受强制性开放获取政策约束的文章 - Thomas Machleidt了解详情
可在其他位置公开访问的文章：14 篇
Discovery of potent and selective covalent inhibitors of JNK
T Zhang, F Inesta-Vaquera, M Niepel, J Zhang, SB Ficarro, T Machleidt, ...
Chemistry & biology 19 (1), 140-154, 2012
强制性开放获取政策： US National Institutes of Health
Application of BRET to monitor ligand binding to GPCRs
LA Stoddart, EKM Johnstone, AJ Wheal, J Goulding, MB Robers, ...
Nature methods 12 (7), 661-663, 2015
强制性开放获取政策： Australian Research Council, National Health and Medical Research Council …
Target engagement and drug residence time can be observed in living cells with BRET
MB Robers, ML Dart, CC Woodroofe, CA Zimprich, TA Kirkland, ...
Nature communications 6 (1), 10091, 2015
强制性开放获取政策： US National Institutes of Health
Quantitative, wide-spectrum kinase profiling in live cells for assessing the effect of cellular ATP on target engagement
JD Vasta, CR Corona, J Wilkinson, CA Zimprich, JR Hartnett, MR Ingold, ...
Cell chemical biology 25 (2), 206-214. e11, 2018
强制性开放获取政策： US National Institutes of Health, Genome Canada, Wellcome Trust
Identification of a new JNK inhibitor targeting the JNK-JIP interaction site
JL Stebbins, SK De, T Machleidt, B Becattini, J Vazquez, C Kuntzen, ...
Proceedings of the National Academy of Sciences 105 (43), 16809-16813, 2008
强制性开放获取政策： US National Institutes of Health
Design, synthesis, and structure− activity relationship of substrate competitive, selective, and in vivo active triazole and thiadiazole inhibitors of the c-Jun N-terminal kinase
SK De, JL Stebbins, LH Chen, M Riel-Mehan, T Machleidt, R Dahl, ...
Journal of medicinal chemistry 52 (7), 1943-1952, 2009
强制性开放获取政策： US National Institutes of Health
Exploiting an Asp-Glu “switch” in glycogen synthase kinase 3 to design paralog-selective inhibitors for use in acute myeloid leukemia
FF Wagner, L Benajiba, AJ Campbell, M Weïwer, JR Sacher, JP Gale, ...
Science translational medicine 10 (431), eaam8460, 2018
强制性开放获取政策： US National Institutes of Health, National Institute of Health and Medical …
Real-time analysis of the binding of fluorescent VEGF165a to VEGFR2 in living cells: effect of receptor tyrosine kinase inhibitors and fate of internalized agonist-receptor …
LE Kilpatrick, R Friedman-Ohana, DC Alcobia, K Riching, CJ Peach, ...
Biochemical Pharmacology 136, 62-75, 2017
强制性开放获取政策： UK Biotechnology and Biological Sciences Research Council
Simultaneous inhibition of DNA-PK and Polϴ improves integration efficiency and precision of genome editing
S Wimberger, N Akrap, M Firth, J Brengdahl, S Engberg, MK Schwinn, ...
Nature communications 14 (1), 4761, 2023
强制性开放获取政策： European Commission
Design and characterization of a potent and selective dual ATP-and substrate-competitive subnanomolar bidentate c-Jun N-terminal kinase (JNK) inhibitor
JL Stebbins, SK De, P Pavlickova, V Chen, T Machleidt, LH Chen, ...
Journal of medicinal chemistry 54 (18), 6206-6214, 2011
强制性开放获取政策： US National Institutes of Health
Discovery of 2-(5-nitrothiazol-2-ylthio) benzo [d] thiazoles as novel c-Jun N-terminal kinase inhibitors
SK De, LH Chen, JL Stebbins, T Machleidt, M Riel-Mehan, R Dahl, ...
Bioorganic & medicinal chemistry 17 (7), 2712-2717, 2009
强制性开放获取政策： US National Institutes of Health
Synthesis and optimization of thiadiazole derivatives as a novel class of substrate competitive c-Jun N-terminal kinase inhibitors
SK De, V Chen, JL Stebbins, LH Chen, JF Cellitti, T Machleidt, E Barile, ...
Bioorganic & medicinal chemistry 18 (2), 590-596, 2010
强制性开放获取政策： US National Institutes of Health
Design, synthesis, and structure–activity relationship studies of thiophene-3-carboxamide derivatives as dual inhibitors of the c-Jun N-terminal kinase
SK De, E Barile, V Chen, JL Stebbins, JF Cellitti, T Machleidt, CB Carlson, ...
Bioorganic & medicinal chemistry 19 (8), 2582-2588, 2011
强制性开放获取政策： US National Institutes of Health
Identification of known drugs targeting the endoplasmic reticulum stress response
K Bi, K Nishihara, T Machleidt, S Hermanson, J Wang, S Sakamuru, ...
Analytical and bioanalytical chemistry 407, 5343-5351, 2015
强制性开放获取政策： US National Institutes of Health
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