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Jaideep Bharate
Jaideep Bharate
Senior Research Investigator at Syngene International Ltd
在 syngeneintl.com 的电子邮件经过验证 - 首页
标题
引用次数
引用次数
年份
Metal-free domino one-pot protocols for quinoline synthesis
JB Bharate, RA Vishwakarma, SB Bharate
RSC advances 5 (52), 42020-42053, 2015
1712015
Discovery of 3, 3′-diindolylmethanes as potent antileishmanial agents
SB Bharate, JB Bharate, SI Khan, BL Tekwani, MR Jacob, R Mudududdla, ...
European journal of medicinal chemistry 63, 435-443, 2013
1072013
Cu–Mn spinel oxide catalyzed synthesis of imidazo [1, 2-a] pyridines through domino three-component coupling and 5-exo-dig cyclization in water
JB Bharate, SK Guru, SK Jain, S Meena, PP Singh, S Bhushan, B Singh, ...
RSC advances 3 (43), 20869-20876, 2013
502013
Tandem one-pot synthesis of flavans by recyclable silica–HClO 4 catalyzed Knoevenagel condensation and [4+ 2]-Diels–Alder cycloaddition
SB Bharate, R Mudududdla, JB Bharate, N Battini, S Battula, RR Yadav, ...
Organic & Biomolecular Chemistry 10 (26), 5143-5150, 2012
432012
Metal-Free, ionic liquid-mediated synthesis of functionalized quinolines
JB Bharate, SB Bharate, RA Vishwakarma
ACS combinatorial science 16 (11), 624-630, 2014
422014
Synthesis, and the antioxidant, neuroprotective and P-glycoprotein induction activity of 4-arylquinoline-2-carboxylates
JB Bharate, A Wani, S Sharma, SI Reja, M Kumar, RA Vishwakarma, ...
Organic & Biomolecular Chemistry 12 (32), 6267-6277, 2014
392014
Efficient synthesis of 2, 3-dihydroquinazolin-4 (1H)-ones using heterogeneous solid acid catalysts: unexpected formation of
SB Bharate, N Mupparapu, S Manda, JB Bharate, R Mudududdla, ...
Arkivoc 8, 308-318, 2012
382012
Discovery of 4-acetyl-3-(4-fluorophenyl)-1-(p-tolyl)-5-methylpyrrole as a dual inhibitor of human P-glycoprotein and Staphylococcus aureus Nor A efflux pump
JB Bharate, S Singh, A Wani, S Sharma, P Joshi, IA Khan, A Kumar, ...
Organic & Biomolecular Chemistry 13 (19), 5424-5431, 2015
352015
Cobalt (ii) catalyzed C (sp)–H bond functionalization of alkynes with phenyl hydrazines: facile access to diaryl 1, 2-diketones
JB Bharate, S Abbat, R Sharma, PV Bharatam, RA Vishwakarma, ...
Organic & Biomolecular Chemistry 13 (18), 5235-5242, 2015
322015
Montmorillonite clay catalyzed synthesis of functionalized pyrroles through domino four-component coupling of amines, aldehydes, 1, 3-dicarbonyl compounds and nitroalkanes
JB Bharate, R Sharma, S Aravinda, VK Gupta, B Singh, SB Bharate, ...
RSC advances 3 (44), 21736-21742, 2013
322013
ortho-Amidoalkylation of Phenols via Tandem One-Pot Approach Involving Oxazine Intermediate
R Mudududdla, SK Jain, JB Bharate, AP Gupta, B Singh, ...
The Journal of Organic Chemistry 77 (19), 8821-8827, 2012
302012
CuBr catalyzed aerobic oxidative coupling of 2-aminopyridines with cinnamaldehydes: direct access to 3-formyl-2-phenyl-imidazo [1, 2-a] pyridines
JB Bharate, S Abbat, PV Bharatam, RA Vishwakarma, SB Bharate
Organic & Biomolecular Chemistry 13 (28), 7790-7794, 2015
222015
Synthesis and P-glycoprotein induction activity of colupulone analogs
JB Bharate, YS Batarseh, A Wani, S Sharma, RA Vishwakarma, ...
Organic & biomolecular chemistry 13 (19), 5488-5496, 2015
202015
Rational design, synthesis and biological evaluation of pyrimidine-4, 6-diamine derivatives as type-II inhibitors of FLT3 selective against c-KIT
JB Bharate, N McConnell, G Naresh, L Zhang, NR Lakkaniga, L Ding, ...
Scientific reports 8 (1), 3722, 2018
152018
KF/alumina catalyzed regioselective benzylation and benzoylation using solvent-free grind-stone chemistry
SK Jain, S Meena, B Singh, JB Bharate, P Joshi, VP Singh, ...
RSC advances 2 (24), 8929-8933, 2012
152012
Deformylation of indole and azaindole-3-carboxaldehydes using anthranilamide and solid acid heterogeneous catalyst via quinazolinone intermediate
RR Yadav, N Battini, R Mudududdla, JB Bharate, N Muparappu, ...
Tetrahedron Letters 53 (17), 2222-2225, 2012
142012
Discovery of imidazo [1, 2-a] pyridine-thiophene derivatives as FLT3 and FLT3 mutants inhibitors for acute myeloid leukemia through structure-based optimization of an NEK2 …
L Zhang, NR Lakkaniga, JB Bharate, N Mcconnell, X Wang, A Kharbanda, ...
European journal of medicinal chemistry 225, 113776, 2021
132021
QSAR and pharmacophore modeling of N-acetyl-2-aminobenzothiazole class of phosphoinositide-3-kinase-α inhibitors
SB Bharate, B Singh, JB Bharate, SK Jain, S Meena, RA Vishwakarma
Medicinal Chemistry Research 22, 890-899, 2013
112013
Discovery of N-trisubstituted pyrimidine derivatives as type I RET and RET gatekeeper mutant inhibitors with a novel kinase binding pose
L Zhang, M Moccia, DC Briggs, JB Bharate, NR Lakkaniga, P Knowles, ...
Journal of medicinal chemistry 65 (2), 1536-1551, 2022
82022
Quantification of the polyisoprenylated benzophenones garcinol and isogarcinol using multiple reaction monitoring LC/electrospray ionization-MS/MS analysis of ultrasound …
JB Bharate, RA Vishwakarma, SB Bharate, M Kushwaha, AP Gupta
Journal of AOAC International 97 (5), 1317-1322, 2014
72014
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