From inhibition to degradation: targeting the antiapoptotic protein myeloid cell leukemia 1 (MCL1) JW Papatzimas, E Gorobets, R Maity, MI Muniyat, JL MacCallum, P Neri, ... Journal of medicinal chemistry 62 (11), 5522-5540, 2019 | 93 | 2019 |
Rational chemical design of molecular glue degraders ES Toriki, JW Papatzimas, K Nishikawa, D Dovala, AO Frank, MJ Hesse, ... ACS central science 9 (5), 915-926, 2023 | 65 | 2023 |
Thiaporphyrin-mediated photocatalysis using red light JG Lee, JW Papatzimas, AD Bromby, E Gorobets, DJ Derksen RSC advances 6 (64), 59269-59272, 2016 | 30 | 2016 |
A facile synthesis of ligands for the von Hippel–Lindau E3 ligase C Steinebach, SA Voell, LP Vu, A Bricelj, I Sosič, G Schnakenburg, ... Synthesis 52 (17), 2521-2527, 2020 | 26 | 2020 |
ADAM protease inhibition overcomes resistance of breast cancer stem-like cells to γδ T cell immunotherapy I Dutta, D Dieters-Castator, JW Papatzimas, A Medina, J Schueler, ... Cancer letters 496, 156-168, 2021 | 15 | 2021 |
A general strategy for the preparation of thalidomide-conjugate linkers JW Papatzimas, E Gorobets, DK Brownsey, R Maity, NJ Bahlis, ... Synlett 28 (20), 2881-2885, 2017 | 14 | 2017 |
DCAF16-Based Covalent Handle for the Rational Design of Monovalent Degraders M Lim, TD Cong, LM Orr, ES Toriki, AC Kile, JW Papatzimas, E Lee, Y Lin, ... ACS Central Science, 2024 | 5 | 2024 |
Identification of ligand linkage vectors for the development of p300/CBP degraders DK Brownsey, BC Rowley, E Gorobets, K Mihara, R Maity, JW Papatzimas, ... RSC Medicinal Chemistry 13 (6), 726-730, 2022 | 4 | 2022 |
A vinylogous Norrish reaction as a strategy for light-mediated ring expansion E Gorobets, JW Papatzimas, J Dourado, G Yousefalizadeh, JG Lee, ... Chemical Communications 58 (17), 2910-2913, 2022 | 3 | 2022 |
Sulfamoyl benzene derivatives and uses thereof T Trang, DJ Derksen, K Navis, E Gorobets, J Papatzimas US Patent App. 18/024,443, 2024 | | 2024 |
Correction to “Rational Chemical Design of Molecular Glue Degraders” ES Toriki, JW Papatzimas, K Nishikawa, D Dovala, AO Frank, MJ Hesse, ... ACS Central Science 9 (8), 1702-1702, 2023 | | 2023 |
Correction to “Rational Chemical Design of Molecular Glue Degraders” DK Nomura, ES Toriki, JW Papatzimas, K Nishikawa, D Dovala, AO Frank, ... ACS Central Science 9 (8), , 1702, 2023 | | 2023 |
Rational Chemical Design of Molecular Glue Degraders J McKenna, D Dovala, A Frank, M Hesse, J Song, M Bruce-Smythe, ... ACS Central Science, 2023 | | 2023 |
Synthesis and Biological Evaluation of Heterobifunctional Small Molecules for Proteasome-Mediated Protein Degradation of Myeloid Cell Leukemia 1 (MCL1) JW Papatzimas Synthesis 2020, 09-14, 2020 | | 2020 |