Investigating the Influence of (Deoxy)fluorination on the Lipophilicity of Non‐UV‐Active Fluorinated Alkanols and Carbohydrates by a New log P Determination … B Linclau, Z Wang, G Compain, V Paumelle, CQ Fontenelle, N Wells, ... Angewandte Chemie International Edition 55 (2), 674-678, 2016 | 146 | 2016 |
Keteniminium ion-initiated cascade cationic polycyclization C Theunissen, B Metayer, N Henry, G Compain, J Marrot, A Martin-Mingot, ... Journal of the American Chemical Society 136 (36), 12528-12531, 2014 | 120 | 2014 |
Stereoselective hydrofluorination of ynamides: a straightforward synthesis of novel α-fluoroenamides G Compain, K Jouvin, A Martin-Mingot, G Evano, J Marrot, S Thibaudeau Chemical communications 48 (42), 5196-5198, 2012 | 120 | 2012 |
A Journey in the Chemistry of Ynamides: from Synthesis to Applications G Evano, N Blanchard, G Compain, A Coste, CS Demmer, W Gati, ... Chemistry Letters 45 (6), 574-585, 2016 | 98 | 2016 |
Chemo-and stereoselective synthesis of fluorinated enamides from ynamides in HF/pyridine: second-generation approach to potent ureas bioisosteres B Metayer, G Compain, K Jouvin, A Martin-Mingot, C Bachmann, J Marrot, ... The Journal of Organic Chemistry 80 (7), 3397-3410, 2015 | 72 | 2015 |
Intramolecular OH⋅⋅⋅ Fluorine Hydrogen Bonding in Saturated, Acyclic Fluorohydrins: The γ‐Fluoropropanol Motif B Linclau, F Peron, E Bogdan, N Wells, Z Wang, G Compain, ... Chemistry–A European Journal 21 (49), 17808-17816, 2015 | 48 | 2015 |
Superacid synthesis of halogen containing N-substituted-4-aminobenzene sulfonamides: new selective tumor-associated carbonic anhydrase inhibitors G Compain, A Martin-Mingot, A Maresca, S Thibaudeau, CT Supuran Bioorganic & medicinal chemistry 21 (6), 1555-1563, 2013 | 45 | 2013 |
Indium (III)-catalyzed transformations of alkynes: recent advances in carbo-and heterocyclization reactions SR Pathipati, A van der Werf, N Selander Synthesis 49 (22), 4931-4941, 2017 | 41 | 2017 |
Influence of Alcohol β‐Fluorination on Hydrogen‐Bond Acidity of Conformationally Flexible Substrates J Graton, G Compain, F Besseau, E Bogdan, JM Watts, L Mtashobya, ... Chemistry–A European Journal 23 (12), 2811-2819, 2017 | 40 | 2017 |
Influence of Fluorination on the Conformational Properties and Hydrogen‐Bond Acidity of Benzyl Alcohol Derivatives E Bogdan, G Compain, L Mtashobya, JY Le Questel, F Besseau, ... Chemistry–A European Journal 21 (32), 11462-11474, 2015 | 35 | 2015 |
A β-glucuronidase-responsive albumin-binding prodrug for potential selective kinase inhibitor-based cancer chemotherapy G Compain, N Oumata, J Clarhaut, E Péraudeau, B Renoux, H Galons, ... European Journal of Medicinal Chemistry 158, 1-6, 2018 | 27 | 2018 |
Cationic polycyclization of ynamides: building up molecular complexity C Theunissen, B Métayer, M Lecomte, N Henry, HC Chan, G Compain, ... Organic & biomolecular chemistry 15 (20), 4399-4416, 2017 | 26 | 2017 |
Anti-Markovnikov additions to N-allylic derivatives involving ammonium–carbenium superelectrophiles G Compain, A Martin-Mingot, G Frapper, C Bachmann, MP Jouannetaud, ... Chemical Communications 48 (47), 5877-5879, 2012 | 26 | 2012 |
Selective Anti-Markovnikov Cyclization and Hydrofluorination Reaction in Superacid HF/SbF5: A Tool in the Design of Nitrogen-Containing (Fluorinated) Polycyclic … G Compain, C Bonneau, A Martin-Mingot, S Thibaudeau The Journal of Organic Chemistry 78 (9), 4463-4472, 2013 | 18 | 2013 |
A copper-catalyzed N-alkynylation route to 2-substituted N-alkynyl pyrroles and their cyclization into pyrrolo [2, 1-c] oxazin-1-ones: a formal total synthesis of peramine BJ Reinus, SM Kerwin Synthesis 49 (11), 2544-2554, 2017 | 16 | 2017 |
Bond Strength and Reactivity Scales for Lewis Superacid Adducts: A Comparative Study with In(OTf)3 and Al(OTf)3 G Compain, L Sikk, L Massi, JF Gal, E Duñach ChemPhysChem 18 (6), 683-691, 2017 | 14 | 2017 |
α‐Fluoro‐o‐cresols: The Key Role of Intramolecular Hydrogen Bonding in Conformational Preference and Hydrogen‐Bond Acidity E Bogdan, A Quarré de Verneuil, F Besseau, G Compain, B Linclau, ... ChemPhysChem 17 (17), 2702-2709, 2016 | 13 | 2016 |
Iterative structure-based optimization of short peptides targeting the bacterial sliding clamp C Monsarrat, G Compain, C André, S Engilberge, I Martiel, V Oliéric, ... Journal of Medicinal Chemistry 64 (23), 17063-17078, 2021 | 10 | 2021 |
Dications in superacid HF/SbF5: When superelectrophilic activation makes possible fluorination and/or C–H bond activation A Martin-Mingot, G Compain, F Liu, MP Jouannetaud, C Bachmann, ... Journal of Fluorine Chemistry 134, 56-62, 2012 | 10 | 2012 |
Antibacterial activity of a dual peptide targeting the Escherichia coli sliding clamp and the ribosome C André, F Veillard, P Wolff, AM Lobstein, G Compain, C Monsarrat, ... RSC Chemical Biology 1 (3), 137-147, 2020 | 8 | 2020 |