Probing the biology of natural products: molecular editing by diverted total synthesis AM Szpilman, EM Carreira Angewandte Chemie International Edition 49 (50), 9592-9628, 2010 | 193 | 2010 |
Synthesis and biological evaluation of amphotericin B derivatives AA Volmer, AM Szpilman, EM Carreira Natural product reports 27 (9), 1329-1349, 2010 | 158 | 2010 |
Cycloaddition reactions AM Szpilman, EM Carreira Silver in Organic Chemistry, 43-82, 2010 | 142* | 2010 |
Enolonium species—umpoled enolates S Arava, JN Kumar, S Maksymenko, MA Iron, KN Parida, P Fristrup, ... Angewandte Chemie 129 (10), 2643-2647, 2017 | 96 | 2017 |
A short synthesis and biological evaluation of potent and nontoxic antimalarial bridged bicyclic β-sulfonyl-endoperoxides MD Bachi, EE Korshin, R Hoos, AM Szpilman, P Ploypradith, S Xie, ... Journal of medicinal chemistry 46 (12), 2516-2533, 2003 | 85 | 2003 |
Total syntheses of yingzhaosu A and of its C (14)-epimer including the first evaluation of their antimalarial and cytotoxic activities AM Szpilman, EE Korshin, H Rozenberg, MD Bachi The Journal of Organic Chemistry 70 (9), 3618-3632, 2005 | 67 | 2005 |
Synthesis of 35‐Deoxy Amphotericin B Methyl Ester: A Strategy for Molecular Editing AM Szpilman, DM Cereghetti, NR Wurtz, JM Manthorpe, EM Carreira Angewandte Chemie International Edition 47 (23), 4335-4338, 2008 | 66 | 2008 |
Oxidative Umpolung α-Alkylation of Ketones OS Shneider, E Pisarevsky, P Fristrup, AM Szpilman Organic letters 17 (2), 282-285, 2015 | 58 | 2015 |
An efficient synthesis of bridged-bicyclic peroxides structurally related to antimalarial yingzhaosu A based on radical co-oxygenation of thiols and monoterpenes EE Korshin, R Hoos, AM Szpilman, L Konstantinovski, GH Posner, ... Tetrahedron 58 (12), 2449-2469, 2002 | 58 | 2002 |
Synthesis and Biophysical Studies on 35‐Deoxy Amphotericin B Methyl Ester AM Szpilman, DM Cereghetti, JM Manthorpe, NR Wurtz, EM Carreira Chemistry–A European Journal 15 (29), 7117-7128, 2009 | 56 | 2009 |
Mechanism of the Copper/TEMPO‐Catalyzed Aerobic Oxidation of Alcohols MA Iron, AM Szpilman Chemistry–A European Journal 23 (6), 1368-1378, 2017 | 55 | 2017 |
Transition-metal-free intermolecular α-arylation of ketones via enolonium species S Maksymenko, KN Parida, GK Pathe, AA More, YB Lipisa, AM Szpilman Organic letters 19 (23), 6312-6315, 2017 | 54 | 2017 |
Untersuchung der Biologie von Naturstoffen: systematische Strukturvariation durch umgelenkte Totalsynthese AM Szpilman, EM Carreira Angewandte Chemie 122 (50), 9786-9823, 2010 | 50 | 2010 |
Synthesis and biological studies of 35‐deoxy amphotericin B methyl ester AM Szpilman, JM Manthorpe, EM Carreira Angewandte Chemie International Edition 47 (23), 4339-4342, 2008 | 50 | 2008 |
Iron (II)-induced degradation of antimalarial β-sulfonyl endoperoxides. Evidence for the generation of potentially cytotoxic carbocations AM Szpilman, EE Korshin, R Hoos, GH Posner, MD Bachi The Journal of Organic Chemistry 66 (20), 6531-6540, 2001 | 49 | 2001 |
Organocatalytic oxidation of aldehydes to mixed anhydrides H Toledo, E Pisarevsky, A Abramovich, AM Szpilman Chemical Communications 49 (39), 4367-4369, 2013 | 48 | 2013 |
Novel Water-Soluble Amphotericin B-PEG Conjugates with Low Toxicity and Potent in Vivo Efficacy A Halperin, Y Shadkchan, E Pisarevsky, AM Szpilman, H Sandovsky, ... Journal of Medicinal Chemistry 59 (3), 1197-1206, 2016 | 47 | 2016 |
α-N-Heteroarylation and α-Azidation of Ketones via Enolonium Species AA More, GK Pathe, KN Parida, S Maksymenko, YB Lipisa, AM Szpilman The Journal of organic chemistry 83 (4), 2442-2447, 2018 | 41 | 2018 |
Design concept for α-hydrogen-substituted nitroxides M Amar, S Bar, MA Iron, H Toledo, B Tumanskii, LJW Shimon, ... Nature Communications 6, 6070, 2015 | 41 | 2015 |
Organocatalytic oxidative dimerization of alcohols to esters A Abramovich, H Toledo, E Pisarevsky, AM Szpilman Synlett 23 (15), 2261-2265, 2012 | 38 | 2012 |