Facile Synthesis and Antibacterial, Antitubercular, and Anticancer Activities of Novel 1, 4‐Dihydropyridines K Sirisha, G Achaiah, VM Reddy Archiv der Pharmazie 343 (6), 342-352, 2010 | 112 | 2010 |
Synthesis, antibacterial and antimycobacterial activities of some new 4-aryl/heteroaryl-2, 6-dimethyl-3, 5-bis-N-(aryl)-carbamoyl-1, 4-dihydropyridines K Sirisha, D Bikshapathi, G Achaiah, VM Reddy European journal of medicinal chemistry 46 (5), 1564-1571, 2011 | 108 | 2011 |
Novel targets for antiinflammatory and antiarthritic agents RG Kulkarni, G Achaiah, G Narahari Sastry Current pharmaceutical design 12 (19), 2437-2454, 2006 | 72 | 2006 |
Synthesis of new pyrrolo [2, 3-d] pyrimidine derivatives and evaluation of their activities against human colon cancer cell lines SJ Tangeda, A Garlapati European journal of medicinal chemistry 45 (4), 1453-1458, 2010 | 71 | 2010 |
Molecular modeling studies of phenoxypyrimidinyl imidazoles as p38 kinase inhibitors using QSAR and docking GK Ravindra, G Achaiah, GN Sastry European journal of medicinal chemistry 43 (4), 830-838, 2008 | 57 | 2008 |
Quaternary salts of 4, 3′ and 4, 4′ bis-pyridinium monooximes: synthesis and biological activity SR Chennamaneni, V Vobalaboina, A Garlapati Bioorganic & medicinal chemistry letters 15 (12), 3076-3080, 2005 | 44 | 2005 |
Quaternary salts of 4, 3′ and 4, 4′ bis-pyridinium monooximes. Part 2: Synthesis and biological activity CS Rao, V Venkateswarlu, G Achaiah Bioorganic & medicinal chemistry letters 16 (8), 2134-2138, 2006 | 40 | 2006 |
Strategies to design pyrazolyl urea derivatives for p38 kinase inhibition: a molecular modeling study RG Kulkarni, P Srivani, G Achaiah, GN Sastry Journal of Computer-Aided Molecular Design 21, 155-166, 2007 | 37 | 2007 |
Molecular docking studies and in vitro screening of new dihydropyridine derivatives as human MRP1 inhibitors K Sirisha, MC Shekhar, K Umasankar, P Mahendar, A Sadanandam, ... Bioorganic & medicinal chemistry 19 (10), 3249-3254, 2011 | 36 | 2011 |
Fluorinated non-imidazole histamine H3 receptor antagonists HS K. Isensee ,M.Amon, A. Garlapati , X. Ligneau , J.-C. Camelin , M. Capet ... Bioorg. Med. Chem. Lett 19, 2172-2175, 2009 | 35 | 2009 |
Rational design and synthesis of novel 2-(substituted-2 H-chromen-3-yl)-5-aryl-1 H-imidazole derivatives as an anti-angiogenesis and anti-cancer agent G Gudipudi, SR Sagurthi, S Perugu, G Achaiah, GLD Krupadanam RSC Advances 4 (99), 56489-56501, 2014 | 27 | 2014 |
Design, synthesis, in silico studies, and evaluation of novel chalcones and their pyrazoline derivatives for antibacterial and antitubercular activities S Pola, KK Banoth, M Sankaranarayanan, R Ummani, A Garlapati Medicinal Chemistry Research 29, 1819-1835, 2020 | 26 | 2020 |
Synthesis, p38 kinase inhibitory and anti-inflammatory activity of new substituted benzimidazole derivatives R G Kulkarni, S A Laufer, C V M, A Garlapati Medicinal Chemistry 9 (1), 91-99, 2013 | 25 | 2013 |
Synthesis of 6‐Alkyl/Aralkyl‐5a, 11‐dihydro‐9‐nitro (1) benzopyrano‐(2, 3‐b)(1, 5) benzodiazepin‐13‐ones as Possible Antipsychotic Agents. TK Devi, G Achaiah, VM Reddy ChemInform 20 (7), no-no, 1989 | 21 | 1989 |
Pyrazole derivatives as potent inhibitors of c-Jun N-terminal kinase: Synthesis and SAR studies A Doma, R Kulkarni, R Palakodety, GN Sastry, J Sridhara, A Garlapati Bioorganic & Medicinal Chemistry 22 (21), 6209-6219, 2014 | 16 | 2014 |
Topical advances in PIM kinases and their inhibitors: Medicinal chemistry perspectives V Walhekar, C Bagul, D Kumar, A Muthal, G Achaiah, R Kulkarni Biochimica et Biophysica Acta (BBA)-Reviews on Cancer 1877 (3), 188725, 2022 | 15 | 2022 |
Review on 2-substituted benzothiazoles: Diversity of synthetic methods and biological activities G Achaiah, NS Goud, KP Kumar, P Mayuri International Journal of Pharmaceutical Sciences and Research 7 (4), 1375, 2016 | 15 | 2016 |
Synthesis and cytotoxic activity of new chalcones and their flavonol derivatives RR Kotha, RG Kulkarni, AK Garige, SG Nerella, A Garlapati Med. Chem 7, 353-360, 2017 | 14 | 2017 |
Synthesis and biological activities of 3-[n-(4-oxo-2-substituted-3-quinazolinyl) formimidoyl] chromones G Achaiah, VM Reddy, VSAK Malla Reddy, K Shanker Indian J. Pharm. Sci 53, 253-5, 1991 | 13 | 1991 |
Design, synthesis and evaluation of new 2, 6-dihydroimidazo [1, 2-c] pyrimido [5, 4-e]-pyrimidine-5 (3H)-thiones as possible antihistaminic/antiasthmatic agents K Sirisha, G Achaiah, ARR Rao Indian journal of pharmaceutical sciences 76 (6), 519, 2014 | 12 | 2014 |