Mol* Viewer: modern web app for 3D visualization and analysis of large biomolecular structures D Sehnal, S Bittrich, M Deshpande, R Svobodová, K Berka, V Bazgier, ... Nucleic acids research 49 (W1), W431-W437, 2021 | 765 | 2021 |
MOLEonline: a web-based tool for analyzing channels, tunnels and pores (2018 update) L Pravda, D Sehnal, D Toušek, V Navrátilová, V Bazgier, K Berka, ... Nucleic acids research 46 (W1), W368-W373, 2018 | 256 | 2018 |
Membrane-attached mammalian cytochromes P450: An overview of the membrane's effects on structure, drug binding, and interactions with redox partners M Šrejber, V Navrátilová, M Paloncýová, V Bazgier, K Berka, ... Journal of inorganic biochemistry 183, 117-136, 2018 | 171 | 2018 |
Novel N-substituted indole Schiff bases as dual inhibitors of cyclooxygenase-2 and 5-lipoxygenase enzymes: Synthesis, biological activities in vitro and docking study PF Lamie, WAM Ali, V Bazgier, L Rárová European journal of medicinal chemistry 123, 803-813, 2016 | 95 | 2016 |
Novel thidiazuron-derived inhibitors of cytokinin oxidase/dehydrogenase J Nisler, D Kopečný, R Končitíková, M Zatloukal, V Bazgier, K Berka, ... Plant Molecular Biology 92, 235-248, 2016 | 59 | 2016 |
A novel series of highly potent 2, 6, 9-trisubstituted purine cyclin-dependent kinase inhibitors T Gucky, R Jorda, M Zatloukal, V Bazgier, K Berka, E Reznickova, T Béres, ... Journal of medicinal chemistry 56 (15), 6234-6247, 2013 | 59 | 2013 |
Antiallergic effects of pigments isolated from green sea urchin (Strongylocentrotus droebachiensis) shells ON Pozharitskaya, AN Shikov, MN Makarova, SA Ivanova, VM Kosman, ... Planta medica 79 (18), 1698-1704, 2013 | 55 | 2013 |
Synthesis, biological evaluation and molecular modeling of a novel series of 7-azaindole based tri-heterocyclic compounds as potent CDK2/Cyclin E inhibitors CB Baltus, R Jorda, C Marot, K Berka, V Bazgier, V Kryštof, G Prié, ... European journal of medicinal chemistry 108, 701-719, 2016 | 48 | 2016 |
Discovery of N2-(4-Amino-cyclohexyl)-9-cyclopentyl-N6-(4-morpholin-4-ylmethyl-phenyl)-9H-purine-2,6-diamine as a Potent FLT3 Kinase Inhibitor for Acute … T Gucky, E Reznickova, T Radošová Muchová, R Jorda, Z Klejova, ... Journal of Medicinal Chemistry 61 (9), 3855-3869, 2018 | 42 | 2018 |
Acetylated deoxycholic (DCA) and cholic (CA) acids are potent ligands of pregnane X (PXR) receptor A Carazo, L Hyrsova, J Dusek, H Chodounska, A Horvatova, K Berka, ... Toxicology Letters 265, 86-96, 2017 | 40 | 2017 |
Synthesis and kinase inhibitory activity of new sulfonamide derivatives of pyrazolo [4, 3-e][1, 2, 4] triazines M Mojzych, V Šubertová, A Bielawska, K Bielawski, V Bazgier, K Berka, ... European Journal of Medicinal Chemistry 78, 217-224, 2014 | 38 | 2014 |
Design, synthesis and biological activities of new brassinosteroid analogues with a phenyl group in the side chain M Kvasnica, J Oklestkova, V Bazgier, L Rárová, P Korinkova, J Mikulík, ... Organic & Biomolecular Chemistry 14 (37), 8691-8701, 2016 | 26 | 2016 |
Synthesis of novel galeterone derivatives and evaluation of their in vitro activity against prostate cancer cell lines R Jorda, E Řezníčková, U Kiełczewska, J Maj, JW Morzycki, ... European journal of medicinal chemistry 179, 483-492, 2019 | 25 | 2019 |
Biological activities of new monohydroxylated brassinosteroid analogues with a carboxylic group in the side chain M Kvasnica, J Oklestkova, V Bazgier, L Rarova, K Berka, M Strnad Steroids 85, 58-64, 2014 | 25 | 2014 |
Novel thiazolidinedione-hydroxamates as inhibitors of Mycobacterium tuberculosis virulence factor Zmp1 V Šlachtová, M Šebela, E Torfs, L Oorts, D Cappoen, K Berka, V Bazgier, ... European Journal of Medicinal Chemistry 185, 111812, 2020 | 20 | 2020 |
Characterization of a Pyrazolo[4,3‐d]pyrimidine Inhibitor of Cyclin‐Dependent Kinases 2 and 5 and Aurora A With Pro‐Apoptotic and Anti‐Angiogenic Activity In Vitro E Řezníčková, S Weitensteiner, L Havlíček, R Jorda, T Gucký, K Berka, ... Chemical Biology & Drug Design 86 (6), 1528-1540, 2015 | 20 | 2015 |
Synthesis of dihydrotestosterone derivatives modified in the A-ring with (hetero) arylidene, pyrazolo [1, 5-a] pyrimidine and triazolo [1, 5-a] pyrimidine moieties and their … MA Kiss, M Peřina, V Bazgier, NV May, Á Baji, R Jorda, É Frank The Journal of Steroid Biochemistry and Molecular Biology 211, 105904, 2021 | 18 | 2021 |
MolMeDB: molecules on membranes database J Juračka, M Šrejber, M Melíková, V Bazgier, K Berka Database 2019, baz078, 2019 | 16 | 2019 |
Synthesis of novel aryl brassinosteroids through alkene cross-metathesis and preliminary biological study P Korinkova, V Bazgier, J Oklestkova, L Rarova, M Strnad, M Kvasnica Steroids 127, 46-55, 2017 | 15 | 2017 |
2, 6, 9-Trisubstituted purines as CRK3 kinase inhibitors with antileishmanial activity in vitro E Řezníčková, A Popa, T Gucký, M Zatloukal, L Havlíček, V Bazgier, ... Bioorganic & medicinal chemistry letters 25 (11), 2298-2301, 2015 | 14 | 2015 |