| Small heterocycles in multicomponent reactions BH Rotstein, S Zaretsky, V Rai, AK Yudin Chemical reviews 114 (16), 8323-8359, 2014 | 948 | 2014 |
| Decarboxylative Intramolecular Arene Alkylation Using N-(Acyloxy)phthalimides, an Organic Photocatalyst, and Visible Light TC Sherwood, HY Xiao, RG Bhaskar, EM Simmons, S Zaretsky, ... The Journal of Organic Chemistry 84 (13), 8360-8379, 2019 | 62 | 2019 |
| Passive membrane permeability of macrocycles can be controlled by exocyclic amide bonds JL Hickey, S Zaretsky, MA St. Denis, S Kumar Chakka, MM Morshed, ... Journal of medicinal chemistry 59 (11), 5368-5376, 2016 | 62 | 2016 |
| Exocyclic control of turn induction in macrocyclic peptide scaffolds. S Zaretsky, CCG Scully, AJ Lough, AK Yudin Chemistry-A European Journal 19 (52), 2013 | 59 | 2013 |
| Solid‐Phase Parallel Synthesis of Functionalised Medium‐to‐Large Cyclic Peptidomimetics through Three‐Component Coupling Driven by Aziridine Aldehyde Dimers AP Treder, JL Hickey, MCJ Tremblay, S Zaretsky, CCG Scully, J Mancuso, ... Chemistry–A European Journal 21 (25), 9249-9255, 2015 | 30 | 2015 |
| Mechanistic investigation of aziridine aldehyde-driven peptide macrocyclization: the imidoanhydride pathway S Zaretsky, JL Hickey, J Tan, D Pichugin, MAS Denis, S Ler, BKW Chung, ... Chemical Science 6 (10), 5446-5455, 2015 | 30 | 2015 |
| Bending rigid molecular rods: formation of oligoproline macrocycles CCG Scully, V Rai, G Poda, S Zaretsky, DC Burns, RS Houliston, T Lou, ... Chemistry–A European Journal 18 (49), 15612-15617, 2012 | 28 | 2012 |
| Rational design of calpain inhibitors based on calpastatin peptidomimetics KE Low, S Ler, KJ Chen, RL Campbell, JL Hickey, J Tan, CCG Scully, ... Journal of Medicinal Chemistry 59 (11), 5403-5415, 2016 | 26 | 2016 |
| Predicting performance of photochemical transformations for scaling up in different platforms by combining high-throughput experimentation with computational modeling M Sezen-Edmonds, JE Tabora, BM Cohen, S Zaretsky, EM Simmons, ... Organic Process Research & Development 24 (10), 2128-2138, 2020 | 25 | 2020 |
| Novel bisphosphonate inhibitors of the human farnesyl pyrophosphate synthase JW De Schutter, S Zaretsky, S Welbourn, A Pause, YS Tsantrizos Bioorganic & medicinal chemistry letters 20 (19), 5781-5786, 2010 | 24 | 2010 |
| Stereocontrolled disruption of the Ugi reaction toward the production of chiral piperazinones: substrate scope and process development S Zaretsky, S Adachi, BH Rotstein, JL Hickey, CCG Scully, JD St. Denis, ... The Journal of Organic Chemistry 79 (21), 9948-9957, 2014 | 20 | 2014 |
| Predicting cyclic peptide chemical shifts using quantum mechanical calculations S Zaretsky, JL Hickey, MAS Denis, CCG Scully, AL Roughton, DJ Tantillo, ... Tetrahedron 70 (42), 7655-7663, 2014 | 20 | 2014 |
| Bicycle synthesis through peptide macrocyclization using aziridine aldehydes followed by late stage disulfide bond installation BKW Chung, JL Hickey, CCG Scully, S Zaretsky, AK Yudin MedChemComm 4 (7), 1124-1128, 2013 | 20 | 2013 |
| L-Proline-Catalysed One-Pot aza-Diels–Alder Reaction in Water: Regioselective Synthesis of Spiro (isoxazolo [5, 4-b] pyridine-5, 5′-pyrimidine) Derivatives Y Dommaraju, S Borthakur, D Prajapati Synlett 29 (09), 1195-1198, 2018 | 18 | 2018 |
| Catalyst-free synthesis of fused triazolo-diazepino [5, 6-b] quinoline derivatives via a sequential Ugi-4CR–nucleophilic substitution–intramolecular Click reaction S Balalaie, A Vaezghaemi, N Zarezadeh, F Rominger, HR Bijanzadeh Synlett 29 (08), 1095-1101, 2018 | 17 | 2018 |
| Shifting the energy landscape of multicomponent reactions using aziridine aldehyde dimers: a mechanistic study L Belding, S Zaretsky, BH Rotstein, AK Yudin, T Dudding The Journal of Organic Chemistry 79 (20), 9465-9471, 2014 | 17 | 2014 |
| One-pot synthesis of [1, 2, 3] triazolo [1, 5-a] quinoxalin-4 (5H)-ones by a metal-free sequential ugi-4CR/alkyne–azide cycloaddition reaction YM Yan, HY Li, M Zhang, RX Wang, CG Zhou, ZX Ren, MW Ding Synlett 31 (01), 73-76, 2020 | 12 | 2020 |
| New Efficient Synthesis of 1, 2, 4-Trisubstituted Furans by a Sequential Passerini/Wittig/Isomerization Reaction Starting from Baylis–Hillman β-Bromo Aldehydes ZL Ren, M Sun, ZR Guan, MW Ding Synlett 29 (01), 106-110, 2018 | 12 | 2018 |
| Recent advances in the synthesis of cyclic pseudopeptides S Zaretsky, AK Yudin Drug Discovery Today: Technologies 26, 3-10, 2017 | 11 | 2017 |
| Twisted amide electrophiles enable cyclic peptide sequencing S Zaretsky, V Rai, G Gish, MW Forbes, M Kofler, CY Joy, J Tan, JL Hickey, ... Organic & Biomolecular Chemistry 13 (27), 7384-7388, 2015 | 11 | 2015 |
