Inhibition of β-Amyloid aggregation Through a Designed β-hairpin Peptide A Jha, M Ganesh Kumar, HN Gopi, KM Paknikar Langmuir, 2017 | 45 | 2017 |
Thiol-to-amine cyclization reaction enables screening of large libraries of macrocyclic compounds and the generation of sub-kilodalton ligands AACH S. S. Kale,* M. Bergeron-Brlek,* Y. Wu,* M. G. Kumar,* M. V. Pham, J ... Science Advances 5 (8), eaaw2851, 2019 | 41 | 2019 |
Synthesis of α, β-unsaturated γ-amino esters with unprecedented high (E)-stereoselectivity and their conformational analysis in peptides SM Mali, A Bandyopadhyay, SV Jadhav, M Ganesh Kumar, HN Gopi Organic & biomolecular chemistry 9 (19), 6566-6574, 2011 | 39 | 2011 |
Non‐classical Helices with cis Carbon–Carbon Double Bonds in the Backbone: Structural Features of α,γ‐Hybrid Peptide Foldamers M Ganesh Kumar, VJ Thombare, MM Katariya, K Veeresh, KMP Raja, ... Angewandte Chemie 128 (27), 7978-7982, 2016 | 32 | 2016 |
Exploring β-hydroxy γ-amino acids (statines) in the design of hybrid peptide foldamers A Bandyopadhyay, A Malik, M Ganesh Kumar, HN Gopi Organic letters 16 (1), 294-297, 2013 | 26 | 2013 |
HBTU mediated 1-hydroxybenzotriazole (HOBt) conjugate addition: synthesis and stereochemical analysis of β-benzotriazole N-oxide substituted γ-amino acids and hybrid peptides SM Mali, M Ganesh Kumar, MM Katariya, HN Gopi Organic & biomolecular chemistry 12 (42), 8462-8472, 2014 | 25 | 2014 |
Synthesis and direct assay of large macrocycle diversities by combinatorial late-stage modification at picomole scale S Habeshian, ML Merz, G Sangouard, GK Mothukuri, M Schüttel, ... Nature Communications 13 (1), 3823, 2022 | 22 | 2022 |
Design of stable β-hairpin mimetics through backbone disulfide bonds M Ganesh Kumar, SM Mali, KMP Raja, HN Gopi Organic letters 17 (2), 230-233, 2015 | 16 | 2015 |
Macrocycle synthesis strategy based on step-wise “adding and reacting” three components enables screening of large combinatorial libraries GK Mothukuri, SS Kale, CL Stenbratt, A Zorzi, J Vesin, JB Chapalay, ... Chemical Science 11 (30), 7858-7863, 2020 | 14 | 2020 |
Synthesis and stereochemical analysis of β-nitromethane substituted γ-amino acids and peptides MG Kumar, SM Mali, HN Gopi Organic & biomolecular chemistry 11 (5), 803-813, 2013 | 13 | 2013 |
γ-and β-Peptide Foldamers from Common Multifaceted Building Blocks: Synthesis and Structural Characterization M Ganesh Kumar, HN Gopi Organic letters 17 (19), 4738-4741, 2015 | 12 | 2015 |
Solid-phase peptide synthesis on disulfide-linker resin followed by reductive release affords pure thiol-functionalized peptides Z Bognar, GK Mothukuri, AL Nielsen, ML Merz, PMF Pânzar, C Heinis Organic & Biomolecular Chemistry 20 (29), 5699-5703, 2022 | 11 | 2022 |
Direct Transformation of N-Protected α, β-Unsaturated γ-Amino Amides into γ-Lactams through a Base-Mediated Molecular Rearrangement M Ganesh Kumar, K Veeresh, SA Nalawade, RV Nithun, HN Gopi The Journal of Organic Chemistry 84 (23), 15145-15153, 2019 | 11 | 2019 |
Engineering polypeptide folding through trans double bonds: transformation of miniature β-meanders to hybrid helices M Ganesh Kumar, SN Benke, KMP Raja, HN Gopi Chemical Communications 51 (69), 13397-13399, 2015 | 7 | 2015 |
Synthesis of Tetrasubstituted Symmetrical Pyrazines from β‐Keto γ‐Amino Esters: A Mild Strategy for Self‐Dimerization of Peptides M Ganesh Kumar, VJ Thombare, RD Bhaisare, A Adak, HN Gopi European Journal of Organic Chemistry 2015 (1), 135-141, 2015 | 5 | 2015 |
In Vitro-Evolved Peptides Bind Monomeric Actin and Mimic Actin-Binding Protein Thymosin-β4 CH Raphael J. Gübeli, Davide Bertoldo, Kenji Shimada, Christian B. Gerhold ... ACS Chem. Biol. 16 (5), 820–828, 2021 | 2 | 2021 |
Helices with additional H‐bonds: crystallographic conformations of α, γ‐hybrid peptides helices composed of β‐hydroxy γ‐amino acids (statines) A Malik, M Ganesh Kumar, A Bandyopadhyay, HN Gopi Peptide Science 108 (1), 2017 | 1 | 2017 |
Large Libraries of Structurally Diverse Macrocycles Suitable for Membrane Permeation AL Nielsen, Z Bognar, GK Mothukuri, A Zarda, M Schüttel, ML Merz, X Ji, ... Angewandte Chemie, e202400350, 2024 | | 2024 |
Crystal structure analysis of helix–turn–helix type motifs in α, γ-hybrid peptides SA Nalawade, MG Kumar, DRP Kumar, M Singh, S Dey, HN Gopi CrystEngComm 26 (7), 913-917, 2024 | | 2024 |
Method for preparing a library of peptides or a peptide C Heinis, S Habeshian, GK Mothukuri, M Schüttel, M Merz, G Sangouard, ... | | 2022 |