The benzazole scaffold: a SWAT to combat Alzheimer's disease S Noel, S Cadet, E Gras, C Hureau Chemical Society Reviews 42 (19), 7747-7762, 2013 | 207 | 2013 |
Potent acetylcholinesterase inhibitors: design, synthesis and structure–activity relationships of alkylene linked bis-galanthamine and galanthamine–galanthaminium salts C Guillou, A Mary, DZ Renko, E Gras, C Thal Bioorganic & Medicinal Chemistry Letters 10 (7), 637-639, 2000 | 129 | 2000 |
An Efficient Total Synthesis of (+/-)-Galanthamine We are grateful to the CNRS for financial support, and the French Ministry of Education and Research for Ph. D grants to JLB … C Guillou, JL Beunard, E Gras, C Thal Angewandte Chemie (International ed. in English) 40 (24), 4745-4746, 2001 | 114 | 2001 |
Thioflavin derivatives as markers for amyloid‐β fibrils: insights into structural features important for high‐affinity binding R Leuma Yona, S Mazères, P Faller, E Gras ChemMedChem: Chemistry Enabling Drug Discovery 3 (1), 63-66, 2008 | 87 | 2008 |
Recent developments in the chemistry of lithiated epoxides DM Hodgson, E Gras Synthesis 2002 (12), 1625-1642, 2002 | 75 | 2002 |
Coordination complexes and biomolecules: A wise wedding for catalysis upgrade M Hoarau, C Hureau, E Gras, P Faller Coordination Chemistry Reviews 308, 445-459, 2016 | 73 | 2016 |
Base free aryl coupling of diazonium compounds and boronic esters: self-activation allowing an overall highly practical process H Bonin, D Delbrayelle, P Demonchaux, E Gras Chemical communications 46 (15), 2677-2679, 2010 | 73 | 2010 |
Selective mono N-methylation of anilines with methanol catalyzed by rhenium complexes: An experimental and theoretical study D Wei, O Sadek, V Dorcet, T Roisnel, C Darcel, E Gras, E Clot, JB Sortais Journal of catalysis 366, 300-309, 2018 | 67 | 2018 |
Two Functions, One Molecule: A Metal‐Binding and a Targeting Moiety to Combat Alzheimer's Disease C Hureau, I Sasaki, E Gras, P Faller ChemBioChem 11 (7), 950-953, 2010 | 62 | 2010 |
Mild and Direct C–H Arylation of Quinoxalin-2 (1H)-ones with Aryldiazonium Salts under Metal-Free Conditions K Yin, R Zhang Synlett 29 (05), 597-602, 2018 | 46 | 2018 |
A new water-soluble Cu (II) chelator that retrieves Cu from Cu (amyloid-β) species, stops associated ROS production and prevents Cu (II)‐induced Aβ aggregation S Noël, F Perez, JT Pedersen, B Alies, S Ladeira, S Sayen, E Guillon, ... Journal of Inorganic Biochemistry 117, 322-325, 2012 | 44 | 2012 |
Chiral epoxides by desymmetrizing deprotonation of meso-epoxides. D Hodgson, E Gras Angewandte Chemie (International ed. in English) 41 (13), 2002 | 43 | 2002 |
Enantioselective synthesis of epoxides by α-deprotonation—electrophile trapping of achiral epoxides DM Hodgson, TJ Buxton, ID Cameron, E Gras, EHM Kirton Organic & biomolecular chemistry 1 (23), 4293-4301, 2003 | 42 | 2003 |
Metal‐free intermolecular azide–alkyne cycloaddition promoted by glycerol M Rodríguez‐Rodríguez, E Gras, MA Pericàs, M Gómez Chemistry–A European Journal 21 (51), 18706-18710, 2015 | 32 | 2015 |
Highly practical boronic acid surrogates for the Suzuki–Miyaura cross-coupling H Bonin, R Leuma-Yona, B Marchiori, P Demonchaux, E Gras Tetrahedron Letters 52 (10), 1132-1135, 2011 | 32 | 2011 |
A formal synthesis of (±) lycoramine via an intramolecular Heck reaction E Gras, C Guillou, C Thal Tetrahedron letters 40 (52), 9243-9244, 1999 | 31 | 1999 |
Dioxazaborocanes: old adducts, new tricks H Bonin, T Delacroix, E Gras Organic & Biomolecular Chemistry 9 (13), 4714-4724, 2011 | 30 | 2011 |
Copper-catalyzed one-pot synthesis of chalcogen-benzothiazoles/imidazo [1, 2-a] pyridines with sulfur/selenium powder and aryl boronic acids T Guo, XN Wei, YL Zhu, H Chen, SL Han, YC Ma Synlett 29 (11), 1530-1536, 2018 | 28 | 2018 |
Naphthylaminoborane: From structural switches to frustrated Lewis pair reactivity D Pla, O Sadek, S Cadet, B Mestre-Voegtlé, E Gras Dalton Transactions 44 (42), 18340-18346, 2015 | 28 | 2015 |
Expanding the Balz–Schiemann Reaction: Organotrifluoroborates Serve as Competent Sources of Fluoride Ion for Fluoro‐Dediazoniation T Mohy El Dine, O Sadek, E Gras, DM Perrin Chemistry–A European Journal 24 (56), 14933-14937, 2018 | 23 | 2018 |