| SuFEx click chemistry enabled late-stage drug functionalization Z Liu, J Li, S Li, G Li, KB Sharpless, P Wu Journal of the American Chemical Society 140 (8), 2919-2925, 2018 | 242 | 2018 |
| Palladium-catalyzed intramolecular asymmetric C–H functionalization/cyclization reaction of metallocenes: an efficient approach toward the synthesis of planar chiral … R Deng, Y Huang, X Ma, G Li, R Zhu, B Wang, YB Kang, Z Gu Journal of the American Chemical Society 136 (12), 4472-4475, 2014 | 197 | 2014 |
| Ligand-Promoted meta-C–H Amination and Alkynylation P Wang, GC Li, P Jain, ME Farmer, J He, PX Shen, JQ Yu Journal of the American Chemical Society 138 (42), 14092-14099, 2016 | 179 | 2016 |
| SuFEx-enabled, agnostic discovery of covalent inhibitors of human neutrophil elastase Q Zheng, JL Woehl, S Kitamura, D Santos-Martins, CJ Smedley, G Li, ... Proceedings of the National Academy of Sciences 116 (38), 18808-18814, 2019 | 156 | 2019 |
| Ligand-Enabled Stereoselective β-C(sp3)–H Fluorination: Synthesis of Unnatural Enantiopure anti-β-Fluoro-α-amino Acids RY Zhu, K Tanaka, GC Li, J He, HY Fu, SH Li, JQ Yu Journal of the American Chemical Society 137 (22), 7067-7070, 2015 | 156 | 2015 |
| Ligand‐enabled β‐C–H arylation of α‐amino acids without installing exogenous directing groups G Chen, Z Zhuang, GC Li, TG Saint‐Denis, Y Hsiao, CL Joe, JQ Yu Angewandte Chemie 129 (6), 1528-1531, 2017 | 126 | 2017 |
| Pd-Catalyzed Chemoselective Catellani Ortho-Arylation of Iodopyrroles: Rapid Total Synthesis of Rhazinal X Sui, R Zhu, G Li, X Ma, Z Gu Journal of the American Chemical Society 135 (25), 9318-9321, 2013 | 112 | 2013 |
| Diversity oriented clicking (DOC): divergent synthesis of SuFExable pharmacophores from 2‐substituted‐alkynyl‐1‐sulfonyl fluoride (SASF) hubs CJ Smedley, G Li, AS Barrow, TL Gialelis, MC Giel, A Ottonello, Y Cheng, ... Angewandte Chemie 132 (30), 12560-12569, 2020 | 94 | 2020 |
| Using sulfuramidimidoyl fluorides that undergo sulfur(vi) fluoride exchange for inverse drug discovery GJ Brighty, RC Botham, S Li, L Nelson, DE Mortenson, G Li, C Morisseau, ... Nature chemistry 12 (10), 906-913, 2020 | 93 | 2020 |
| SuFExable polymers with helical structures derived from thionyl tetrafluoride S Li, G Li, B Gao, SP Pujari, X Chen, H Kim, F Zhou, LM Klivansky, Y Liu, ... Nature chemistry 13 (9), 858-867, 2021 | 90 | 2021 |
| Ligand‐Enabled Auxiliary‐Free meta‐C−H Arylation of Phenylacetic Acids GC Li, P Wang, ME Farmer, JQ Yu Angewandte Chemie 129 (24), 6978-6981, 2017 | 71 | 2017 |
| Diversity oriented clicking delivers β-substituted alkenyl sulfonyl fluorides as covalent human neutrophil elastase inhibitors Y Cheng, G Li, CJ Smedley, MC Giel, S Kitamura, JL Woehl, G Bianco, ... Proceedings of the National Academy of Sciences 119 (37), e2208540119, 2022 | 17 | 2022 |
| Identification of clickable HIV-1 capsid-targeting probes for viral replication inhibition WM McFadden, MC Casey-Moore, GAL Bare, KA Kirby, X Wen, G Li, ... Cell Chemical Biology 31 (3), 477-486. e7, 2024 | 1 | 2024 |
| Synthesis and structure–activity relationships of aryl fluorosulfate-based inhibitors as novel antitubercular agents B Yang, P Sukheja, B Qin, G Li, GAL Bare, A Cascioferro, MS Love, ... Bioorganic & Medicinal Chemistry Letters 98, 129596, 2024 | 1 | 2024 |
