Design, synthesis and biological evaluation of (E)-5-styryl-1, 2, 4-oxadiazoles as anti-tubercular agents AA Upare, PK Gadekar, H Sivaramakrishnan, N Naik, VM Khedkar, ... Bioorganic Chemistry 86, 507-512, 2019 | 55 | 2019 |
A fluorinated analog of ISO-1 blocks the recognition and biological function of MIF and is orally efficacious in a murine model of colitis NM Dagia, DV Kamath, P Bhatt, RD Gupte, SS Dadarkar, L Fonseca, ... European journal of pharmacology 607 (1-3), 201-212, 2009 | 43 | 2009 |
Design, synthesis and biological evaluation of novel azaspiro analogs of linezolid as antibacterial and antitubercular agents PK Gadekar, A Roychowdhury, PS Kharkar, VM Khedkar, M Arkile, ... European Journal of Medicinal Chemistry 122, 475-487, 2016 | 39 | 2016 |
Novel derivatives of ISO-1 as potent inhibitors of MIF biological function S Balachandran, A Rodge, PK Gadekar, VN Yadav, D Kamath, ... Bioorganic & medicinal chemistry letters 19 (16), 4773-4776, 2009 | 26 | 2009 |
Synthesis and biological activity of novel MIF antagonists S Balachandran, PK Gadekar, S Parkale, VN Yadav, D Kamath, ... Bioorganic & medicinal chemistry letters 21 (5), 1508-1511, 2011 | 21 | 2011 |
Design, synthesis and biological evaluation of 2, 3-dihydroimidazo [2, 1-b] thiazoles as dual EGFR and IGF1R inhibitors PK Gadekar, G Urunkar, A Roychowdhury, R Sharma, J Bose, S Khanna, ... Bioorganic Chemistry 115, 105151, 2021 | 16 | 2021 |
Reductive removal of methoxyacetyl protective group using sodium borohydride PK Gadekar, M Hoermann, F Corbo, R Sharma, S Sarveswari, ... Tetrahedron Letters 55 (2), 503-506, 2014 | 6 | 2014 |
Chemical Optimization of CBL0137 for Human African Trypanosomiasis Lead Drug Discovery MPP BaljinderSingh,AmritaSharma,NareshGunaganti,MitchRivers,PradipK.Gadekar ... Journal of medicinal Chemistry, 2023 | 5 | 2023 |
Chlorotrifluoroethylidenes: an efficient and convenient approach to their synthesis AA Upare, PK Gadekar, K Jadhav, H Sivaramakrishnan, SM Roopan RSC advances 10 (30), 17427-17431, 2020 | 2 | 2020 |
Design, Synthesis, and the Effects of (E)-9-Oxooctadec-10-en-12-ynoic Acid Analogues to Promote Glucose Uptake RR Kshirsagar, PK Gadekar, VM Khedkar, V Vijayakumar ACS omega 6 (37), 24118-24127, 2021 | 1 | 2021 |
Part I: Thiazoles Chapter 1 Synthesis, Properties, and Biological Applications of 1, 3-Thiazoles 3 NR Darekar, VM Khedkar, PK Gadekar, SD Mhaske, SJ Takate, ... | | 2024 |
EZH2 inhibitors and uses thereof Roychowdhury A., Sharma R., Gupte A., Kandre S., Gadekar P. K. US Patent WO/2015/110999(A1, 2015 | | 2015 |
Substituted Heterocyclic Amine Derivatives as Multikinase Inhibitors for the Treatment of Cancer Roychowdhury A., Sharma R., Gadekar P. K., et al. US Patent WO 2015/128698 A1,, 2015 | | 2015 |
Bicyclic compounds and uses thereof, GPK 4. Sharma R., Gupte A., Roychowdhury A., Jadhav R. D., Kandre S. S ... US Patent PCT/IB2014/060157., 2014 | | 2014 |
Substituted heterocyclic compounds as EZH2 inhibitors GPK Roychowdhury US Patent WO2014155301A1, 2014 | | 2014 |
Design Synthesis And The Medicinal Chemistry Applications Of Azaspiro Analogues PK Gadekar Vellore, 0 | | |