PET Molecular Imaging in Drug Development: The Imaging and Chemistry Perspective SG Nerella, P Singh, T Sanam, CS Digwal Frontiers in Medicine 9, 2022 | 50 | 2022 |
Synthesis and carbonic anhydrase inhibition studies of sulfonamide based indole-1, 2, 3-triazole chalcone hybrids P Singh, B Swain, PS Thacker, DK Sigalapalli, PP Yadav, A Angeli, ... Bioorganic Chemistry 99, 103839, 2020 | 36 | 2020 |
Discovery of certain benzyl/phenethyl thiazolidinone-indole hybrids as potential anti-proliferative agents: Synthesis, molecular modeling and tubulin polymerization inhibition … DK Sigalapalli, V Pooladanda, P Singh, M Kadagathur, SD Guggilapu, ... Bioorganic Chemistry 92, 103188, 2019 | 36 | 2019 |
Anticancer carbonic anhydrase inhibitors: a patent and literature update 2018-2022 SG Nerella, P Singh, M Arifuddin, CT Supuran Expert Opinion on Therapeutic Patents 32 (8), 833-847, 2022 | 25 | 2022 |
Synthesis of a new series of 3-functionalised-1-phenyl-1, 2, 3-triazole sulfamoylbenzamides as carbonic anhydrase I, II, IV and IX inhibitors B Swain, A Angeli, S Angapelly, PS Thacker, P Singh, CT Supuran, ... Journal of Enzyme Inhibition and Medicinal Chemistry 34 (1), 1199-1209, 2019 | 21 | 2019 |
New coumarin/sulfocoumarin linked phenylacrylamides as selective transmembrane carbonic anhydrase inhibitors: Synthesis and in-vitro biological evaluation B Swain, A Angeli, P Singh, CT Supuran, M Arifuddin Bioorganic & Medicinal Chemistry 28 (15), 115586, 2020 | 15 | 2020 |
Synthesis and exploration of 2-morpholino-4-phenylthiazol-5-yl acrylamide derivatives for their effects against carbonic anhydrase I, II, IX and XII isoforms as a non … B Swain, CS Digwal, A Angeli, M Alvala, P Singh, CT Supuran, ... Bioorganic & Medicinal Chemistry 27 (21), 115090, 2019 | 14 | 2019 |
Coumarin‐Thiourea Hybrids Show Potent Carbonic Anhydrase IX and XIII Inhibitory Action PS Thacker, D Srikanth, A Angeli, P Singh, KK Chinchilli, M Arifuddin, ... ChemMedChem 16 (8), 1252-1256, 2021 | 13 | 2021 |
Discovery of a novel series of indolylchalcone-benzenesulfonamide hybrids acting as selective carbonic anhydrase II inhibitors P Singh, PP Yadav, B Swain, PS Thacker, A Angeli, CT Supuran, ... Bioorganic Chemistry 108, 104647, 2021 | 11 | 2021 |
Design and synthesis of benzenesulfonamide‐linked imidazo[2,1‐b][1,3,4]thiadiazole derivatives as carbonic anhydrase I and II inhibitors B Swain, K Aashritha, P Singh, A Angeli, A Kothari, DK Sigalapalli, ... Archiv der Pharmazie 354 (7), 2100028, 2021 | 9 | 2021 |
PET radiotracers and fluorescent probes for imaging human carbonic anhydrase IX and XII in hypoxic tumors SG Nerella, P Singh, PS Thacker, M Arifuddin, CT Supuran Bioorganic Chemistry, 106399, 2023 | 8 | 2023 |
Synthesis of a new series of quinoline/pyridine indole-3-sulfonamide hybrids as selective carbonic anhydrase IX inhibitors P Singh, NS Goud, B Swain, SK Sahoo, A Choli, A Angeli, BS Kushwah, ... Bioorganic & Medicinal Chemistry Letters 70, 128809, 2022 | 8 | 2022 |
Exploration of 2-phenylquinoline-4-carboxamide linked benzene sulfonamide derivatives as isoform selective inhibitors of transmembrane human carbonic anhydrases B Swain, SK Sahoo, P Singh, A Angeli, VM Yaddanapudi, CT Supuran, ... European Journal of Medicinal Chemistry 234, 114247, 2022 | 8 | 2022 |
Ureidosulfocoumarin Derivatives As Selective and Potent Carbonic Anhydrase IX and XII Inhibitors P Singh, D Kumar Sigalapalli, N Sridhar Goud, B Swain, S Kumar Sahoo, ... ChemMedChem 17 (5), e202100725, 2022 | 7 | 2022 |
Design and development of novel series of indole‐3‐sulfonamide ureido derivatives as selective carbonic anhydrase II inhibitors P Singh, A Choli, B Swain, A Angeli, SK Sahoo, VM Yaddanapudi, ... Archiv der Pharmazie 355 (1), 2100333, 2022 | 7 | 2022 |
3-Functionalised benzenesulphonamide based 1, 3, 4-oxadiazoles as selective carbonic anhydrase XIII inhibitors: Design, synthesis and biological evaluation B Swain, P Singh, A Angeli, K Aashritha, N Nagesh, CT Supuran, ... Bioorganic & Medicinal Chemistry Letters 37, 127856, 2021 | 7 | 2021 |
Microwave‐Assisted Copper‐Catalyzed One‐Pot Synthesis of 2‐Aryl/Heteroaryl‐4‐Quinolones via Sequential Intramolecular Aza‐Michael Addition and Oxidation P Singh, S Kumar Sahoo, N Sridhar Goud, B Swain, ... Asian Journal of Organic Chemistry 11 (7), e202200181, 2022 | 5 | 2022 |
Exploration of seryl tRNA synthetase to identify potent inhibitors against leishmanial parasites B Narsimulu, R Qureshi, P Jakkula, P Singh, M Arifuddin, IA Qureshi International Journal of Biological Macromolecules 237, 124118, 2023 | 4 | 2023 |
Isoxazole carboxylic acid methyl ester-based urea and thiourea derivatives as promising antitubercular agents SK Sahoo, O Ommi, S Maddipatla, P Singh, MN Ahmad, G Kaul, ... Molecular Diversity, 1-16, 2022 | 4 | 2022 |
Carbon-11 patents (2012–2022): synthetic methodologies and novel radiotracers for PET imaging SG Nerella, P Singh, S Tulja Expert Opinion on Therapeutic Patents 32 (7), 817-831, 2022 | 3 | 2022 |