Identification of quinoline-chalcone hybrids as potential antiulcer agents KV Sashidhara, SR Avula, V Mishra, GR Palnati, LR Singh, N Singh, ... European journal of medicinal chemistry 89, 638-653, 2015 | 116 | 2015 |
Molecular iodine catalysed one-pot synthesis of chromeno [4, 3-b] quinolin-6-ones under microwave irradiation KV Sashidhara, GR Palnati, LR Singh, A Upadhyay, SR Avula, A Kumar, ... Green Chemistry 17 (7), 3766-3770, 2015 | 64 | 2015 |
Coumarin–benzimidazole hybrids as a potent antimicrobial agent: synthesis and biological elevation LR Singh, SR Avula, S Raj, A Srivastava, GR Palnati, CKM Tripathi, ... The Journal of antibiotics 70 (9), 954-961, 2017 | 57 | 2017 |
A facile and efficient Bi (III) catalyzed synthesis of 1, 1-dihydroperoxides and 1, 2, 4, 5-tetraoxanes KV Sashidhara, SR Avula, LR Singh, GR Palnati Tetrahedron Letters 53 (36), 4880-4884, 2012 | 49 | 2012 |
Designing, synthesis of selective and high-affinity chalcone-benzothiazole hybrids as Brugia malayi thymidylate kinase inhibitors: in vitro validation and docking studies KV Sashidhara, SR Avula, PK Doharey, LR Singh, VM Balaramnavar, ... European Journal of Medicinal Chemistry 103, 418-428, 2015 | 43 | 2015 |
Design, synthesis and anticancer activity of dihydropyrimidinone–semicarbazone hybrids as potential human DNA ligase 1 inhibitors KV Sashidhara, LR Singh, M Shameem, S Shakya, A Kumar, TS Laxman, ... MedChemComm 7 (12), 2349-2363, 2016 | 30 | 2016 |
Coumarin-chalcone hybrid instigates DNA damage by minor groove binding and stabilizes p53 through post translational modifications R Ashraf, Hamidullah, M Hasanain, P Pandey, M Maheshwari, LR Singh, ... Scientific reports 7 (1), 45287, 2017 | 28 | 2017 |
Design, synthesis and in vitro evaluation of coumarin–imidazo [1, 2-a] pyridine derivatives against cancer induced osteoporosis KV Sashidhara, LR Singh, D Choudhary, A Arun, S Gupta, S Adhikary, ... RSC Advances 6 (83), 80037-80048, 2016 | 28 | 2016 |
Discovery of a novel small-molecule inhibitor that targets PP2A–β-catenin signaling and restricts tumor growth and metastasis S Maheshwari, SR Avula, A Singh, LR Singh, GR Palnati, RK Arya, ... Molecular Cancer Therapeutics 16 (9), 1791-1805, 2017 | 18 | 2017 |
Discovery of coumarin-dihydroquinazolinone analogs as niacin receptor 1 agonist with in-vivo anti-obesity efficacy LR Singh, A Kumar, A Upadhyay, S Gupta, GR Palanati, K Sikka, ... European journal of medicinal chemistry 152, 208-222, 2018 | 16 | 2018 |
Functionality study of chalcone-hydroxypyridinone hybrids as tyrosinase inhibitors and influence on anti-tyrosinase activity LR Singh, YL Chen, YY Xie, W Xia, XW Gong, RC Hider, T Zhou Journal of Enzyme Inhibition and Medicinal Chemistry 35 (1), 1562-1567, 2020 | 13 | 2020 |
A catalyst-free one-pot protocol for the construction of substituted isoindolinones under sustainable conditions KV Sashidhara, LR Singh, GR Palnati, SR Avula, R Kant Synlett 27 (16), 2384-2390, 2016 | 13 | 2016 |
In‐house chemical library repurposing: A case example for Pseudomonas aeruginosa antibiofilm activity and quorum sensing inhibition L Ravithej Singh, VC Tripathi, S Raj, A Kumar, S Gupta, S Horam, ... Drug Development Research 79 (8), 383-390, 2018 | 7 | 2018 |
Microwave-assisted efficient synthesis of pyrazole-fibrate derivatives as stimulators of glucose uptake in skeletal muscle cells S Gupta, AK Rai, S Pandey, LR Singh, R Kant, AK Tamrakar, ... Bioorganic & Medicinal Chemistry Letters 34, 127760, 2021 | 6 | 2021 |
Synthetic approaches to FDA approved drugs for asthma and COPD from 1969 to 2020 AA Kazi, BVS Reddy, LR Singh Bioorganic & medicinal chemistry 41, 116212, 2021 | 5 | 2021 |
Anti-Acanthamoeba activity of a semi-synthetic mangostin derivative and its ability in removal of Acanthamoeba triangularis WU19001 on contact lens J Chuprom, S Sangkanu, W Mitsuwan, R Boonhok, W Mahabusarakam, ... PeerJ 10, e14468, 2022 | 1 | 2022 |
An Insight into the Pharmacology of Sulphur Containing Peptide Drugs A Sharma, LR Singh European Journal of Medicinal Chemistry, 116456, 2024 | | 2024 |
Small molecule inhibitors of gpcr gpr68 and related receptors for treating cancer, glioblastoma, and other indications CC Hong, CH Williams, LR Singh US Patent App. 17/602,101, 2022 | | 2022 |
Coumarin-chalcone hybrid instigates DNA damage by minor groove binding and stabilizes p53 through post translational modifications. RA Raghib Ashraf, H Hamidullah, MH Mohammad Hasanain, ... | | 2017 |
Molecular Iodine Catalyzed One-Pot Synthesis of Chromeno[4,3-b]quinolin-6-ones under Microwave Irradiation. AKRK Koneni V. Sashidhara, Gopala Reddy Palnati, L. Ravithej Singh, Amit ... ChemInform Abstract 46 (47), 2015 | | 2015 |