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Shishir Chourey
Shishir Chourey
Principal Scientist, Bristol Myers Squibb
在 bms.com 的电子邮件经过验证
标题
引用次数
引用次数
年份
Role of metal ion in specific recognition of pyrophosphate ion under physiological conditions and hydrolysis of the phosphoester linkage by alkaline phosphatase
P Das, NB Chandar, S Chourey, H Agarwalla, B Ganguly, A Das
Inorganic Chemistry 52 (19), 11034-11041, 2013
622013
Inhibition of 5-oxo-6, 8, 11, 14-eicosatetraenoic acid-induced activation of neutrophils and eosinophils by novel indole OXE receptor antagonists
V Gore, S Gravel, C Cossette, P Patel, S Chourey, Q Ye, J Rokach, ...
Journal of medicinal chemistry 57 (2), 364-377, 2014
322014
Two potent OXE-R antagonists: assignment of stereochemistry
P Patel, CN Reddy, V Gore, S Chourey, Q Ye, YP Ouedraogo, S Gravel, ...
ACS Medicinal Chemistry Letters 5 (7), 815-819, 2014
182014
Pharmacokinetics and metabolism of selective oxoeicosanoid (OXE) receptor antagonists and their effects on 5-oxo-6, 8, 11, 14-eicosatetraenoic acid (5-oxo-ETE)-induced …
C Cossette, S Chourey, Q Ye, C Nagendra Reddy, V Gore, S Gravel, ...
Journal of Medicinal Chemistry 59 (22), 10127-10146, 2016
162016
Biosynthesis and actions of 5-oxoeicosatetraenoic acid (5-oxo-ETE) on feline granulocytes
C Cossette, S Gravel, CN Reddy, V Gore, S Chourey, Q Ye, NW Snyder, ...
Biochemical pharmacology 96 (3), 247-255, 2015
152015
Stereoselective synthesis of two highly potent 5-oxo-ETE receptor antagonists
CN Reddy, Q Ye, S Chourey, S Gravel, WS Powell, J Rokach
Tetrahedron letters 56 (49), 6896-6899, 2015
142015
Novel highly potent OXE receptor antagonists with prolonged plasma lifetimes that are converted to active metabolites in vivo in monkeys
Q Ye, S Chourey, CN Reddy, R Wang, C Cossette, S Gravel, ...
British Journal of Pharmacology 177 (2), 388-401, 2020
112020
Inhibition of allergen‐induced dermal eosinophilia by an oxoeicosanoid receptor antagonist in non‐human primates
LA Miller, C Cossette, S Chourey, Q Ye, CN Reddy, J Rokach, WS Powell
British Journal of Pharmacology 177 (2), 360-371, 2020
102020
In vivo α-hydroxylation of a 2-alkylindole antagonist of the OXE receptor for the eosinophil chemoattractant 5-oxo-6, 8, 11, 14-eicosatetraenoic acid in monkeys
S Chourey, Q Ye, CN Reddy, C Cossette, S Gravel, M Zeller, ...
Biochemical pharmacology 138, 107-118, 2017
102017
Novel highly potent and metabolically resistant oxoeicosanoid (OXE) receptor antagonists that block the actions of the granulocyte chemoattractant 5-oxo-6, 8, 11, 14 …
S Chourey, Q Ye, CN Reddy, R Wang, C Cossette, S Gravel, ...
Journal of Medicinal Chemistry 61 (14), 5934-5948, 2018
92018
Stereoselective Synthesis of Maresin-like Lipid Mediators
S Hong, Y Lu, M Morita, S Saito, Y Kobayashi, B Jun, NG Bazan, X Xu, ...
Synlett 30 (03), 343-347, 2019
82019
Metabolism and pharmacokinetics of a potent N-acylindole antagonist of the OXE receptor for the eosinophil chemoattractant 5-oxo-6, 8, 11, 14-eicosatetraenoic acid (5-oxo-ETE …
CN Reddy, H Alhamza, S Chourey, Q Ye, V Gore, C Cossette, S Gravel, ...
European Journal of Pharmaceutical Sciences 115, 88-99, 2018
82018
Targeting the OXE receptor with a selective antagonist inhibits allergen‐induced pulmonary inflammation in non‐human primates
C Cossette, LA Miller, Q Ye, S Chourey, CN Reddy, J Rokach, WS Powell
British journal of pharmacology 179 (2), 322-336, 2022
72022
Structure-activity relationship study of β-oxidation resistant indole-based 5-oxo-6, 8, 11, 14-eicosatetraenoic acid (5-oxo-ETE) receptor antagonists
Q Ye, S Chourey, R Wang, NR Chintam, S Gravel, WS Powell, J Rokach
Bioorganic & medicinal chemistry letters 27 (20), 4770-4776, 2017
72017
Design and synthesis of affinity chromatography ligands for the purification of 5-hydroxyeicosanoid dehydrogenase
CN Reddy, Q Ye, P Patel, S Sivendran, S Chourey, R Wang, JR Anumolu, ...
Bioorganic & Medicinal Chemistry 25 (1), 116-125, 2017
72017
Base-dependent formation of cis and trans olefins and their application in the synthesis of 5-oxo-ETE receptor antagonists
V Gore, S Chourey, Q Ye, P Patel, Y Ouedraogo, S Gravel, WS Powell, ...
Bioorganic & Medicinal Chemistry Letters 24 (15), 3385-3388, 2014
62014
Metabolism of anti-inflammatory OXE (oxoeicosanoid) receptor antagonists by nonhuman primates
C Cossette, S Chourey, Q Ye, CN Reddy, R Wang, S Poulet, ...
European Journal of Pharmaceutical Sciences 172, 106144, 2022
12022
Concise Syntheses of Microsomal Metabolites of a Potent OXE (Oxoeicosanoid) Receptor Antagonist
S Chourey, R Wang, Q Ye, CN Reddy, S Sun, N Takenaka, WS Powell, ...
Chemical and Pharmaceutical Bulletin 71 (7), 534-544, 2023
2023
Corrigendum to" In vivo α-hydroxylation of a 2-alkylindole antagonist of the OXE receptor for the eosinophil chemoattractant 5-oxo-6, 8, 11, 14-eicosatetraenoic acid in monkeys …
S Chourey, Q Ye, CN Reddy, C Cossette, S Gravel, M Zeller, ...
Biochemical pharmacology 154, 174, 2018
2018
Structural modifications of OXE receptor antagonists towards improved in vivo metabolic stability
S Chourey, Q Ye, C Reddy, R Wang, S Gravel, C Cossette, ...
ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY 253, 2017
2017
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