| “A sweet combination”: developing saccharin and acesulfame K structures for selectively targeting the tumor-associated carbonic anhydrases IX and XII S Bua, C Lomelino, AB Murray, SM Osman, ZA ALOthman, M Bozdag, ... Journal of Medicinal Chemistry 63 (1), 321-333, 2019 | 29 | 2019 |
| (+)-Catharanthine potentiates the GABAA receptor by binding to a transmembrane site at the β (+)/α (-) interface near the TM2-TM3 loop HR Arias, CM Borghese, AL Germann, SR Pierce, A Bonardi, A Nocentini, ... Biochemical pharmacology 199, 114993, 2022 | 2 | 2022 |
| 1, 2, 3-Benzoxathiazine-2, 2-dioxides–effective inhibitors of human carbonic anhydrases J Ivanova, M Abdoli, A Nocentini, R Žalubovskis, CT Supuran Journal of Enzyme Inhibition and Medicinal Chemistry 38 (1), 225-238, 2023 | 14 | 2023 |
| 1, 5-diaryl-1, 2, 4-triazole ureas as new SLC-0111 analogues endowed with dual carbonic anhydrase and VEGFR-2 inhibitory activities AE Elsawi, MM Elbadawi, A Nocentini, H Almahli, S Giovannuzzi, ... Journal of Medicinal Chemistry 66 (15), 10558-10578, 2023 | 9 | 2023 |
| 1, 5‐Benzodiazepines as a platform for the design of carbonic anhydrase inhibitors C Ismail, A Nocentini, CT Supuran, JY Winum, R Gharbi Archiv der Pharmazie 355 (3), 2100405, 2022 | 4 | 2022 |
| 2-(2-Hydroxyethyl) piperazine derivatives as potent human carbonic anhydrase inhibitors: Synthesis, enzyme inhibition, computational studies and antiglaucoma activity N Chiaramonte, A Angeli, S Sgambellone, A Bonardi, A Nocentini, ... European Journal of Medicinal Chemistry 228, 114026, 2022 | 2 | 2022 |
| 2-Aminobenzoxazole-appended coumarins as potent and selective inhibitors of tumour-associated carbonic anhydrases A Fuentes-Aguilar, P Merino-Montiel, S Montiel-Smith, S Meza-Reyes, ... Journal of Enzyme Inhibition and Medicinal Chemistry 37 (1), 168-177, 2022 | 16 | 2022 |
| 2-Benzylpiperazine: A new scaffold for potent human carbonic anhydrase inhibitors. Synthesis, enzyme inhibition, enantioselectivity, computational and crystallographic studies … N Chiaramonte, S Bua, M Ferraroni, A Nocentini, A Bonardi, G Bartolucci, ... European Journal of Medicinal Chemistry 151, 363-375, 2018 | 49 | 2018 |
| 3H-1,2-Benzoxaphosphepine 2-oxides as selective inhibitors of carbonic anhydrase IX and XII A Pustenko, A Balašova, A Nocentini, CT Supuran, R Žalubovskis Journal of Enzyme Inhibition and Medicinal Chemistry 38 (1), 216-224, 2023 | 5 | 2023 |
| 3-Hydrazinoisatin-based benzenesulfonamides as novel carbonic anhydrase inhibitors endowed with anticancer activity: Synthesis, in vitro biological evaluation and in silico … MF Abo-Ashour, WM Eldehna, A Nocentini, A Bonardi, S Bua, HS Ibrahim, ... European Journal of Medicinal Chemistry 184, 111768, 2019 | 74 | 2019 |
| 3-Methylthiazolo [3, 2-a] benzimidazole-benzenesulfonamide conjugates as novel carbonic anhydrase inhibitors endowed with anticancer activity: Design, synthesis, biological and … AAM Alkhaldi, MM Al-Sanea, A Nocentini, WM Eldehna, ZM Elsayed, ... European Journal of Medicinal Chemistry 207, 112745, 2020 | 53 | 2020 |
| 4-(3-Phenyl-4-(3,4,5-trimethoxybenzoyl)-1H-pyrrol-1-yl)benzenesulfonamide, a Novel Carbonic Anhydrase and Wnt/β-Catenin Signaling Pathway Dual-Targeting … D Masci, M Puxeddu, L Di Magno, M D’Ambrosio, A Parisi, M Nalli, R Bai, ... Journal of Medicinal Chemistry 66 (21), 14824-14842, 2023 | 1 | 2023 |
| 4-(5-Amino-pyrazol-1-yl) benzenesulfonamide derivatives as novel multi-target anti-inflammatory agents endowed with inhibitory activity against COX-2, 5-LOX and carbonic … MA Ragab, WM Eldehna, A Nocentini, A Bonardi, HE Okda, B Elgendy, ... European Journal of Medicinal Chemistry 250, 115180, 2023 | 19 | 2023 |
| 4-Hydroxy-3-nitro-5-ureido-benzenesulfonamides selectively target the tumor-associated carbonic anhydrase isoforms IX and XII showing hypoxia-enhanced antiproliferative profiles A Nocentini, E Trallori, S Singh, CL Lomelino, G Bartolucci, ... Journal of Medicinal Chemistry 61 (23), 10860-10874, 2018 | 60 | 2018 |
| 4-Substituted benzenesulfonamides featuring cyclic imides moieties exhibit potent and isoform-selective carbonic anhydrase II/IX inhibition AM Alaa, AS El-Azab, AH Ghiaty, P Gratteri, CT Supuran, A Nocentini Bioorganic Chemistry 83, 198-204, 2019 | 25 | 2019 |
| 5-(Sulfamoyl) thien-2-yl 1, 3-oxazole inhibitors of carbonic anhydrase II with hydrophilic periphery S Kalinin, A Kovalenko, A Valtari, A Nocentini, M Gureev, A Urtti, ... Journal of Enzyme Inhibition and Medicinal Chemistry 37 (1), 1005-1011, 2022 | 7 | 2022 |
| 6-Substituted Triazolyl Benzoxaboroles as Selective Carbonic Anhydrase Inhibitors: In Silico Design, Synthesis, and X-ray Crystallography A Nocentini, A Bonardi, C Bazzicalupi, V Alterio, D Esposito, SM Monti, ... Journal of Medicinal Chemistry 66 (12), 8118-8129, 2023 | 3 | 2023 |
| 7-Acylamino-3H-1, 2-benzoxathiepine 2, 2-dioxides as new isoform-selective carbonic anhydrase IX and XII inhibitors A Pustenko, A Nocentini, A Balašova, M Krasavin, R Žalubovskis, ... Journal of enzyme inhibition and medicinal chemistry 35 (1), 650-656, 2020 | 14 | 2020 |
| 7-Aryl-triazolyl-substituted sulfocoumarins are potent, selective inhibitors of the tumor-associated carbonic anhydrase IX and XII A Nocentini, M Ceruso, F Carta, CT Supuran Journal of Enzyme Inhibition and Medicinal Chemistry 31 (6), 1226-1233, 2016 | 49 | 2016 |
| A new kid on the block? Carbonic anhydrases as possible new targets in Alzheimer’s disease G Provensi, F Carta, A Nocentini, CT Supuran, F Casamenti, MB Passani, ... International journal of molecular sciences 20 (19), 4724, 2019 | 73 | 2019 |
PAOLA GRATTERIDepartment NEUROFARBA - Pharmaceutical and nutraceutical section在 unifi.it 的电子邮件经过验证
