| Chimeric RXFP1 and RXFP2 receptors highlight the similar mechanism of activation utilizing their N-terminal low-density lipoprotein class A modules S Bruell, RCK Kong, EJ Petrie, B Hoare, JD Wade, DJ Scott, PR Gooley, ... Frontiers in Endocrinology 4, 171, 2013 | 27 | 2013 |
| Detection of cannabinoid receptor type 2 in native cells and zebrafish with a highly potent, cell-permeable fluorescent probe T Gazzi, B Brennecke, K Atz, C Korn, D Sykes, G Forn-Cuni, P Pfaff, ... Chemical Science 13 (19), 5539-5545, 2022 | 20 | 2022 |
| Multi-component mechanism of H2 Relaxin binding to RXFP1 through NanoBRET kinetic analysis BL Hoare, S Bruell, A Sethi, PR Gooley, MJ Lew, MA Hossain, A Inoue, ... IScience 11, 93-113, 2019 | 19 | 2019 |
| Using the novel HiBiT tag to label cell surface relaxin receptors for BRET proximity analysis BL Hoare, M Kocan, S Bruell, DJ Scott, RAD Bathgate Pharmacology Research & Perspectives 7 (4), e00513, 2019 | 12 | 2019 |
| Functional solubilization of the β2-adrenoceptor using diisobutylene maleic acid CR Harwood, DA Sykes, BL Hoare, FM Heydenreich, R Uddin, ... Iscience 24 (12), 2021 | 9 | 2021 |
| A real-time, plate-based BRET assay for detection of cGMP in primary cells AL Valkovic, M Kocan, B Hoare, S Marshall, DJ Scott, RAD Bathgate International Journal of Molecular Sciences 23 (3), 1908, 2022 | 4 | 2022 |
| Bi-allelic variants in INSL3 and RXFP2 cause bilateral cryptorchidism and male infertility AK Dicke, J Albrethsen, BL Hoare, MJ Wyrwoll, AS Busch, D Fietz, A Pilatz, ... Human Reproduction 38 (7), 1412-1423, 2023 | 3 | 2023 |
| Measurement of non-purified GPCR thermostability using the homogenous ThermoBRET assay BL Hoare, A Kaur, CR Harwood, NC Dijon, ND Holliday, DA Sykes, ... bioRxiv, 2020.08. 05.237982, 2020 | 2 | 2020 |
| Development of a synthetic relaxin-3/INSL5 chimeric peptide ligand for NanoBiT complementation binding assays H Wu, BL Hoare, TNG Handley, MA Hossain, RAD Bathgate Biochemical Pharmacology 224, 116238, 2024 | 1 | 2024 |
| Activation of Multiple G Protein Pathways to Characterize the Five Dopamine Receptor Subtypes Using Bioluminescence Technology D Mönnich, LJ Humphrys, C Höring, BL Hoare, L Forster, S Pockes ACS Pharmacology & Translational Science 7 (3), 834-854, 2024 | 1 | 2024 |
| ThermoBRET: A Ligand‐Engagement Nanoscale Thermostability Assay Applied to GPCRs BL Hoare, DN Tippett, A Kaur, SA Cullum, T Miljuš, EJ Koers, ... ChemBioChem 25 (2), e202300459, 2024 | 1* | 2024 |
| Kinetic Profiling of Ligands and Fragments Binding to GPCRs by TR-FRET DA Sykes, L Borrega-Roman, CR Harwood, B Hoare, JM Lochray, ... Biophysical and Computational Tools in Drug Discovery, 1-32, 2021 | 1 | 2021 |
| Developing insulin-like peptide 5-based antagonists for the G protein-coupled receptor, RXFP4 H Wu, TNG Handley, BL Hoare, HA Hartono, DJ Scott, DK Chalmers, ... Biochemical Pharmacology 224, 116239, 2024 | | 2024 |
| Long-Circulating Vasoactive 1, 18-Octadecanedioic Acid–Terlipressin Conjugate O Berger, W Choi, CH Ko, MP Thompson, MJ Avram, DJ Scott, BL Hoare, ... ACS Pharmacology & Translational Science 7 (5), 1252-1261, 2024 | | 2024 |
| A universal cannabinoid CB1 and CB2 receptor TR-FRET kinetic ligand binding assay. L Borrega-Roman, BL Hoare, M Kosar, RC Sarott, KJ Patej, J Bouma, ... bioRxiv, 2024.07. 16.603654, 2024 | | 2024 |
| Development and application of a kinetic ligand binding assay for the cannabinoid receptor 1 using resonance energy transfer approaches B Hoare, D Sykes, T Gazzi, M Nazare, U Grether, D Veprintsev BRITISH JOURNAL OF PHARMACOLOGY 177 (11), 2528-2529, 2020 | | 2020 |
| Drug Derived Fluorescent Probes for the Specific Visualization of Cannabinoid Type 2 Receptor-A Toolbox Approach B Brennecke, K Atz, C Korn, D Sykes, RC Sarott, MV Westphal, P Pfaff, ... | | 2019 |
