What Makes a Kinase Promiscuous for Inhibitors? SM Hanson, G Georghiou, MK Thakur, WT Miller, JS Rest, JD Chodera, ... Cell chemical biology 26 (3), 390-399. e5, 2019 | 82 | 2019 |
A small molecule inhibitor of Nicotinamide N-methyltransferase for the treatment of metabolic disorders A Kannt, S Rajagopal, SV Kadnur, J Suresh, RK Bhamidipati, ... Scientific reports 8 (1), 3660, 2018 | 81 | 2018 |
The structure of XIAP BIR2: understanding the selectivity of the BIR domains C Lukacs, C Belunis, R Crowther, W Danho, L Gao, B Goggin, CA Janson, ... Acta Crystallographica Section D: Biological Crystallography 69 (9), 1717-1725, 2013 | 45 | 2013 |
Inhibiting ACK1-mediated phosphorylation of C-terminal Src kinase counteracts prostate cancer immune checkpoint blockade resistance D Sridaran, S Chouhan, K Mahajan, A Renganathan, C Weimholt, ... Nature communications 13 (1), 6929, 2022 | 28 | 2022 |
Expression stability of two housekeeping genes (18S rRNA and G3PDH) during in vitro maturation of follicular oocytes in buffalo (Bubalus bubalis) APS Aswal, S Raghav, S De, M Thakur, SL Goswami, TK Datta Animal reproduction science 103 (1-2), 164-171, 2008 | 21 | 2008 |
Discovery and molecular basis of subtype-selective cyclophilin inhibitors AA Peterson, AM Rangwala, MK Thakur, PS Ward, C Hung, IR Outhwaite, ... Nature Chemical Biology 18 (11), 1184-1195, 2022 | 19 | 2022 |
Co-crystal structures of PTK6: With Dasatinib at 2.24 Å, with novel imidazo [1, 2-a] pyrazin-8-amine derivative inhibitor at 1.70 Å resolution MK Thakur, S Birudukota, S Swaminathan, SK Battula, S Vadivelu, ... Biochemical and biophysical research communications 482 (4), 1289-1295, 2017 | 12 | 2017 |
Crystal structures of monkey and mouse nicotinamide N-methyltransferase (NNMT) bound with end product, 1-methyl nicotinamide S Swaminathan, S Birudukota, MK Thakur, R Parveen, S Kandan, S Juluri, ... Biochemical and biophysical research communications 491 (2), 416-422, 2017 | 10 | 2017 |
Characterization of the luteinizing hormone beta (LH-β) subunit gene in the Indian river buffalo (Bubalus bubalis) MS Basavarajappa, S De, M Thakur, TK Datta, G Dogra, P Yadav, ... General and comparative endocrinology 155 (1), 63-69, 2008 | 7 | 2008 |
Crystal structure of the kinase domain of human protein tyrosine kinase 6 (PTK6) at 2.33 Å resolution MK Thakur, A Kumar, S Birudukota, S Swaminathan, R Tyagi, R Gosu Biochemical and biophysical research communications 478 (2), 637-642, 2016 | 5 | 2016 |
Small molecule modulators to understand the role of IDO1 and TDO2 in cancer SR Garapaty, D Sivanandhan, GPK Seerapu, S Naidu, S Chakelam, ... Cancer Research 77 (13_Supplement), 5578-5578, 2017 | | 2017 |