| Comprehensive in vitro characterization of PD-L1 small molecule inhibitors A Ganesan, M Ahmed, I Okoye, E Arutyunova, D Babu, WL Turnbull, ... Scientific reports 9 (1), 12392, 2019 | 122 | 2019 |
| A study directed to the asymmetric synthesis of the antineoplastic macrolide acutiphycin under enantioselective acyclic stereoselection based on chiral oxazaborolidinone … S Kiyooka, MA Hena The Journal of Organic Chemistry 64 (15), 5511-5523, 1999 | 103 | 1999 |
| Peptidomimetic α-acyloxymethylketone warheads with six-membered lactam P1 glutamine mimic: SARS-CoV-2 3CL protease inhibition, coronavirus antiviral activity, and in vitro … B Bai, A Belovodskiy, M Hena, AS Kandadai, MA Joyce, HA Saffran, ... Journal of Medicinal Chemistry 65 (4), 2905-2925, 2021 | 82 | 2021 |
| Catalyst control in a chiral borane-mediated aldol reaction. Both syn-and anti-aldols in almost optically pure state obtained from one racemic aldehyde S Kiyooka, H Kira, MA Hena Tetrahedron letters 37 (15), 2597-2600, 1996 | 51 | 1996 |
| Peptidomimetic nitrile warheads as SARS-CoV-2 3CL protease inhibitors B Bai, E Arutyunova, MB Khan, J Lu, MA Joyce, HA Saffran, JA Shields, ... RSC medicinal chemistry 12 (10), 1722-1730, 2021 | 45 | 2021 |
| Enantioselective acyclic stereoselection under catalyst control. 2.1 Asymmetric synthesis of syn-and anti-1, 3-diols incorporating an acetate equivalent by the chiral … S Kiyooka, T Yamaguchi, H Maeda, H Kira, MA Hena, M Horiike Tetrahedron letters 38 (20), 3553-3556, 1997 | 43 | 1997 |
| A chiral oxazaborolidinone-promoted aldol reaction with a silyl ketene acetal from ethyl 1, 3-dithiolane-2-carboxylate. Synthesis of acetate aldols in high enantiomeric purity S Kiyooka, MA Hena Tetrahedron: Asymmetry 7 (8), 2181-2184, 1996 | 41 | 1996 |
| An effective extension of the polyacetate chain in the polyene macrolide antibiotic filipin III, based on chiral oxazaborolidinone-promoted asymmetric aldol reactions S Kiyooka, MA Hena, T Yabukami, K Murai, F Goto Tetrahedron Letters 41 (39), 7511-7516, 2000 | 32 | 2000 |
| Toward a practical synthesis of acutiphycin. Highly stereoselective synthesis of C10-epi seco acid derivative via reaction paths shortened by using a series of chiral … MA Hena, CS Kim, M Horiike, S Kiyooka Tetrahedron letters 40 (6), 1161-1164, 1999 | 28 | 1999 |
| A short and efficient synthesis of N-Cbz-galantinic acid under promoter control on enantioselective acyclic stereoselection based on chiral oxazaborolidinone-promoted aldol … S Kiyooka, K Goh, Y Nakamura, H Takesue, MA Hena Tetrahedron Letters 41 (34), 6599-6603, 2000 | 26 | 2000 |
| Novel diastereo-and enantioselectivities in the chiral oxazaborolidinone-promoted asymmetric aldol reaction of highly hindered aldehydes having a quaternary carbon at α … S Kiyooka, H Maeda, MA Hena, M Uchida, CS Kim, M Horiike Tetrahedron letters 39 (45), 8287-8290, 1998 | 24 | 1998 |
| Highly enantioselective synthesis of syn-and anti-propionate aldols without diastereoselection in the chiral oxazaborolidinone-promoted aldol reaction with a silyl ketene … MA Hena, S Terauchi, CS Kim, M Horiike, S Kiyooka Tetrahedron: Asymmetry 9 (11), 1883-1890, 1998 | 23 | 1998 |
| A practical synthesis of essentially enantiopure syn-propionate aldols using a chiral oxazaborolidinone-promoted asymmetric aldol reaction coupled with radical reduction S Kiyooka, KA Shahid, MA Hena Tetrahedron letters 40 (35), 6447-6449, 1999 | 21 | 1999 |
| The discovery of glycine and related amino acid-based factor Xa inhibitors JT Kohrt, KJ Filipski, WL Cody, CF Bigge, F La, K Welch, T Dahring, ... Bioorganic & medicinal chemistry 14 (13), 4379-4392, 2006 | 20 | 2006 |
| Enantioselective synthesis of a key intermediate aldehyde toward the polyene macrolide filipin III, based on a chiral oxazaborolidinone-promoted asymmetric aldol reaction S Kiyooka, MA Hena, F Goto Tetrahedron: Asymmetry 10 (15), 2871-2879, 1999 | 17 | 1999 |
| Discovery of a series of 2-(1H-pyrazol-1-yl) pyridines as ALK5 inhibitors with potential utility in the prevention of dermal scarring ML Boys, F Bian, JB Kramer, CL Chio, XD Ren, H Chen, SD Barrett, ... Bioorganic & medicinal chemistry letters 22 (10), 3392-3397, 2012 | 16 | 2012 |
| Amidine substituted β-lactam compounds, their preparation and use as antibacterial agents B Klenke, I Wiegand, G Schiffer, H Broetz-Oesterhelt, SN Maiti, J Khan, ... US Patent 9,556,165, 2017 | 12* | 2017 |
| (1R, 2S)-4-(2-Cyano-cyclohexyl-oxy)-2-trifluoromethyl-benzonitrile, a potent androgen receptor antagonist for stimulating hair growth and reducing sebum production LY Hu, D Du, J Hoffman, Y Smith, V Fedij, C Kostlan, TR Johnson, ... Bioorganic & medicinal chemistry letters 17 (21), 5983-5988, 2007 | 12 | 2007 |
| Rna virus inhibitor compounds and uses thereof JA Nieman, MJ Lemieux, DL Tyrrell, M Hena, AS Kandadai, ... US Patent App. 17/950,785, 2023 | 1 | 2023 |
| Enantioselective Acyclic Stereoselection under Catalyst (Promoter) Control. Part 5. Towards a Practical Synthesis of Acutiphycin. Highly Stereoselective Synthesis of C10‐epi … MA Hena, CS Kim, M Horiike, S Kiyooka ChemInform 30 (21), no-no, 1999 | 1 | 1999 |
