关注
Dr. Pradip K Gadekar
Dr. Pradip K Gadekar
Northeastern University Boston
在 piramal.com 的电子邮件经过验证
标题
引用次数
引用次数
年份
Design, synthesis and biological evaluation of (E)-5-styryl-1, 2, 4-oxadiazoles as anti-tubercular agents
AA Upare, PK Gadekar, H Sivaramakrishnan, N Naik, VM Khedkar, ...
Bioorganic Chemistry 86, 507-512, 2019
552019
A fluorinated analog of ISO-1 blocks the recognition and biological function of MIF and is orally efficacious in a murine model of colitis
NM Dagia, DV Kamath, P Bhatt, RD Gupte, SS Dadarkar, L Fonseca, ...
European journal of pharmacology 607 (1-3), 201-212, 2009
432009
Design, synthesis and biological evaluation of novel azaspiro analogs of linezolid as antibacterial and antitubercular agents
PK Gadekar, A Roychowdhury, PS Kharkar, VM Khedkar, M Arkile, ...
European Journal of Medicinal Chemistry 122, 475-487, 2016
392016
Novel derivatives of ISO-1 as potent inhibitors of MIF biological function
S Balachandran, A Rodge, PK Gadekar, VN Yadav, D Kamath, ...
Bioorganic & medicinal chemistry letters 19 (16), 4773-4776, 2009
262009
Synthesis and biological activity of novel MIF antagonists
S Balachandran, PK Gadekar, S Parkale, VN Yadav, D Kamath, ...
Bioorganic & medicinal chemistry letters 21 (5), 1508-1511, 2011
212011
Design, synthesis and biological evaluation of 2, 3-dihydroimidazo [2, 1-b] thiazoles as dual EGFR and IGF1R inhibitors
PK Gadekar, G Urunkar, A Roychowdhury, R Sharma, J Bose, S Khanna, ...
Bioorganic Chemistry 115, 105151, 2021
162021
Reductive removal of methoxyacetyl protective group using sodium borohydride
PK Gadekar, M Hoermann, F Corbo, R Sharma, S Sarveswari, ...
Tetrahedron Letters 55 (2), 503-506, 2014
62014
Chemical Optimization of CBL0137 for Human African Trypanosomiasis Lead Drug Discovery
MPP BaljinderSingh,AmritaSharma,NareshGunaganti,MitchRivers,PradipK.Gadekar ...
Journal of medicinal Chemistry, 2023
52023
Chlorotrifluoroethylidenes: an efficient and convenient approach to their synthesis
AA Upare, PK Gadekar, K Jadhav, H Sivaramakrishnan, SM Roopan
RSC advances 10 (30), 17427-17431, 2020
22020
Design, Synthesis, and the Effects of (E)-9-Oxooctadec-10-en-12-ynoic Acid Analogues to Promote Glucose Uptake
RR Kshirsagar, PK Gadekar, VM Khedkar, V Vijayakumar
ACS omega 6 (37), 24118-24127, 2021
12021
Part I: Thiazoles Chapter 1 Synthesis, Properties, and Biological Applications of 1, 3-Thiazoles 3
NR Darekar, VM Khedkar, PK Gadekar, SD Mhaske, SJ Takate, ...
2024
EZH2 inhibitors and uses thereof
Roychowdhury A., Sharma R., Gupte A., Kandre S., Gadekar P. K.
US Patent WO/2015/110999(A1, 2015
2015
Substituted Heterocyclic Amine Derivatives as Multikinase Inhibitors for the Treatment of Cancer
Roychowdhury A., Sharma R., Gadekar P. K., et al.
US Patent WO 2015/128698 A1,, 2015
2015
Bicyclic compounds and uses thereof,
GPK 4. Sharma R., Gupte A., Roychowdhury A., Jadhav R. D., Kandre S. S ...
US Patent PCT/IB2014/060157., 2014
2014
Substituted heterocyclic compounds as EZH2 inhibitors
GPK Roychowdhury
US Patent WO2014155301A1, 2014
2014
Design Synthesis And The Medicinal Chemistry Applications Of Azaspiro Analogues
PK Gadekar
Vellore, 0
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