Synthesis of ortho substituted arylboronic esters by in situ trapping of unstable lithio intermediates J Kristensen, M Lysén, P Vedsø, M Begtrup Organic letters 3 (10), 1435-1437, 2001 | 151 | 2001 |
Radiosynthesis and in vivo evaluation of a series of substituted 11C-phenethylamines as 5-HT2A agonist PET tracers A Ettrup, M Hansen, MA Santini, J Paine, N Gillings, M Palner, S Lehel, ... European journal of nuclear medicine and molecular imaging 38, 681-693, 2011 | 135 | 2011 |
Synthesis and Structure–Activity Relationships of N-Benzyl Phenethylamines as 5-HT2A/2C Agonists M Hansen, K Phonekeo, JS Paine, S Leth-Petersen, M Begtrup, ... ACS chemical neuroscience 5 (3), 243-249, 2014 | 127 | 2014 |
Palladium‐Catalyzed Asymmetric Allylic Alkylation of α‐Aryl Ketones BM Trost, GM Schroeder, J Kristensen Angewandte Chemie 114 (18), 3642-3645, 2002 | 126 | 2002 |
Inhibitors of histone demethylases B Lohse, JL Kristensen, LH Kristensen, K Agger, K Helin, M Gajhede, ... Bioorganic & medicinal chemistry 19 (12), 3625-3636, 2011 | 120 | 2011 |
Serotonin 2A receptor agonist binding in the human brain with [11C]-Cimbi-36 A Ettrup, S da Cunha-Bang, B McMahon, S Lehel, A Dyssegaard, ... Journal of Cerebral Blood Flow & Metabolism, 2014 | 100 | 2014 |
Synthesis of 4-substituted 1-(benzyloxy) pyrazoles via iodine− magnesium exchange of 1-(benzyloxy)-4-iodopyrazole J Felding, J Kristensen, T Bjerregaard, L Sander, P Vedsø, M Begtrup The Journal of Organic Chemistry 64 (11), 4196-4198, 1999 | 84 | 1999 |
Convergent synthesis of 6-substituted phenanthridines via anionic ring closure M Lysén, JL Kristensen, P Vedsø, M Begtrup Organic letters 4 (2), 257-259, 2002 | 78 | 2002 |
Development of a 11 C-labeled tetrazine for rapid tetrazine–trans-cyclooctene ligation MM Herth, VL Andersen, S Lehel, J Madsen, GM Knudsen, JL Kristensen Chemical Communications 49 (36), 3805-3807, 2013 | 75 | 2013 |
Trans-Cyclooctene-Functionalized PeptoBrushes with Improved Reaction Kinetics of the Tetrazine Ligation for Pretargeted Nuclear Imaging EJL Stéen, JT Jørgensen, K Johann, K Nørregaard, B Sohr, D Svatunek, ... ACS nano 14 (1), 568-584, 2019 | 70 | 2019 |
Lipophilicity and Click Reactivity Determine the Performance of Bioorthogonal Tetrazine Tools in Pretargeted In Vivo Chemistry EJL Stéen, JT Jørgensen, C Denk, UM Battisti, K Nørregaard, PE Edem, ... ACS pharmacology & translational science 4 (2), 824-833, 2021 | 65 | 2021 |
Identification of a new metabolite of GHB: gamma-hydroxybutyric acid glucuronide IN Petersen, C Tortzen, JL Kristensen, DS Pedersen, T Breindahl Journal of analytical toxicology 37 (5), 291-297, 2013 | 56 | 2013 |
Design, synthesis, and biological evaluation of Erythrina alkaloid analogues as neuronal nicotinic acetylcholine receptor antagonists F Crestey, AA Jensen, M Borch, JT Andreasen, J Andersen, T Balle, ... Journal of Medicinal Chemistry 56 (23), 9673-9682, 2013 | 55 | 2013 |
DARK classics in chemical neuroscience: NBOMes CBM Poulie, AA Jensen, AL Halberstadt, JL Kristensen ACS chemical neuroscience 11 (23), 3860-3869, 2019 | 52 | 2019 |
Hallucinogen-like effects of 2-([2-(4-cyano-2,5-dimethoxyphenyl) ethylamino]methyl)phenol (25CN-NBOH), a novel N-benzylphenethylamine with 100-fold selectivity for 5-HT … WE Fantegrossi, BW Gray, JM Bailey, DA Smith, M Hansen, JL Kristensen Psychopharmacology 232, 1039-1047, 2015 | 52 | 2015 |
Metabolic fate of hallucinogenic NBOMes S Leth-Petersen, C Gabel-Jensen, N Gillings, S Lehel, HD Hansen, ... Chemical research in toxicology 29 (1), 96-100, 2016 | 51 | 2016 |
Detailed characterization of the in vitro pharmacological and pharmacokinetic properties of N-(2-hydroxybenzyl)-2, 5-dimethoxy-4-cyanophenylethylamine (25CN-NBOH), a highly … AA Jensen, JD McCorvy, S Leth-Petersen, C Bundgaard, G Liebscher, ... Journal of Pharmacology and Experimental Therapeutics 361 (3), 441-453, 2017 | 50 | 2017 |
In Situ Generation of the Ohira–Bestmann Reagent from Stable Sulfonyl Azide: Scalable Synthesis of Alkynes from Aldehydes TH Jepsen, JL Kristensen The Journal of Organic Chemistry 79 (19), 9423-9426, 2014 | 50 | 2014 |
Synthesis of enantiopure 3-substituted morpholines J Bornholdt, J Felding, JL Kristensen The Journal of Organic Chemistry 75 (21), 7454-7457, 2010 | 50 | 2010 |
Direct Cu-mediated aromatic 18 F-labeling of highly reactive tetrazines for pretargeted bioorthogonal PET imaging R García-Vázquez, UM Battisti, JT Jørgensen, V Shalgunov, L Hvass, ... Chemical science 12 (35), 11668-11675, 2021 | 49 | 2021 |