| Synthesis and pharmacological investigation of 3-(substituted 1-phenylethanone)-4-(substituted phenyl)-1, 2, 3, 4-tetrahydropyrimidine-5-carboxylates RV Chikhale, RP Bhole, PB Khedekar, KP Bhusari European journal of medicinal chemistry 44 (9), 3645-3653, 2009 | 143 | 2009 |
| Overview of the development of DprE1 inhibitors for combating the menace of tuberculosis RV Chikhale, MA Barmade, PR Murumkar, MR Yadav Journal of medicinal chemistry 61 (19), 8563-8593, 2018 | 127 | 2018 |
| Development of selective DprE1 inhibitors: Design, synthesis, crystal structure and antitubercular activity of benzothiazolylpyrimidine-5-carboxamides R Chikhale, S Menghani, R Babu, R Bansode, G Bhargavi, N Karodia, ... European journal of medicinal chemistry 96, 30-46, 2015 | 122 | 2015 |
| DNA G-quadruplex and i-motif structure formation is interdependent in human cells JJ King, KL Irving, CW Evans, RV Chikhale, R Becker, CJ Morris, ... Journal of the American Chemical Society 142 (49), 20600-20604, 2020 | 98 | 2020 |
| CD4+ effector T cells accelerate Alzheimer’s disease in mice J Machhi, P Yeapuri, Y Lu, E Foster, R Chikhale, J Herskovitz, ... Journal of neuroinflammation 18, 1-23, 2021 | 76 | 2021 |
| Identification of potential anti-TMPRSS2 natural products through homology modelling, virtual screening and molecular dynamics simulation studies RV Chikhale, VK Gupta, GE Eldesoky, SM Wabaidur, SA Patil, MA Islam Journal of Biomolecular Structure and Dynamics 39 (17), 6660-6675, 2021 | 74 | 2021 |
| Chandipura virus: an emerging tropical pathogen S Menghani, R Chikhale, A Raval, P Wadibhasme, P Khedekar Acta tropica 124 (1), 1-14, 2012 | 67 | 2012 |
| Mycobacterium enoyl acyl carrier protein reductase (InhA): A key target for antitubercular drug discovery MS Prasad, RP Bhole, PB Khedekar, RV Chikhale Bioorganic Chemistry 115, 105242, 2021 | 66 | 2021 |
| Design, synthesis and anticancer studies of novel aminobenzazolyl pyrimidines as tyrosine kinase inhibitors R Chikhale, S Thorat, RK Choudhary, N Gadewal, P Khedekar Bioorganic chemistry 77, 84-100, 2018 | 59 | 2018 |
| Design, synthesis and pharmacological evaluation of pyrimidobenzothiazole-3-carboxylate derivatives as selective L-type calcium channel blockers R Chikhale, S Thorat, A Pant, A Jadhav, KC Thatipamula, R Bansode, ... Bioorganic & medicinal chemistry 23 (20), 6689-6713, 2015 | 53 | 2015 |
| Mycobacterial membrane protein large 3 (MmpL3) inhibitors: a promising approach to combat tuberculosis MD Umare, PB Khedekar, RV Chikhale ChemMedChem 16 (20), 3136-3148, 2021 | 40 | 2021 |
| Generation of phenothiazine with potent anti-TLK1 activity for prostate cancer therapy V Singh, S Bhoir, RV Chikhale, J Hussain, D Dwyer, RA Bryce, ... Iscience 23 (9), 2020 | 25 | 2020 |
| Unlocking the potential of PROTACs: A comprehensive review of protein degradation strategies in disease therapy RP Bhole, PR Kute, RV Chikhale, CG Bonde, A Pant, SS Gurav Bioorganic Chemistry 139, 106720, 2023 | 23 | 2023 |
| i-Motif formation and spontaneous deletions in human cells M Martella, F Pichiorri, RV Chikhale, MAS Abdelhamid, ZAE Waller, ... Nucleic Acids Research 50 (6), 3445-3455, 2022 | 22 | 2022 |
| TLK1-mediated RAD54 phosphorylation spatio-temporally regulates Homologous Recombination Repair I Ghosh, Y Kwon, AB Shabestari, R Chikhale, J Chen, C Wiese, P Sung, ... Nucleic acids research 51 (16), 8643-8662, 2023 | 13 | 2023 |
| Current biomarkers and treatment strategies in Alzheimer disease: An overview and future perspectives RP Bhole, RV Chikhale, KM Rathi IBRO neuroscience reports 16, 8-42, 2024 | 11 | 2024 |
| Tracing the GSAP–APP C-99 interaction site in the β-amyloid pathway leading to Alzheimer’s Disease D Angira, R Chikhale, K Mehta, RA Bryce, V Thiruvenkatam ACS Chemical Neuroscience 10 (8), 3868-3879, 2019 | 10 | 2019 |
| Targeting dormant phenotype acquired mycobacteria using natural products by exploring its important targets: In vitro and in silico studies S Sharma, R Chikhale, N Shinde, AM Khan, VK Gupta Frontiers in Cellular and Infection Microbiology 13, 1111997, 2023 | 9 | 2023 |
| Identification of novel hit molecules targeting M. tuberculosis polyketide synthase 13 by combining generative AI and physics-based methods RV Chikhale, R Choudhary, J Malhotra, GE Eldesoky, P Mangal, PC Patil Computers in Biology and Medicine 176, 108573, 2024 | 8 | 2024 |
| Identification of sugar-containing natural products that interact with i-motif DNA RV Chikhale, D Guneri, R Yuan, CJ Morris, ZAE Waller Bioorganic & Medicinal Chemistry Letters 73, 128886, 2022 | 7 | 2022 |
Zoe WallerProfessor of Drug Discovery, School of Pharmacy, UCL在 ucl.ac.uk 的电子邮件经过验证
