Covalent inhibitors of protein–protein interactions targeting lysine, tyrosine, or histidine residues L Gambini, C Baggio, P Udompholkul, J Jossart, AF Salem, JJP Perry, ... Journal of medicinal chemistry 62 (11), 5616-5627, 2019 | 113 | 2019 |
Brain–behavior correlates of optimizing learning through interleaved practice CHJ Lin, BJ Knowlton, MC Chiang, M Iacoboni, P Udompholkul, AD Wu Neuroimage 56 (3), 1758-1772, 2011 | 109 | 2011 |
Interleaved practice enhances skill learning and the functional connectivity of fronto‐parietal networks CH Lin, MC Chiang, BJ Knowlton, M Iacoboni, P Udompholkul, AD Wu Human brain mapping 34 (7), 1542-1558, 2013 | 86 | 2013 |
Reduction of circulating Cancer cells and metastases in breast-Cancer models by a potent EphA2-agonistic peptide–drug conjugate AF Salem, S Wang, S Billet, JF Chen, P Udompholkul, L Gambini, ... Journal of medicinal chemistry 61 (5), 2052-2061, 2018 | 64 | 2018 |
Age related differences in the neural substrates of motor sequence learning after interleaved and repetitive practice CHJ Lin, MC Chiang, AD Wu, M Iacoboni, P Udompholkul, ... Neuroimage 62 (3), 2007-2020, 2012 | 62 | 2012 |
Aryl-fluorosulfate-based lysine covalent pan-inhibitors of apoptosis protein (IAP) antagonists with cellular efficacy C Baggio, P Udompholkul, L Gambini, AF Salem, J Jossart, JJP Perry, ... Journal of medicinal chemistry 62 (20), 9188-9200, 2019 | 51 | 2019 |
Contextual interference effects in sequence learning for young and older adults. CHJ Lin, AD Wu, P Udompholkul, BJ Knowlton Psychology and aging 25 (4), 929, 2010 | 50 | 2010 |
Design of potent pan-IAP and Lys-covalent XIAP selective inhibitors using a thermodynamics driven approach C Baggio, L Gambini, P Udompholkul, AF Salem, A Aronson, A Dona, ... Journal of medicinal chemistry 61 (14), 6350-6363, 2018 | 44 | 2018 |
Design, synthesis, and structural characterization of lysine covalent BH3 peptides targeting Mcl-1 L Gambini, P Udompholkul, C Baggio, A Muralidharan, N Kenjić, Z Assar, ... Journal of medicinal chemistry 64 (8), 4903-4912, 2021 | 28 | 2021 |
Structure-Based Design of Novel EphA2 Agonistic Agents with Nanomolar Affinity in Vitro and in Cell L Gambini, AF Salem, P Udompholkul, XF Tan, C Baggio, N Shah, ... ACS chemical biology 13 (9), 2633-2644, 2018 | 28 | 2018 |
Enhanced motor learning in older adults is accompanied by increased bilateral frontal and fronto-parietal connectivity CHJ Lin, MC Chiang, AD Wu, M Iacoboni, P Udompholkul, ... Brain connectivity 2 (2), 56-68, 2012 | 28 | 2012 |
Stability and cell permeability of sulfonyl fluorides in the design of Lys‐covalent antagonists of protein‐protein interactions L Gambini, P Udompholkul, AF Salem, C Baggio, M Pellecchia ChemMedChem 15 (22), 2176-2184, 2020 | 19 | 2020 |
Enthalpy-based screening of focused combinatorial libraries for the identification of potent and selective ligands C Baggio, P Udompholkul, E Barile, M Pellecchia ACS Chemical Biology 12 (12), 2981-2989, 2017 | 18 | 2017 |
Lysine covalent antagonists of melanoma inhibitors of apoptosis protein P Udompholkul, C Baggio, L Gambini, G Alboreggia, M Pellecchia Journal of Medicinal Chemistry 64 (21), 16147-16158, 2021 | 17 | 2021 |
Characterization of a Potent and Orally Bioavailable Lys-Covalent Inhibitor of Apoptosis Protein (IAP) Antagonist P Udompholkul, A Garza-Granados, G Alboreggia, C Baggio, J McGuire, ... Journal of Medicinal Chemistry 66 (12), 8159-8169, 2023 | 14 | 2023 |
Targefrin: a potent agent targeting the ligand binding domain of EphA2 C Baggio, P Udompholkul, L Gambini, M Pellecchia Journal of Medicinal Chemistry 65 (22), 15443-15456, 2022 | 11 | 2022 |
Therapeutic targeting of pancreatic cancer via EphA2 dimeric agonistic agents AF Salem, L Gambini, P Udompholkul, C Baggio, M Pellecchia Pharmaceuticals 13 (5), 90, 2020 | 11 | 2020 |
N‐locking stabilization of covalent helical peptides: Application to Bfl‐1 antagonists C Baggio, P Udompholkul, L Gambini, J Jossart, AF Salem, M Håkansson, ... Chemical biology & drug design 95 (4), 412-426, 2020 | 8 | 2020 |
Effective Tumor Targeting by EphA2-Agonist-Biotin-Streptavidin Conjugates P Udompholkul, C Baggio, L Gambini, Y Sun, M Zhao, RM Hoffman, ... Molecules 26 (12), 3687, 2021 | 5 | 2021 |
Mixture-Based Screening of Focused Combinatorial Libraries by Nmr: Application to the Antiapoptotic Protein Hmcl-1 G Alboreggia, P Udompholkul, C Baggio, M Pellecchia Journal of Medicinal Chemistry 66 (14), 10108-10118, 2023 | 3 | 2023 |