catalysis conditions in recyclable water RR Thakore, BS Takale, Y Hu, S Ramer, J Kostal, F Gallou, BH Lipshutz Tetrahedron 87, 132090, 2021 | 25 | 2021 |
Late‐stage Pd‐catalyzed Cyanations of Aryl/Heteroaryl Halides in Aqueous Micellar Media RR Thakore, BS Takale, V Singhania, F Gallou, BH Lipshutz ChemCatChem 13 (1), 212-216, 2021 | 25 | 2021 |
Recent Applications of Pd-Catalyzed Suzuki–Miyaura and Buchwald–Hartwig Couplings in Pharmaceutical Process Chemistry BS Takale, FY Kong, RR Thakore Organics 3 (1), 1-21, 2022 | 24 | 2022 |
Recent advances in Cu-catalyzed C (sp3)–Si and C (sp3)–B bond formation BS Takale, RR Thakore, E Etemadi-Davan, BH Lipshutz Beilstein Journal of Organic Chemistry 16 (1), 691-737, 2020 | 21 | 2020 |
Bisulfite addition compounds as substrates for reductive aminations in water X Li, KS Iyer, RR Thakore, DK Leahy, JD Bailey, BH Lipshutz Organic Letters 23 (18), 7205-7208, 2021 | 14 | 2021 |
Conformationally flexible C3-symmetric 1, 3-oxazoles as molecular scaffolds SR Shah, RR Thakore, TA Vyas, B Sridhar Synlett 27 (02), 294-300, 2016 | 14 | 2016 |
Environmentally responsible and cost-effective synthesis of the antimalarial drug pyronaridine JRA Kincaid, RD Kavthe, JC Caravez, BS Takale, RR Thakore, ... Organic Letters 24 (18), 3342-3346, 2022 | 12 | 2022 |
Sustainable routes to amines in recyclable water using ppm Pd catalysis RR Thakore, KS Iyer, BH Lipshutz Current Opinion in Green and Sustainable Chemistry 31, 100493, 2021 | 11 | 2021 |
Environmentally Benign Media: Water, AOS, and Water/Organic Solvent Azeotropic Mixtures RR Thakore, BS Takale | | 2021 |
Highly cost effective and sustainable ppm palladium pre-catalysts mediated cyanation and Stille couplings in water B Takale, B Lipshutz, RR Thakore American Chemical Society SciMeetings 1 (2), 2020 | | 2020 |