Development of novel pyridine-thiazole hybrid molecules as potential anticancer agents I Ivasechko, I Yushyn, P Roszczenko, J Senkiv, N Finiuk, D Lesyk, ... Molecules 27 (19), 6219, 2022 | 15 | 2022 |
Synthesis and Biological Activity Evaluation of Polyfunctionalized Anthraquinonehydrazones A Lozynskyi, S Holota, I Yushyn, O Sabadakh, O Karpenko, V Novikov, ... Letters in Drug Design & Discovery 18 (2), 199-209, 2021 | 10 | 2021 |
Synthesis of new structurally diverse thiazolidinone-derived compounds based on reaction of isorhodanine with ortho-substituted aldehydes, α-keto-and β-aroylacrylic acids A Lozynskyi, B Zimenkovsky, I Yushyn, D Kaminskyy, O Karpenko, ... Journal of Molecular Structure 1217, 128448, 2020 | 8 | 2020 |
Synthesis and Biological Activity Evaluation of Novel 5-Methyl-7-phenyl-3H-thiazolo[4,5-b]pyridin-2-ones A Lozynskyi, Y Konechnyi, J Senkiv, I Yushyn, D Khyluk, O Karpenko, ... Scientia Pharmaceutica 89 (4), 52, 2021 | 6 | 2021 |
Thiopyrano [2, 3-d] thiazole structures as promising scaffold with anticancer potential N Finiuk, N Zelisko, O Klyuchivska, I Yushyn, A Lozynskyi, A Cherniienko, ... Chemico-Biological Interactions 368, 110246, 2022 | 5 | 2022 |
Synthesis and structure elucidation of thiopyrano [2, 3-d] thiazole-6-carbonitriles as adducts of Michael reaction A Lozynskyi, I Yushyn, Y Shepeta, O Karpenko, AK Gzella, R Lesyk Journal of Molecular Structure 1256, 132574, 2022 | 5 | 2022 |
2,2-Dichloro-N-[5-[2-[3-(4-methoxyphenyl)-5-phenyl-3,4-dihydro-2H-pyrazol-2-yl]-2-oxoethyl]sulfanyl-1,3,4-thiadiazol-2-yl]acetamide I Yushyn, S Holota, R Lesyk Molbank 2022 (1), M1328, 2022 | 5 | 2022 |
N-(3-Cyano-4,5,6,7-tetrahydrobenzothiophen-2-yl)-2-[[5-[(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)amino]-1,3,4-thiadiazol-2-yl]sulfanyl]acetamide S Holota, I Yushyn, D Khyluk, R Vynnytska, R Lesyk Molbank 2021 (2), M1211, 2021 | 4 | 2021 |
Synthesis and evaluation of biological activity of 1-[2-amino-4-methylthiazol-5-yl]-3-arylpropenones AV Lozynskyi, IM Yushyn, YT Konechnyi, OM Roman, OV Matiykiv, ... Biopolymers and Cell, 389-399, 2021 | 3 | 2021 |
rel-2-[4-Chloro-2-[(5R,6R,7S)-6-[5-(4-methoxyphenyl)-3-(2-naphthyl)-3,4-dihydropyrazole-2-carbonyl]-5-methyl-2-oxo-3,5,6,7-tetrahydrothiopyrano[2,3-d]thiazol … I Yushyn, S Holota, O Ivantsiv, R Lesyk Molbank 2022 (3), M1410, 2022 | 1 | 2022 |
Influence of the 4-thiazolidinone derivative Les-6490 on the inflammatory process in rats compared to nimesulide. TM Rumynska, IM Yushyn, SM Holota, AR Hural, DV Mural, OV Dudok, ... Biopolymers & Cell 40 (2), 2024 | | 2024 |
A New 4-Thiazolidinone Derivative (Les-6490) as a Gut Microbiota Modulator: Antimicrobial and Prebiotic Perspectives Y Konechnyi, T Rumynska, I Yushyn, S Holota, V Turkina, M Ryviuk Rydel, ... Antibiotics 13 (4), 291, 2024 | | 2024 |
SYNTHESIS AND EVALUATION OF THE ANTICANCER ACTIVITY OF 2-AMINOISOINDOLE-THIZOLIDINONE HYBRIDS OMV Fedusevych, IM Yushyn, IL Demchuk, RB Lesyk | | 2023 |
3-(2-Diisopropylaminoethyl)-5-(4-methoxybenzylidene) thiazolidine-2, 4-dione S Holota, I Yushyn, A Gzella, R Lesyk Molbank 2022 (3), M1394, 2022 | | 2022 |
Синтез нових 5-заміщених 2-піразолілтіазол-4-онів як потенційних біологічно активних сполук IM Yushyn, AV Lozynskyi, OMV Fedusevych, OY Vovchuk, RB Lesyk Current issues in pharmacy and medicine: science and practice 13 (2), 2020 | | 2020 |
СИНТЕЗ ТА ОЦІНКА ПРОТИПУХЛОВОЇ АКТИВНОСТІ 2-АМІНОІЗОІНДОЛ ТІАЗОЛІДИНОНОВИХ ГІБРИДІВ OMV Fedusevych, IM Yushyn, IL Demchuk, RB Lesyk Фармацевтичний часопис, 5-11, 0 | | |