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Gwenaëlle Jézéquel
Gwenaëlle Jézéquel
Postdoc at Helmholtz Institute, Saarbrücken
在 helmholtz-hips.de 的电子邮件经过验证
标题
引用次数
引用次数
年份
Fighting antibiotic resistance—strategies and (pre) clinical developments to find new antibacterials
S Walesch, J Birkelbach, G Jézéquel, FPJ Haeckl, JD Hegemann, ...
EMBO reports 24 (1), e56033, 2023
1022023
Cytotoxic Prenylated Stilbenes Isolated from Macaranga tanarius
T Péresse, G Jézéquel, PM Allard, VC Pham, DTM Huong, F Blanchard, ...
Journal of natural products 80 (10), 2684-2691, 2017
562017
Structure-Based Design of α-Substituted Mercaptoacetamides as Inhibitors of the Virulence Factor LasB from Pseudomonas aeruginosa
C Kaya, I Walter, A Alhayek, R Shafiei, G Jézéquel, A Andreas, ...
ACS Infectious Diseases 8 (5), 1010-1021, 2022
152022
The Structures and Binding Modes of Small-Molecule Inhibitors of Pseudomonas aeruginosa Elastase LasB
V Camberlein, G Jézéquel, J Haupenthal, AKH Hirsch
Antibiotics 11 (8), 1060, 2022
102022
Structure-Based Design of a Lead Compound Derived from Natural Schweinfurthins with Antitumor Properties That Target Oxysterol-Binding Protein
G Jézéquel, C Rampal, C Guimard, D Kovacs, J Polidori, J Bigay, ...
Journal of Medicinal Chemistry 66 (20), 14208-14220, 2023
62023
Synthesis and anti-leishmanial properties of quinolones derived from zanthosimuline
G Jézéquel, LNF Cardoso, F Olivon, I Dennemont, C Apel, M Litaudon, ...
Molecules 27 (22), 7892, 2022
22022
Target-Directed Dynamic Combinatorial Chemistry Affords Binders of Mycobacterium tuberculosis IspE
M Braun-Cornejo, C Ornago, V Sonawane, J Haupenthal, AM Kany, ...
ACS omega, 2024
2024
Funktionalisierung von Chlorotonilen: Dehalogenil als vielversprechende Leitverbindung für die in vivo‐Anwendung
W Hofer, F Deschner, G Jézéquel, L Pessanha de Carvalho, ...
Angewandte Chemie 136 (19), e202319765, 2024
2024
Functionalization of Chlorotonils: Dehalogenil as Promising Lead Compound for In Vivo Application
W Hofer, F Deschner, G Jézéquel, L Pessanha de Carvalho, ...
Angewandte Chemie International Edition 63 (19), e202319765, 2024
2024
Bio-inspired synthesis and profiling of a potent antiviral flavonol targeting the lipid exchanger OSBP
G Jézéquel, Z Grimanelli, C Guimard, J Bigay, J Haddad, J Bignon, ...
2024
Target-directed dynamic combinatorial chemistry affords inhibitors of Nsp10 as potential antivirals against SARS-CoV-2
RP Jumde, G Jézéquel, M Saramago, N Frank, S Adam, MV Cunha, ...
2023
Process for the biobased synthesis of schweinfurthins G, K and R
M Litaudon, F Roussi, S Desrat, G Jézéquel, C Rampal, HDT Mai
2023
Efficient synthetic strategy to access analogues of an original natural bioactive flavone
C Guimard, G Jézéquel, L Askenatzis, B Mesmin, J Bignon, S Desrat, ...
Journées de Chimie Organique (JCO) 2022, 2022
2022
Targeting OSBP degradation by PROTACs derived from schweinfurthin for cancer therapy
C Guimard, G Jézéquel, L Askenatzis, J Bignon, S Desrat, F Roussi
27th EFMC International Symposium on Medicinal Chemistry, 2022
2022
Compound of the 7a, 8, 9, 10, 11, 11a-hexahydro-1H, 7H-pyrano [2, 3-c] xanthene type, method of preparation thereof, intermediates thereof and therapeutic applications thereof
F Roussi, S Desrat, G Jézéquel, M Litaudon, J Bignon, B Mesmin, ...
2022
Novel process for the biobased synthesis of Schweinfurthins G, K and R.
F Roussi, M Litaudon, S Desrat, C Rampal, G Jézéquel, CP Van, ...
2022
Structure-based design of a-substituted mercaptoacetamides as inhibitors of the virulence factor LasB from Pseudomonas aeruginosa.
C Kaya, I Walter, A Alhayek, R Shafiei, G Jézéquel, A Andreas, ...
2022
Synthèse et pharmacomodulation de composés antitumoraux naturels à motif hexahydroxanthène
G Jezequel
Université Paris-Saclay (ComUE), 2019
2019
New dual molecules as an innovative strategy against glioblastoma: synthesis and biological evaluation
G Jézéquel, T Péresse, T Virolle, J Bignon, S Desrat, F Roussi
8th EFMC International Symposium on Advances in Synthetic and Medicinal …, 2019
2019
Dual molecule to enhance biological activity of an anticancer drug targeting glioblastoma
G Jézéquel, T Péresse, M Litaudon, T Virolle, J Bignon, S Desrat, ...
16th Belgian Organic Synthesis Symposium (BOSS), 2018
2018
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