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Simone Giovannuzzi
Simone Giovannuzzi
Post-doctoral Researcher, University of Florence
在 unifi.it 的电子邮件经过验证
标题
引用次数
引用次数
年份
Coumarins effectively inhibit bacterial α-carbonic anhydrases
S Giovannuzzi, CS Hewitt, A Nocentini, C Capasso, DP Flaherty, ...
Journal of Enzyme Inhibition and Medicinal Chemistry 37 (1), 333-338, 2022
312022
Inhibition studies of bacterial α-carbonic anhydrases with phenols
S Giovannuzzi, CS Hewitt, A Nocentini, C Capasso, G Costantino, ...
Journal of Enzyme Inhibition and Medicinal Chemistry 37 (1), 666-671, 2022
222022
Dithiocarbamates effectively inhibit the α-carbonic anhydrase from Neisseria gonorrhoeae
S Giovannuzzi, NS Abutaleb, CS Hewitt, F Carta, A Nocentini, MN Seleem, ...
Journal of Enzyme Inhibition and Medicinal Chemistry 37 (1), 1-8, 2022
212022
4-(3-Alkyl/benzyl-guanidino) benzenesulfonamides as selective carbonic anhydrase VII inhibitors
M Abdoli, S Giovannuzzi, CT Supuran, R Žalubovskis
Journal of Enzyme Inhibition and Medicinal Chemistry 37 (1), 1568-1576, 2022
162022
Aromatic sulfonamides including a sulfonic acid tail: new membrane impermeant carbonic anhydrase inhibitors for targeting selectively the cancer-associated isoforms
S Giovannuzzi, M D’Ambrosio, C Luceri, SM Osman, M Pallecchi, ...
International Journal of Molecular Sciences 23 (1), 461, 2021
152021
May Sulfonamide Inhibitors of Carbonic Anhydrases from Mammaliicoccus sciuri Prevent Antimicrobial Resistance Due to Gene Transfer to Other Harmful …
V De Luca, S Giovannuzzi, CT Supuran, C Capasso
International Journal of Molecular Sciences 23 (22), 13827, 2022
122022
Coumarins inhibit η-class carbonic anhydrase from Plasmodium falciparum
S Giovannuzzi, V De Luca, A Nocentini, C Capasso, CT Supuran
Journal of Enzyme Inhibition and Medicinal Chemistry 37 (1), 680-685, 2022
112022
Discovery of indolinone-bearing benzenesulfonamides as new dual carbonic anhydrase and VEGFR-2 inhibitors possessing anticancer and pro-apoptotic properties
S Saied, M Shaldam, MM Elbadawi, S Giovannuzzi, A Nocentini, ...
European Journal of Medicinal Chemistry 259, 115707, 2023
92023
1, 5-diaryl-1, 2, 4-triazole ureas as new SLC-0111 analogues endowed with dual carbonic anhydrase and VEGFR-2 inhibitory activities
AE Elsawi, MM Elbadawi, A Nocentini, H Almahli, S Giovannuzzi, ...
Journal of Medicinal Chemistry 66 (15), 10558-10578, 2023
92023
Continued structural exploration of sulfocoumarin as selective inhibitor of tumor-associated human carbonic anhydrases ix and XII
S Giovannuzzi, C Capasso, A Nocentini, CT Supuran
Molecules 27 (13), 4076, 2022
72022
Inhibition of pathogenic bacterial carbonic anhydrases by monothiocarbamates
S Giovannuzzi, AK Marapaka, NS Abutaleb, F Carta, HW Liang, ...
Journal of Enzyme Inhibition and Medicinal Chemistry 38 (1), 2284119, 2023
62023
Inhibition studies with simple and complex (in)organic anions of the γ-carbonic anhydrase from Mammaliicoccus (Staphylococcus) sciuri, MscCAγ
S Giovannuzzi, V De Luca, C Capasso, CT Supuran
Journal of Enzyme Inhibition and Medicinal Chemistry 38 (1), 2173748, 2023
52023
Boron-containing carbonic anhydrases inhibitors
S Giovannuzzi, A Nikitjuka, BRP Resende, M Smietana, A Nocentini, ...
Bioorganic Chemistry, 106976, 2023
42023
Potent inhibitors of tumor associated carbonic anhydrases endowed with cathepsin B inhibition
A Kumar, P Arya, V Sharma, S Giovannuzzi, N Raghav, CT Supuran, ...
Archiv der Pharmazie 356 (11), 2300349, 2023
42023
Development of Penicillin-Based Carbonic Anhydrase Inhibitors Targeting Multidrug-Resistant Neisseria gonorrhoeae
A Bonardi, A Nocentini, S Giovannuzzi, N Paoletti, A Ammara, S Bua, ...
Journal of Medicinal Chemistry, 2024
32024
Identification of thienopyrimidine derivatives tethered with sulfonamide and other moieties as carbonic anhydrase inhibitors: design, synthesis and anti-proliferative activity
S Higazy, N Samir, A El-Khouly, S Giovannuzzi, P Begines, HM Gaber, ...
Bioorganic Chemistry 144, 107089, 2024
32024
Potent and selective carbonic anhydrase inhibition activities of pyrazolones bearing benzenesulfonamides
S Akocak, N Lolak, S Giovannuzzi, CT Supuran
Bioorganic & Medicinal Chemistry Letters 95, 129479, 2023
32023
Discovery and Mechanistic Studies of Dual-Target Hits for Carbonic Anhydrase IX and VEGFR-2 as Potential Agents for Solid Tumors: X-ray, In Vitro, In Vivo, and In Silico …
SM Hefny, TF El-Moselhy, N El-Din, S Giovannuzzi, T Bin Traiki, ...
Journal of Medicinal Chemistry 67 (9), 7406-7430, 2024
22024
1, 2, 3‐Triazole‐based esters and carboxylic acids as nonclassical carbonic anhydrase inhibitors capable of cathepsin B inhibition
K Siwach, M Rani, L Vats, S Giovannuzzi, AK Paul, M Brahma, N Kumari, ...
Archiv der Pharmazie 357 (3), 2300372, 2024
22024
Design and synthesis of sulfonamides incorporating a biotin moiety: Carbonic anhydrase inhibitory effects, antiproliferative activity and molecular modeling studies
P Begines, A Bonardi, A Nocentini, P Gratteri, S Giovannuzzi, R Ronca, ...
Bioorganic & Medicinal Chemistry 94, 117467, 2023
22023
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