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Deepak Shilkar
Deepak Shilkar
Cactus Communications
在 ucl.ac.uk 的电子邮件经过验证 - 首页
标题
引用次数
引用次数
年份
The Mycobactin biosynthesis pathway: A prospective therapeutic target in the battle against tuberculosis
M Shyam, D Shilkar, H Verma, A Dev, BN Sinha, F Brucoli, S Bhakta, ...
Journal of Medicinal Chemistry 64 (1), 71-100, 2020
432020
Non-carboxylic acid inhibitors of aldose reductase based on N-substituted thiazolidinedione derivatives
MUM Siddique, A Thakur, D Shilkar, S Yasmin, D Halakova, L Kovacikova, ...
European journal of medicinal chemistry 223, 113630, 2021
212021
Approaches for targeting the mycobactin biosynthesis pathway for novel anti-tubercular drug discovery: Where we stand
M Shyam, D Shilkar, G Rakshit, V Jayaprakash
Expert opinion on drug discovery 17 (7), 699-715, 2022
192022
A short survey of dengue protease inhibitor development in the past 6 years (2015–2020) with an emphasis on similarities between DENV and SARS-CoV-2 proteases
S Murtuja, D Shilkar, B Sarkar, BN Sinha, V Jayaprakash
Bioorganic & Medicinal Chemistry 49, 116415, 2021
132021
Anticancer agents based on Plastoquinone analogs with N-phenylpiperazine: Structure-activity relationship and mechanism of action in breast cancer cells
AT Jannuzzi, M Yıldız, N Bayrak, H Yıldırım, D Shilkar, V Jayaprakash, ...
Chemico-Biological Interactions 349, 109673, 2021
112021
Exploration of brominated Plastoquinone analogs: Discovery and structure-activity relationships of small antimicrobial lead molecules
M Yıldız, N Bayrak, H Yıldırım, E Mataracı-Kara, D Shilkar, V Jayaprakash, ...
Bioorganic Chemistry 116, 105316, 2021
72021
Carbonic anhydrase inhibitory activity of phthalimide-capped benzene sulphonamide derivatives
D Shilkar, MU Mohd Siddique, S Bua, S Yasmin, M Patil, AK Timiri, ...
Journal of Enzyme Inhibition and Medicinal Chemistry 38 (1), 2235089, 2023
62023
Brain permeable curcumin-based pyrazoline analogs: MAO inhibitory and antioxidant activity
VN Badavath, A Thakur, D Shilkar, C Nath, O Acevedo, G Ucar, ...
Journal of Molecular Structure 1268, 133681, 2022
52022
Aminated Quinolinequinones as Privileged Scaffolds for Antibacterial Agents: Synthesis, In Vitro Evaluation, and Putative Mode of Action
H Yıldırım, N Bayrak, M Yıldız, E Mataracı-Kara, S Korkmaz, D Shilkar, ...
ACS omega 7 (46), 41915-41928, 2022
52022
Highly Active Small Aminated Quinolinequinones against Drug-Resistant Staphylococcus aureus and Candida albicans
H Yıldırım, N Bayrak, M Yıldız, FN Yılmaz, E Mataracı-Kara, D Shilkar, ...
Molecules 27 (9), 2923, 2022
52022
Molecular determinants, clinical manifestations and effects of immunization on cardiovascular health during COVID-19 pandemic era-a review
A Chatterjee, R Saha, A Mishra, D Shilkar, V Jayaprakash, P Sharma, ...
Current Problems in Cardiology 48 (8), 101250, 2023
42023
UHPLC‐ESI‐QTOF‐MS/MS Based Identification, Quantification, and Assessment of in Silico Molecular Interactions of Major Phytochemicals from Bioactive Fractions of Clerodendrum …
P Kumar Deb, D Shilkar, B Sarkar
Chemistry & Biodiversity 19 (10), e202200617, 2022
42022
Exploring the anticancer effects of brominated plastoquinone analogs with promising cytotoxic activity in MCF-7 breast cancer cells via cell cycle arrest and oxidative stress …
AT Jannuzzi, AM Yilmaz Goler, N Bayrak, M Yıldız, H Yıldırım, ...
Pharmaceuticals 15 (7), 777, 2022
32022
Cytotoxic activity of quinolinequinones in cancer: In vitro studies, molecular docking, and ADME/PK profiling
AT Jannuzzi, AM Yilmaz Goler, D Shilkar, S Mondal, VN Basavanakatti, ...
Chemical Biology & Drug Design 102 (5), 1133-1154, 2023
22023
Discovery of quinolinequinones with N-phenylpiperazine by conversion of hydroxyquinoline as a new class of antimicrobial agents targeting resistant pathogenic microorganisms
M Yıldız, N Bayrak, H Yıldırım, SM Çakmak, FN Yılmaz, E Mataracı-Kara, ...
Bioorganic Chemistry 128, 106045, 2022
12022
A Critical Observation on the Design and Development of Reported Peptide Inhibitors of DENV NS2B-NS3 Protease in the Last Two Decades
S Murtuja, D Shilkar, B Sarkar, BN Sinha, V Jayaprakash
Mini Reviews in Medicinal Chemistry 22 (8), 1108-1130, 2022
2022
Identification of Dengue NS2B-NS3 Protease Inhibitors Through High-Throughput Virtual Screening—Impacts on Drug Development Against the Dengue Virus
S Murtuja, D Shilkar, B Sarkar, BN Sinha, V Jayaprakash
Human Viruses: Diseases, Treatments and Vaccines: The New Insights, 93-120, 2021
2021
Design and Development of Dengue Protease Inhibitors
M Sheikh, D Shilkar, V Jayaprakash, B Sarkar, BN Sinha
Proceedings of International Conference on Drug Discovery (ICDD), 2020
2020
Design and Development of Dengue NS5 Methyltransferase Inhibitors
S Kumari, MG Moazzam, D Shilkar, V Jayaprakash
Proceedings of International Conference on Drug Discovery (ICDD), 2020
2020
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