| Construction of Natural-Product-Like Cyclophane-Braced Peptide Macrocycles via sp3 C–H Arylation B Li, X Li, B Han, Z Chen, X Zhang, G He, G Chen Journal of the American Chemical Society 141 (23), 9401-9407, 2019 | 120 | 2019 |
| Postassembly modifications of peptides via metal-catalyzed C–H functionalization HR Tong, B Li, G Li, G He, G Chen CCS Chemistry 3 (3), 1797-1820, 2021 | 80 | 2021 |
| Streamlined construction of peptide macrocycles via palladium-catalyzed intramolecular S-arylation in solution and on DNA P Yang, X Wang, B Li, Y Yang, J Yue, Y Suo, H Tong, G He, X Lu, G Chen Chemical Science 12 (16), 5804-5810, 2021 | 42 | 2021 |
| Construction of Cyclophane-Braced Peptide Macrocycles via Palladium-Catalyzed Picolinamide-Directed Intramolecular C(sp2)–H Arylation B Han, B Li, L Qi, P Yang, G He, G Chen Organic Letters 22 (17), 6879-6883, 2020 | 39 | 2020 |
| Cooperative stapling of native peptides at lysine and tyrosine or arginine with formaldehyde B Li, H Tang, A Turlik, Z Wan, XS Xue, L Li, X Yang, J Li, G He, KN Houk, ... Angewandte Chemie International Edition 60 (12), 6646-6652, 2021 | 33 | 2021 |
| Synthesis of Cyclophane-Braced Peptide Macrocycles via Palladium-Catalyzed Intramolecular C(sp3)–H Arylation of N-Methyl Alanine at C-Termini X Li, L Qi, B Li, Z Zhao, G He, G Chen Organic Letters 22 (15), 6209-6213, 2020 | 31 | 2020 |
| Extendable stapling of unprotected peptides by crosslinking two amines with o-phthalaldehyde B Li, L Wang, X Chen, X Chu, H Tang, J Zhang, G He, L Li, G Chen Nature Communications 13 (1), 311, 2022 | 29 | 2022 |
| Construction of complex macromulticyclic peptides via stitching with formaldehyde and guanidine B Li, Z Wan, H Zheng, S Cai, HW Tian, H Tang, X Chu, G He, DS Guo, ... Journal of the American Chemical Society 144 (22), 10080-10090, 2022 | 18 | 2022 |
| Improved synthesis of unnatural amino acids for peptide stapling B Li, J Zhang, Y Xu, X Yang, L Li Tetrahedron Letters 58 (24), 2374-2377, 2017 | 18 | 2017 |
| A rapid and sensitive method for chiroptical sensing of α-amino acids via click-like labeling with o-phthalaldehyde and p-toluenethiol B Li, J Zhang, L Li, G Chen Chemical Science 12 (7), 2504-2508, 2021 | 17 | 2021 |
| Construction of peptide macrocycles via palladium-catalyzed multiple S-arylation: an effective strategy to expand the structural diversity of cross-linkers X Chu, L Shen, B Li, P Yang, C Du, X Wang, G He, S Messaoudi, G Chen Organic Letters 23 (20), 8001-8006, 2021 | 15 | 2021 |
| Construction of peptide macrocycles via radical-mediated intramolecular C–H alkylations X Hu, X Chen, B Li, G He, G Chen Organic Letters 23 (3), 716-721, 2021 | 15 | 2021 |
| Bioconjugation via Hetero‐Selective Clamping of Two Different Amines with ortho‐Phthalaldehyde X Chu, B Li, HY Liu, X Sun, X Yang, G He, C Zhou, W Xuan, SL Liu, ... Angewandte Chemie 135 (2), e202212199, 2023 | 12 | 2023 |
| Teraryl braces in macrocycles: synthesis and conformational landscape remodeling of peptides P Yang, MJ Širvinskas, B Li, NW Heller, H Rong, G He, AK Yudin, ... Journal of the American Chemical Society 145 (25), 13968-13978, 2023 | 10 | 2023 |
| De novo development of small cyclic peptides that are orally bioavailable ML Merz, S Habeshian, B Li, JAGL David, AL Nielsen, X Ji, K Il Khwildy, ... Nature Chemical Biology 20 (5), 624-633, 2024 | 6 | 2024 |
| Palladium‐Catalyzed Methionine‐Facilitated β and γ C(sp3)–H Arylation of N‐Terminal Aliphatic Amino Acids of Peptides X Chen, B Li, H Tong, L Qi, G He, G Chen Chinese Journal of Chemistry 40 (21), 2502-2506, 2022 | 6 | 2022 |
| Formaldehyde-Mediated Hydride Liberation of Alkylamines for Intermolecular Reactions in Hexafluoroisopropanol S Cai, H Tang, B Li, Y Shao, D Zhang, H Zheng, T Qiao, X Chu, G He, ... Journal of the American Chemical Society 146 (9), 5952-5963, 2024 | 4 | 2024 |
| Ring-locking strategy facilitating determination of absolute optical purity of 2-amino-1-butanol by reverse-phase high-performance liquid chromatography B Li, J Zhang, BB Yang, L Li, XX Yang RSC advances 7 (72), 45714-45720, 2017 | 4 | 2017 |
| Solid Phase Synthesis of Thioether‐linked Peptide Macrocycles via Palladium‐Catalyzed Intramolecular S‐Arylation and S‐Alkenylation P Yang, C Zhang, B Li, G He, G Chen Asian Journal of Organic Chemistry 10 (11), 2888-2891, 2021 | 3 | 2021 |
| Research progress in the synthesis and bioactivity of stapled peptide B LI, X YANG, L LI Acta Pharmaceutica Sinica, 685-698, 2017 | 2 | 2017 |
