| Structure–activity relationship of pyrrolyl diketo acid derivatives as dual inhibitors of HIV-1 integrase and reverse transcriptase ribonuclease H domain G Cuzzucoli Crucitti, M Métifiot, L Pescatori, A Messore, VN Madia, ... Journal of medicinal chemistry 58 (4), 1915-1928, 2015 | 85 | 2015 |
| Activity of caffeic acid derivatives against Candida albicans biofilm D De Vita, L Friggeri, FD D’Auria, F Pandolfi, F Piccoli, S Panella, ... Bioorganic & medicinal chemistry letters 24 (6), 1502-1505, 2014 | 84 | 2014 |
| Recent advances in recovery of lycopene from tomato waste: A potent antioxidant with endless benefits VN Madia, D De Vita, D Ialongo, V Tudino, A De Leo, L Scipione, ... Molecules 26 (15), 4495, 2021 | 65 | 2021 |
| Basic quinolinonyl diketo acid derivatives as inhibitors of HIV integrase and their activity against RNase H function of reverse transcriptase R Costi, M Métifiot, S Chung, G Cuzzucoli Crucitti, K Maddali, L Pescatori, ... Journal of Medicinal Chemistry 57 (8), 3223-3234, 2014 | 65 | 2014 |
| Inhibition of Leishmania infantum trypanothione reductase by diaryl sulfide derivatives F Saccoliti, G Angiulli, G Pupo, L Pescatori, VN Madia, A Messore, ... Journal of enzyme inhibition and medicinal chemistry 32 (1), 304-310, 2017 | 64 | 2017 |
| 6-(1-Benzyl-1H-pyrrol-2-yl)-2,4-dioxo-5-hexenoic Acids as Dual Inhibitors of Recombinant HIV-1 Integrase and Ribonuclease H, Synthesized by a Parallel … R Costi, M Métifiot, F Esposito, G Cuzzucoli Crucitti, L Pescatori, ... Journal of medicinal chemistry 56 (21), 8588-8598, 2013 | 64 | 2013 |
| Comparison of different methods for the extraction of cannabinoids from cannabis D De Vita, VN Madia, V Tudino, F Saccoliti, A De Leo, A Messore, ... Natural product research 34 (20), 2952-2958, 2020 | 63 | 2020 |
| Synthesis and antifungal activity of a new series of 2-(1H-imidazol-1-yl)-1-phenylethanol derivatives D De Vita, L Scipione, S Tortorella, P Mellini, B Di Rienzo, G Simonetti, ... European Journal of Medicinal Chemistry 49, 334-342, 2012 | 61 | 2012 |
| N-Substituted Quinolinonyl Diketo Acid Derivatives as HIV Integrase Strand Transfer Inhibitors and Their Activity against RNase H Function of Reverse Transcriptase L Pescatori, M Métifiot, S Chung, T Masoaka, G Cuzzucoli Crucitti, ... Journal of medicinal chemistry 58 (11), 4610-4623, 2015 | 47 | 2015 |
| Inhibition of the α-carbonic anhydrase from Vibrio cholerae with amides and sulfonamides incorporating imidazole moieties D De Vita, A Angeli, F Pandolfi, M Bortolami, R Costi, R Di Santo, ... Journal of enzyme inhibition and medicinal chemistry 32 (1), 798-804, 2017 | 41 | 2017 |
| Acetylcholinesterase inhibitors for the treatment of Alzheimer’s disease–a patent review (2016–present) M Bortolami, D Rocco, A Messore, R Di Santo, R Costi, VN Madia, ... Expert Opinion on Therapeutic Patents 31 (5), 399-420, 2021 | 40 | 2021 |
| New deferiprone derivatives as multi-functional cholinesterase inhibitors: design, synthesis and in vitro evaluation M Bortolami, F Pandolfi, D De Vita, C Carafa, A Messore, R Di Santo, ... European Journal of Medicinal Chemistry 198, 112350, 2020 | 40 | 2020 |
| Novel benzazole derivatives endowed with potent antiheparanase activity VN Madia, A Messore, L Pescatori, F Saccoliti, V Tudino, A De Leo, ... Journal of medicinal chemistry 61 (15), 6918-6936, 2018 | 37 | 2018 |
| New pyridine derivatives as inhibitors of acetylcholinesterase and amyloid aggregation F Pandolfi, D De Vita, M Bortolami, A Coluccia, R Di Santo, R Costi, ... European journal of medicinal chemistry 141, 197-210, 2017 | 35 | 2017 |
| (Thiazol-2-yl) hydrazone derivatives from acetylpyridines as dual inhibitors of MAO and AChE: synthesis, biological evaluation and molecular modeling studies M D’Ascenzio, P Chimenti, MC Gidaro, C De Monte, D De Vita, A Granese, ... Journal of Enzyme Inhibition and Medicinal Chemistry 30 (6), 908-919, 2015 | 35 | 2015 |
| Searching for new agents active against Candida albicans biofilm: A series of indole derivatives, design, synthesis and biological evaluation F Pandolfi, F D'Acierno, M Bortolami, D De Vita, F Gallo, A De Meo, ... European Journal of Medicinal Chemistry 165, 93-106, 2019 | 34 | 2019 |
| Design, Synthesis, and Biological Evaluation of New 1-(Aryl-1H-pyrrolyl)(phenyl)methyl-1H-imidazole Derivatives as Antiprotozoal Agents F Saccoliti, VN Madia, V Tudino, A De Leo, L Pescatori, A Messore, ... Journal of Medicinal Chemistry 62 (3), 1330-1347, 2019 | 33 | 2019 |
| Design, Synthesis, and Structure–Activity Relationship of N-Arylnaphthylamine Derivatives as Amyloid Aggregation Inhibitors R Di Santo, R Costi, G Cuzzucoli Crucitti, L Pescatori, F Rosi, L Scipione, ... Journal of medicinal chemistry 55 (19), 8538-8548, 2012 | 33 | 2012 |
| On the structure of intermediate adducts arising from dithionite reduction of pyridinium salts: a novel class of derivatives of the parent sulfinic acid V Carelli, F Liberatore, L Scipione, R Musio, O Sciacovelli Tetrahedron Letters 41 (8), 1235-1240, 2000 | 33 | 2000 |
| Exploring the anti-biofilm activity of cinnamic acid derivatives in Candida albicans D De Vita, G Simonetti, F Pandolfi, R Costi, R Di Santo, FD D’Auria, ... Bioorganic & medicinal chemistry letters 26 (24), 5931-5935, 2016 | 32 | 2016 |
Roberto Di SantoProfessore di Chimica Farmaceutica, Sapienza Università di Roma在 uniroma1.it 的电子邮件经过验证
