| Development of high-specificity fluorescent probes to enable cannabinoid type 2 receptor studies in living cells RC Sarott, MV Westphal, P Pfaff, C Korn, DA Sykes, T Gazzi, B Brennecke, ... Journal of the American Chemical Society 142 (40), 16953-16964, 2020 | 40 | 2020 |
| Detection of cannabinoid receptor type 2 in native cells and zebrafish with a highly potent, cell-permeable fluorescent probe T Gazzi, B Brennecke, K Atz, C Korn, D Sykes, G Forn-Cuni, P Pfaff, ... Chemical Science 13 (19), 5539-5545, 2022 | 20 | 2022 |
| Cannabinoid receptor type 2 ligands: an analysis of granted patents since 2010 B Brennecke, T Gazzi, K Atz, J Fingerle, P Kuner, T Schindler, G Weck, ... Pharmaceutical Patent Analyst 10 (3), 111-163, 2021 | 18 | 2021 |
| Probing 2H‐Indazoles as Templates for SGK1, Tie2, and SRC Kinase Inhibitors J Schoene, T Gazzi, P Lindemann, M Christmann, A Volkamer, M Nazaré ChemMedChem 14 (16), 1514-1527, 2019 | 9 | 2019 |
| Synthesis, Inhibition of Mycobacterium tuberculosis Enoyl-acyl Carrier Protein Reductase and Antimycobacterial Activity of Novel Pentacyanoferrate(II … TP Gazzi, M Rotta, AD Villela, V Rodrigues-Junior, LKB Martinelli, ... Journal of the Brazilian Chemical Society 28 (10), 2028-2037, 2017 | 8 | 2017 |
| Diverse chemotypes drive biased signaling by cannabinoid receptors T Miljuš, FM Heydenreich, T Gazzi, A Kimbara, M Rogers-Evans, ... bioRxiv, 2020.11. 09.375162, 2020 | 6 | 2020 |
| Fluorescent probes for monoacylglycerol lipase (magl) J Benz, T Gazzi, L Gobbi, U Grether, B Hornsperger, C Kroll, B Kuhn, ... US Patent App. 17/700,987, 2022 | 4 | 2022 |
| Drug derived fluorescent probes for the specific visualization of cannabinoid type 2 receptor-a toolbox approach T Gazzi, B Brennecke, K Atz, C Korn, D Sykes, RC Sarott, MV Westphal, ... | 3 | 2019 |
| A greener approach toward gadolinium-based contrast agents TP Gazzi, LA Basso, DS Santos, P Machado RSC advances 4 (19), 9880-9884, 2014 | 3 | 2014 |
| Highly Specific, Fluorescent Cannabinoid Type 2 Receptor Probes Enable Applications in Microscopy, Flow Cytometry and FRET-based Binding Assays R Sarott, M Westphal, P Pfaff, C Korn, D Sykes, T Gazzi, B Brennecke, ... | 2 | 2019 |
| Highly Selective Drug-Derived Fluorescent Probes for the Cannabinoid Receptor Type 1 (CB1R) L Mach, A Omran, J Bouma, S Radetzki, DA Sykes, W Guba, X Li, ... Journal of Medicinal Chemistry, 2024 | 1 | 2024 |
| Aβ Chronic Exposure Promotes an Activation State of Microglia through Endocannabinoid Signalling Imbalance L Scipioni, D Tortolani, F Ciaramellano, F Fanti, T Gazzi, M Sergi, ... International Journal of Molecular Sciences 24 (7), 6684, 2023 | 1 | 2023 |
| Kinetic Profiling of Ligands and Fragments Binding to GPCRs by TR-FRET DA Sykes, L Borrega-Roman, CR Harwood, B Hoare, JM Lochray, ... Biophysical and Computational Tools in Drug Discovery, 1-32, 2021 | 1 | 2021 |
| Chemical Synthesis of Secretoglobin 3A2 Covalent Homodimer and Photocaged Monomeric Variants T Gazzi, M Heinke, F Landolt, JW Bode Angewandte Chemie International Edition, e202404992, 2024 | | 2024 |
| DOTA‐Based Plectin‐1 Targeted Contrast Agent Enables Detection of Pancreatic Cancer in Human Tissue T Gazzi, M Lesina, Q Wang, A Berninger, S Radetzki, IE Demir, ... Angewandte Chemie, e202318485, 2024 | | 2024 |
| Visualization of membrane localization and functional state of CB2R pools by matched agonist and inverse agonist probe pairs M Wasinka-Kalwa, A Omran, L Mach, J Bouma, L Scipioni, X Li, ... | | 2024 |
| A universal cannabinoid CB1 and CB2 receptor TR-FRET kinetic ligand binding assay. L Borrega-Roman, BL Hoare, M Kosar, RC Sarott, KJ Patej, J Bouma, ... bioRxiv, 2024.07. 16.603654, 2024 | | 2024 |
| Generation of a TR-FRET-based assay for the determination of cannabinoid CB1 receptor ligand binding kinetics L Borrega, B Hoare, T Gazzi, M Nazare, U Grether, D Sykes, D Veprintsev BRITISH JOURNAL OF PHARMACOLOGY 178 (2), 442-443, 2021 | | 2021 |
| Development and application of a kinetic ligand binding assay for the cannabinoid receptor 1 using resonance energy transfer approaches B Hoare, D Sykes, T Gazzi, M Nazare, U Grether, D Veprintsev BRITISH JOURNAL OF PHARMACOLOGY 177 (11), 2528-2529, 2020 | | 2020 |
| Illuminating Protein-Targets: Design and Synthesis of New Optical Imaging Probes for Studies of the Cannabinoid Type 2 Receptor and Plectin-1 T Gazzi PQDT-Global, 2020 | | 2020 |
