VOSO4 catalyzed highly efficient synthesis of benzimidazoles, benzothiazoles, and quinoxalines CS Digwal, U Yadav, AP Sakla, PVS Ramya, S Aaghaz, A Kamal Tetrahedron Letters 57 (36), 4012-4016, 2016 | 72 | 2016 |
Synthesis and biological evaluation of curcumin inspired indole analogues as tubulin polymerization inhibitors PVS Ramya, S Angapelly, L Guntuku, CS Digwal, BN Babu, VGM Naidu, ... European Journal of Medicinal Chemistry 127, 100-114, 2017 | 70 | 2017 |
Synthesis and biological evaluation of curcumin inspired imidazo [1, 2-a] pyridine analogues as tubulin polymerization inhibitors PVS Ramya, L Guntuku, S Angapelly, CS Digwal, UJ Lakshmi, ... European journal of medicinal chemistry 143, 216-231, 2018 | 53 | 2018 |
PET molecular imaging in drug development: the imaging and chemistry perspective SG Nerella, P Singh, T Sanam, CS Digwal Frontiers in Medicine 9, 812270, 2022 | 50 | 2022 |
Curcumin inspired 2-chloro/phenoxy quinoline analogues: Synthesis and biological evaluation as potential anticancer agents AK P. V. Sri Ramya, Lalita Guntuku, Srinivas Angapelly, Shailaja Karri ... Bioorganic & Medicinal Chemistry Letters, 2018 | 48 | 2018 |
Structural and functional complexity of HSP90 in cellular homeostasis and disease G Chiosis, CS Digwal, JB Trepel, L Neckers Nature Reviews Molecular Cell Biology 24 (11), 797-815, 2023 | 37 | 2023 |
A Chemical Biology Approach to the Chaperome in Cancer—HSP90 and Beyond T Taldone, T Wang, A Rodina, NVK Pillarsetty, CS Digwal, S Sharma, ... Cold Spring Harbor perspectives in biology, a034116, 2019 | 36 | 2019 |
Discovery of curcumin inspired sulfonamide derivatives as a new class of carbonic anhydrase isoforms I, II, IX, and XII inhibitors PVS Ramya, S Angapelly, A Angeli, CS Digwal, M Arifuddin, BN Babu, ... Journal of Enzyme Inhibition and Medicinal Chemistry 32 (1), 1274-1281, 2017 | 32 | 2017 |
Vanadium-Catalyzed Oxidative C (CO)–C (CO) Bond Cleavage for C–N Bond Formation: One-Pot Domino Transformation of 1, 2-Diketones and Amidines into Imides and Amides CS Digwal, U Yadav, PVS Ramya, S Sana, B Swain, A Kamal The Journal of Organic Chemistry 82 (14), 7332-7345, 2017 | 29 | 2017 |
Chemical tools for epichaperome-mediated interactome dysfunctions of the central nervous system A Bolaender, D Zatorska, H He, S Joshi, S Sharma, CS Digwal, HJ Patel, ... Nature Communications 12 (1), 4669, 2021 | 21 | 2021 |
Imidazo[1,2-a]pyridines linked with thiazoles/thiophene motif through keto spacer as potential cytotoxic agents and NF-κB inhibitors MA Kamala K. Vasu, Chander Singh Digwal, Amit N. Pandya, Dhaivat H. Pandya ... Bioorganic & Medicinal Chemistry Letters, 2017 | 19 | 2017 |
Disease‐specific interactome alterations via epichaperomics: the case for Alzheimer’s disease SD Ginsberg, TA Neubert, S Sharma, CS Digwal, P Yan, C Timbus, ... The FEBS journal 289 (8), 2047-2066, 2022 | 18 | 2022 |
Hypervalent iodine (III) catalyzed rapid and efficient access to benzimidazoles, benzothiazoles and quinoxalines: Biological evaluation of some new benzimidazole-imidazo [1, 2 … PVS Ramya, S Angapelly, RS Rani, CS Digwal, CG Kumar, BN Babu, ... Arabian Journal of Chemistry 13 (1), 120-133, 2020 | 18 | 2020 |
Synthesis and exploration of 2-morpholino-4-phenylthiazol-5-yl acrylamide derivatives for their effects against carbonic anhydrase I, II, IX and XII isoforms as a non … B Swain, CS Digwal, A Angeli, M Alvala, P Singh, CT Supuran, ... Bioorganic & Medicinal Chemistry 27 (21), 115090, 2019 | 14 | 2019 |
Pharmacologically controlling protein-protein interactions through epichaperomes for therapeutic vulnerability in cancer S Joshi, EDG Gomes, T Wang, A Corben, T Taldone, S Gandu, C Xu, ... Communications Biology 4 (1), 1333, 2021 | 13 | 2021 |
Design and synthesis of 5‐Morpholino‐Thiophene‐Indole/Oxindole hybrids as cytotoxic agents U Yadav, AP Sakla, R Tokala, ST Nyalam, A Khurana, CS Digwal, V Talla, ... ChemistrySelect 5 (14), 4356-4363, 2020 | 11 | 2020 |
Systems-level analyses of protein-protein interaction network dysfunctions via epichaperomics identify cancer-specific mechanisms of stress adaptation A Rodina, C Xu, CS Digwal, S Joshi, Y Patel, AR Santhaseela, S Bay, ... Nature communications 14 (1), 3742, 2023 | 10 | 2023 |
Chemical probes and methods for single-cell detection and quantification of epichaperomes in hematologic malignancies S Merugu, S Sharma, J Kaner, C Digwal, M Sugita, S Joshi, T Taldone, ... Methods in enzymology 639, 289-311, 2020 | 10 | 2020 |
How aberrant N-glycosylation can alter protein functionality and ligand binding: An atomistic view M Castelli, P Yan, A Rodina, CS Digwal, P Panchal, G Chiosis, E Moroni, ... Structure 31 (8), 987-1004. e8, 2023 | 9 | 2023 |
An efficient RuCl3· H2O/I2 catalytic system: A facile access to 3-aroylimidazo [1, 2-a] pyridines from 2-aminopyridines and chalcones PVS Ramya, S Angapelly, CS Digwal, U Yadav, BN Babu, A Kamal Journal of Saudi Chemical Society 22 (1), 90-100, 2018 | 7 | 2018 |