| Anticancer activity of stilbene‐based derivatives B De Filippis, A Ammazzalorso, M Fantacuzzi, L Giampietro, C Maccallini, ... ChemMedChem 12 (8), 558-570, 2017 | 134 | 2017 |
| N‐acylsulfonamides: Synthetic routes and biological potential in medicinal chemistry A Ammazzalorso, B De Filippis, L Giampietro, R Amoroso Chemical biology & drug design 90 (6), 1094-1105, 2017 | 75 | 2017 |
| Synthesis, biological evaluation, and docking study of indole aryl sulfonamides as aromatase inhibitors M Fantacuzzi, B De Filippis, M Gallorini, A Ammazzalorso, L Giampietro, ... European journal of medicinal chemistry 185, 111815, 2020 | 54 | 2020 |
| Novel approaches to the discovery of selective human monoamine oxidase-B inhibitors: is there room for improvement? P Guglielmi, S Carradori, A Ammazzalorso, D Secci Expert Opinion on Drug Discovery 14 (10), 995-1035, 2019 | 48 | 2019 |
| 2-substituted benzothiazoles as antiproliferative agents: Novel insights on structure-activity relationships A Ammazzalorso, S Carradori, R Amoroso, IF Fernández European Journal of Medicinal Chemistry 207, 112762, 2020 | 46 | 2020 |
| Benzothiazole-based N-(phenylsulfonyl)amides as a novel family of PPARα antagonists A Ammazzalorso, A Giancristofaro, A D’Angelo, B De Filippis, ... Bioorganic & medicinal chemistry letters 21 (16), 4869-4872, 2011 | 43 | 2011 |
| Stilbene derivatives as new perspective in antifungal medicinal chemistry B De Filippis, A Ammazzalorso, R Amoroso, L Giampietro Drug Development Research 80 (3), 285-293, 2019 | 42 | 2019 |
| Structural development studies of PPARs ligands based on tyrosine scaffold B De Filippis, P Linciano, A Ammazzalorso, C Di Giovanni, M Fantacuzzi, ... European Journal of Medicinal Chemistry 89, 817-825, 2015 | 39 | 2015 |
| Synthesis, biological evaluation, and docking studies of N-substituted acetamidines as selective inhibitors of inducible nitric oxide synthase C Maccallini, A Patruno, N Besker, JI Alì, A Ammazzalorso, B De Filippis, ... Journal of medicinal chemistry 52 (5), 1481-1485, 2009 | 37 | 2009 |
| Multitarget PPARγ agonists as innovative modulators of the metabolic syndrome A Ammazzalorso, C Maccallini, P Amoia, R Amoroso European Journal of Medicinal Chemistry 173, 261-273, 2019 | 36 | 2019 |
| Synthesis and biological characterization of 3-(imidazol-1-ylmethyl) piperidine sulfonamides as aromatase inhibitors M Di Matteo, A Ammazzalorso, F Andreoli, I Caffa, B De Filippis, ... Bioorganic & Medicinal Chemistry Letters 26 (13), 3192-3194, 2016 | 36 | 2016 |
| Different binding and recognition modes of GL479, a dual agonist of Peroxisome Proliferator-Activated Receptor α/γ JC dos Santos, A Bernardes, L Giampietro, A Ammazzalorso, ... Journal of Structural Biology 191 (3), 332-340, 2015 | 36 | 2015 |
| Synthesis and structure–activity relationships of fibrate-based analogues inside PPARs L Giampietro, A D’Angelo, A Giancristofaro, A Ammazzalorso, ... Bioorganic & medicinal chemistry letters 22 (24), 7662-7666, 2012 | 35 | 2012 |
| Discovery of gemfibrozil analogues that activate PPARα and enhance the expression of gene CPT1A involved in fatty acids catabolism B De Filippis, A Giancristofaro, A Ammazzalorso, A D’Angelo, ... European journal of medicinal chemistry 46 (10), 5218-5224, 2011 | 35 | 2011 |
| Development of CDK4/6 inhibitors: a five years update A Ammazzalorso, M Agamennone, B De Filippis, M Fantacuzzi Molecules 26 (5), 1488, 2021 | 33 | 2021 |
| Effects of PPARα inhibition in head and neck paraganglioma cells R Florio, L De Lellis, V di Giacomo, MC Di Marcantonio, L Cristiano, ... PLoS One 12 (6), e0178995, 2017 | 33 | 2017 |
| Design, synthesis and biological evaluation of imidazole and triazole-based carbamates as novel aromatase inhibitors A Ammazzalorso, M Gallorini, M Fantacuzzi, N Gambacorta, B De Filippis, ... European Journal of Medicinal Chemistry 211, 113115, 2021 | 32 | 2021 |
| Blocking the peroxisome proliferator‐activated receptor (PPAR): an overview A Ammazzalorso, B De Filippis, L Giampietro, R Amoroso ChemMedChem 8 (10), 1609-1616, 2013 | 32 | 2013 |
| N-Substituted acetamidines and 2-methylimidazole derivatives as selective inhibitors of neuronal nitric oxide synthase C Maccallini, A Patruno, F Lannutti, A Ammazzalorso, B De Filippis, ... Bioorganic & medicinal chemistry letters 20 (22), 6495-6499, 2010 | 31 | 2010 |
| Indazole, pyrazole, and oxazole derivatives targeting nitric oxide synthases and carbonic anhydrases C Maccallini, M Di Matteo, D Vullo, A Ammazzalorso, S Carradori, ... ChemMedChem 11 (16), 1695-1699, 2016 | 30 | 2016 |
