Dual-specificity tyrosine phosphorylation-regulated kinase 1A (DYRK1A) inhibitors as potential therapeutics DB Jarhad, KK Mashelkar, HR Kim, M Noh, LS Jeong Journal of medicinal chemistry 61 (22), 9791-9810, 2018 | 103 | 2018 |
Design, synthesis, and anti-RNA virus activity of 6′-fluorinated-aristeromycin analogues J Yoon, G Kim, DB Jarhad, HR Kim, YS Shin, S Qu, PK Sahu, HO Kim, ... Journal of medicinal chemistry 62 (13), 6346-6362, 2019 | 68 | 2019 |
Design, synthesis and anticancer activity of fluorocyclopentenyl-purines and–pyrimidines J Yoon, DB Jarhad, G Kim, A Nayak, LX Zhao, J Yu, HR Kim, JY Lee, ... European Journal of Medicinal Chemistry 155, 406-417, 2018 | 42 | 2018 |
6′-β-Fluoro-homoaristeromycin and 6′-fluoro-homoneplanocin A are potent inhibitors of chikungunya virus replication through their direct effect on viral nonstructural protein 1 K Kovacikova, BM Morren, A Tas, IC Albulescu, R van Rijswijk, DB Jarhad, ... Antimicrobial Agents and Chemotherapy 64 (4), 10.1128/aac. 02532-19, 2020 | 38 | 2020 |
Identification of 6′-β-fluoro-homoaristeromycin as a potent inhibitor of chikungunya virus replication YS Shin, DB Jarhad, MH Jang, K Kovacikova, G Kim, J Yoon, HR Kim, ... European Journal of Medicinal Chemistry 187, 111956, 2020 | 23 | 2020 |
Asymmetric synthesis of (−)-6′-β-fluoro-aristeromycin via stereoselective electrophilic fluorination G Kim, J Yoon, DB Jarhad, YS Shin, MS Majik, VA Mulamoottil, X Hou, ... Organic letters 19 (21), 5732-5735, 2017 | 18 | 2017 |
GPCR Agonist-to-Antagonist Conversion: Enabling the Design of Nucleoside Functional Switches for the A2A Adenosine Receptor A Shiriaeva, D Park, G Kim, Y Lee, X Hou, DB Jarhad, G Kim, J Yu, ... Journal of medicinal chemistry 65 (17), 11648-11657, 2022 | 17 | 2022 |
π4s + π2s Cycloaddition of Spiroepoxycyclohexa-2,4-dienone, Radical Cyclization, and Oxidation–Aldol–Oxidation Cascade: Synthesis of BCDE Ring of … DB Jarhad, V Singh The Journal of Organic Chemistry 81 (10), 4304-4309, 2016 | 14 | 2016 |
Antiproliferative and antimigration activities of fluoro-neplanocin a via inhibition of histone H3 methylation in triple-negative breast cancer WS Byun, WK Kim, J Yoon, DB Jarhad, LS Jeong, SK Lee Biomolecules 10 (4), 530, 2020 | 12 | 2020 |
Asymmetric Synthesis of 2′-C-Methyl-4′-selenonucleosides as Anti-Hepatitis C Virus Agents H Lee, DB Jarhad, J Yu, C Lee, LS Jeong The Journal of Organic Chemistry 84 (22), 14414-14426, 2019 | 12 | 2019 |
Molecular complexity and diversity from aromatics. Intramolecular cycloaddition of cyclohexa-2, 4-dienones and sigmatropic shift in excited state: a unified approach towards … TK Behera, DB Jarhad, SM Mobin, V Singh Tetrahedron 72 (35), 5377-5393, 2016 | 11 | 2016 |
Molecular diversity from aromatics. Cycloaddition of cyclohexa-2, 4-dienones, ring-closing metathesis and sigmatropic shifts: a general and stereoselective route to novel … V Singh, B Das, DB Jarhad, SM Mobin Tetrahedron 71 (4), 560-576, 2015 | 9 | 2015 |
An efficient synthesis of fluoro-neplanocin A analogs using electrophilic fluorination and palladium-catalyzed dehydrosilylation DB Jarhad, MH Jang, YS Shin, G Kim, HR Kim, YE Hyun, J Yoon, ... Organic Chemistry Frontiers 6 (7), 959-966, 2019 | 4 | 2019 |
Synthesis and anti-HIV activity of l-2′,3′-Dideoxy-4′-selenonucleosides (l-4′-Se-ddNs) J Yu, G Kim, DB Jarhad, HR Kim, LS Jeong Archives of pharmacal research 42, 780-789, 2019 | 3 | 2019 |
Correlation study between A3 adenosine receptor binding affinity and anti-renal interstitial fibrosis activity of truncated adenosine derivatives J Yu, G Kim, DB Jarhad, HW Lee, J Lee, CW Park, H Ha, LS Jeong Archives of pharmacal research 42, 773-779, 2019 | 3 | 2019 |
Structure–Activity Relationship of Truncated 2,8-Disubstituted-Adenosine Derivatives as Dual A2A/A3 Adenosine Receptor Antagonists and Their Cancer … G Kim, X Hou, WS Byun, G Kim, DB Jarhad, G Lee, YE Hyun, J Yu, ... Journal of Medicinal Chemistry 66 (17), 12249-12265, 2023 | 2 | 2023 |
Synthesis of enantiomerically pure pyrimidine ribonucleosides locked in the south conformation YE Hyun, DB Jarhad, M Kim, A Yang, G Kim, HR Kim, LS Jeong Organic Letters 24 (50), 9281-9284, 2022 | 2 | 2022 |
Catalyst-controlled regioselective Sonogashira coupling of 9-substituted-6-chloro-2, 8-diiodopurines G Kim, G Lee, G Kim, Y Seo, DB Jarhad, LS Jeong Organic Chemistry Frontiers 9 (20), 5536-5543, 2022 | 2 | 2022 |
4′‐Selenonucleosides: Regio‐and Stereoselective Synthesis of Novel Ribavirin and Acadesine Analogs as Anti‐Hepatitis C Virus (HCV) Agents H Lee, DB Jarhad, A Lee, C Lee, LS Jeong Asian Journal of Organic Chemistry 10 (11), 2993-2999, 2021 | 2 | 2021 |
Asymmetric Synthesis of Fluoro‐MLN4924 as a Selective NEDD8‐Activating Enzyme (NAE) Inhibitor HR Kim, DB Jarhad, PK Sahu, K Sung, D An, YE Hyun, J Yu, LS Jeong Asian Journal of Organic Chemistry 8 (9), 1641-1647, 2019 | 2 | 2019 |