| Vascular endothelial growth factor (VEGF) receptors: drugs and new inhibitors F Musumeci, M Radi, C Brullo, S Schenone Journal of medicinal chemistry 55 (24), 10797-10822, 2012 | 194 | 2012 |
| ATP-competitive inhibitors of mTOR: an update S Schenone, C Brullo, F Musumeci, M Radi, M Botta Current medicinal chemistry 18 (20), 2995-3014, 2011 | 158 | 2011 |
| Biologically Driven Synthesis of Pyrazolo[3,4-d]pyrimidines As Protein Kinase Inhibitors: An Old Scaffold As a New Tool for Medicinal Chemistry and Chemical … S Schenone, M Radi, F Musumeci, C Brullo, M Botta Chemical reviews 114 (14), 7189-7238, 2014 | 141 | 2014 |
| Design, Synthesis, Biological Activity, and ADME Properties of Pyrazolo[3,4-d]pyrimidines Active in Hypoxic Human Leukemia Cells: A Lead Optimization Study M Radi, E Dreassi, C Brullo, E Crespan, C Tintori, V Bernardo, M Valoti, ... Journal of medicinal chemistry 54 (8), 2610-2626, 2011 | 95 | 2011 |
| Novel dual Src/Abl inhibitors for hematologic and solid malignancies S Schenone, C Brullo, F Musumeci, M Botta Expert opinion on investigational drugs 19 (8), 931-945, 2010 | 91 | 2010 |
| Fyn kinase in brain diseases and cancer: the search for inhibitors S Schenone, C Brullo, F Musumeci, M Biava, F Falchi, M Botta Current medicinal chemistry 18 (19), 2921-2942, 2011 | 78 | 2011 |
| Combining X-ray Crystallography and Molecular Modeling toward the Optimization of Pyrazolo[3,4-d]pyrimidines as Potent c-Src Inhibitors Active in Vivo against … C Tintori, AL Fallacara, M Radi, C Zamperini, E Dreassi, E Crespan, ... Journal of Medicinal Chemistry 58 (1), 347-361, 2015 | 75 | 2015 |
| SI113, a SGK1 inhibitor, potentiates the effects of radiotherapy, modulates the response to oxidative stress and induces cytotoxic autophagy in human glioblastoma multiforme cells C Talarico, V Dattilo, L D'Antona, A Barone, N Amodio, S Belviso, ... Oncotarget 7 (13), 15868, 2016 | 69 | 2016 |
| SI113, a specific inhibitor of the Sgk1 kinase activity that counteracts cancer cell proliferation L D''antona, R Amato, C Talarico, F Ortuso, M Menniti, V Dattilo, R Iuliano, ... Cellular physiology and biochemistry 35 (5), 2006-2018, 2015 | 62 | 2015 |
| An update on dual Src/Abl inhibitors F Musumeci, S Schenone, C Brullo, M Botta Future medicinal chemistry 4 (6), 799-822, 2012 | 62 | 2012 |
| A1 receptors ligands: past, present and future trends S Schenone, C Brullo, F Musumeci, O Bruno, M Botta Current topics in medicinal chemistry 10 (9), 878-901, 2010 | 61 | 2010 |
| Pruritus characteristics in a large Italian cohort of psoriatic patients G Damiani, S Cazzaniga, RR Conic, L Naldi, Psocare Registry Network, ... Journal of the European Academy of Dermatology and Venereology 33 (7), 1316-1324, 2019 | 58 | 2019 |
| Identification of potent c-Src inhibitors strongly affecting the proliferation of human neuroblastoma cells M Radi, C Brullo, E Crespan, C Tintori, F Musumeci, M Biava, S Schenone, ... Bioorganic & medicinal chemistry letters 21 (19), 5928-5933, 2011 | 55 | 2011 |
| Latent tuberculosis infection in patients with chronic plaque psoriasis: evidence from the Italian Psocare Registry P Gisondi, S Cazzaniga, S Chimenti, M Maccarone, M Picardo, ... British Journal of Dermatology 172 (6), 1613-1620, 2015 | 51 | 2015 |
| Design, Synthesis, and Biological Evaluation of Pyrazolo[3,4-d]pyrimidines Active in Vivo on the Bcr-Abl T315I Mutant M Radi, C Tintori, F Musumeci, C Brullo, C Zamperini, E Dreassi, ... Journal of Medicinal Chemistry 56 (13), 5382-5394, 2013 | 49 | 2013 |
| In silico identification and biological evaluation of novel selective serum/glucocorticoid-inducible kinase 1 inhibitors based on the pyrazolo-pyrimidine scaffold F Ortuso, R Amato, A Artese, L D’antona, G Costa, C Talarico, F Gigliotti, ... Journal of chemical information and modeling 54 (7), 1828-1832, 2014 | 43 | 2014 |
| The SGK1 Kinase Inhibitor SI113 Sensitizes Theranostic Effects of the 64CuCl2 in Human Glioblastoma Multiforme Cells G Catalogna, C Talarico, V Dattilo, V Gangemi, F Calabria, L D’Antona, ... Cellular Physiology and Biochemistry 43 (1), 108-119, 2017 | 41 | 2017 |
| Studies on the ATP binding site of Fyn kinase for the identification of new inhibitors and their evaluation as potential agents against tauopathies and tumors C Tintori, G La Sala, G Vignaroli, L Botta, AL Fallacara, F Falchi, M Radi, ... Journal of Medicinal Chemistry 58 (11), 4590-4609, 2015 | 39 | 2015 |
| Recent studies on ponatinib in cancers other than chronic myeloid leukemia F Musumeci, C Greco, G Grossi, A Molinari, S Schenone Cancers 10 (11), 430, 2018 | 35 | 2018 |
| Click chemistry, a potent tool in medicinal sciences F Musumeci, S Schenone, A Desogus, E Nieddu, D Deodato, L Botta Current Medicinal Chemistry 22 (17), 2022-2050, 2015 | 35 | 2015 |
