Harnessing Quinone Methides: Total Synthesis of (±)‐Vaticanol A TH Jepsen, SB Thomas, Y Lin, CI Stathakis, I de Miguel, SA Snyder Angewandte Chemie 126 (26), 6865-6869, 2014 | 55 | 2014 |
In Situ Generation of the Ohira–Bestmann Reagent from Stable Sulfonyl Azide: Scalable Synthesis of Alkynes from Aldehydes TH Jepsen, JL Kristensen The Journal of Organic Chemistry 79 (19), 9423-9426, 2014 | 53 | 2014 |
Synthesis of Functionalized Dibenzothiophenes–An Efficient Three‐Step Approach Based on Pd‐Catalyzed C–C and C–S Bond Formations TH Jepsen, M Larsen, M Jørgensen, KA Solanko, AD Bond, A Kadziola, ... European Journal of Organic Chemistry 2011 (1), 53-57, 2011 | 42 | 2011 |
Synthesis and pharmacological evaluation of DHβE analogues as neuronal nicotinic acetylcholine receptor antagonists TH Jepsen, AA Jensen, MH Lund, E Glibstrup, JL Kristensen ACS Medicinal Chemistry Letters 5 (7), 766-770, 2014 | 24 | 2014 |
Fragment-based discovery of pyrazolopyridones as JAK1 inhibitors with excellent subtype selectivity BB Hansen, TH Jepsen, M Larsen, R Sindet, T Vifian, MN Burhardt, ... Journal of Medicinal Chemistry 63 (13), 7008-7032, 2020 | 21 | 2020 |
Three-step synthesis of (thio) xanthene and dibenzothiepine/dibenzoxepine by an intramolecular Mizoroki-Heck reaction of diaryl (thio) ethers TH Jepsen, M Larsen, M Jørgensen, MB Nielsen Synlett 2012 (03), 418-422, 2012 | 21 | 2012 |
Synthesis of dibenzothiophene, dibenzofuran and carbazole donor–acceptor chromophores TH Jepsen, M Larsen, M Jørgensen, MB Nielsen Synthesis 45 (08), 1115-1120, 2013 | 12 | 2013 |
On the scope of Pd-catalyzed carboamination reactions—synthesis of 2, 4-disubstituted pyrrolidines and 2-substituted piperidines and morpholines TH Jepsen, M Larsen, MB Nielsen Tetrahedron 66 (32), 6133-6137, 2010 | 11 | 2010 |
An efficient protocol for synthesizing dibenzodithiapentalenes TH Jepsen, M Larsen, M Jørgensen, MB Nielsen Tetrahedron letters 52 (31), 4045-4047, 2011 | 9 | 2011 |
A strategic approach to [6, 6]-bicyclic lactones: application towards the CD fragment of DHβE TH Jepsen, E Glibstrup, F Crestey, AA Jensen, JL Kristensen Beilstein Journal of Organic Chemistry 13 (1), 988-994, 2017 | 8 | 2017 |
Versatile pyrolytic synthesis of fused polycyclic heteroaromatic compounds RA Aitken, AN Garnett Synthesis 49 (22), 4955-4977, 2017 | 7 | 2017 |
Development of a divergent route to erythrina alkaloids S Clementson, M Jessing, PJ Vital, JL Kristensen Synlett 31 (04), 327-333, 2020 | 3 | 2020 |
Dibenzo [bc, fg][1, 4] oxathiapentalene: an elusive molecule? V Mazzanti, EA Della Pia, M Jevric, TH Jepsen, A Kadziola, O Hammerich, ... Journal of Sulfur Chemistry 34 (6), 588-595, 2013 | 1 | 2013 |
Bicyclic amines as novel JAK kinase inhibitors DR Greve, TH Jepsen, M Larsen, A Ritzen US Patent 10,851,116, 2020 | | 2020 |
Fragment-based discovery of pyrazolopyridones as JAK1 inhibitors with excellent subtype selectivity A Ritzen, T Vifian, R Sindet, B Hansen, M Larsen, T Jepsen, J Larsen, ... ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY 256, 2018 | | 2018 |
Bicyclic amines as novel jak kinase inhibitors DR Greve, TH JEPSEN, M Larsen, A Ritzen | | 2018 |
Total Synthesis of (±)-Vaticanol A EM Carreira, A Joliton Synfacts 10 (08), 0784-0784, 2014 | | 2014 |
Deconstructing Erythrina Alkaloids: New Antagonists for the Neuronal NAChR's & Total Syntheses of (±)-Vaticanol A: PhD Thesis TH Jepsen Faculty of Health and Medical Sciences, University of Copenhagen, 2014 | | 2014 |
An Efficient Protocol for the Synthesis of Dibenzodithiapentalene TH Jepsen, M Larsen, M Jørgensen, MB Nielsen Synfacts 2011 (09), 0950-0950, 2011 | | 2011 |