| Synthesis and anticonvulsant activity of novel and potent 6, 7-methylenedioxyphthalazin-1 (2 H)-ones S Grasso, G De Sarro, A De Sarro, N Micale, M Zappalà, G Puja, ... Journal of medicinal chemistry 43 (15), 2851-2859, 2000 | 279 | 2000 |
| Synthesis of new Δ2-isoxazoline derivatives and their pharmacological characterization as β-adrenergic receptor antagonists P Conti, C Dallanoce, M De Amici, C De Micheli, KN Klotz Bioorganic & medicinal chemistry 6 (4), 401-408, 1998 | 129 | 1998 |
| Drug discovery targeting amino acid racemases P Conti, L Tamborini, A Pinto, A Blondel, P Minoprio, A Mozzarelli, ... Chemical reviews 111 (11), 6919-6946, 2011 | 126 | 2011 |
| Inhibition of rhodesain as a novel therapeutic modality for human African trypanosomiasis R Ettari, L Tamborini, IC Angelo, N Micale, A Pinto, C De Micheli, P Conti Journal of Medicinal Chemistry 56 (14), 5637-5658, 2013 | 100 | 2013 |
| Chemoenzymatic synthesis of chiral isoxazole derivatives M De Amici, C De Micheli, G Carrea, S Spezia The Journal of Organic Chemistry 54 (11), 2646-2650, 1989 | 98 | 1989 |
| A regioselective route to 5-substituted pyrazole-and pyrazoline-3-phosphonic acids and esters P Conti, A Pinto, L Tamborini, V Rizzo, C De Micheli Tetrahedron 63 (25), 5554-5560, 2007 | 89 | 2007 |
| Nitrile oxides in medicinal chemistry-2. synthesis of the two enantiomers of dihydromuscimol M De Amici, C De Micheli, V Misani Tetrahedron 46 (6), 1975-1986, 1990 | 85 | 1990 |
| 1-Aryl-6, 7-methylenedioxy-3H-quinazolin-4-ones as anticonvulsant agents M Zappala, S Grasso, N Micale, G Zuccala, FS Menniti, G Ferreri, ... Bioorganic & medicinal chemistry letters 13 (24), 4427-4430, 2003 | 81 | 2003 |
| 1, 3‐Dipolar Cycloreversions G Bianchi, C De Micheli, R Gandolfi Angewandte Chemie International Edition in English 18 (10), 721-738, 1979 | 77 | 1979 |
| Investigating the Mechanism of Substrate Uptake and Release in the Glutamate Transporter Homologue GltPh through Metadynamics Simulations G Grazioso, V Limongelli, D Branduardi, E Novellino, C De Micheli, ... Journal of the American Chemical Society 134 (1), 453-463, 2012 | 75 | 2012 |
| Isoxazoline derivatives. Part VI. Regioselectivity in the 1, 3-dipolar cycloaddition of nitrile oxides to αβ-unsaturated ketones G Bianchi, C De Micheli, R Gandolfi, P Grünanger, PV Finzi, OV de Pava Journal of the Chemical Society, Perkin Transactions 1, 1148-1155, 1973 | 64 | 1973 |
| Synthesis and anticonvulsant activity of novel and potent 2, 3-benzodiazepine AMPA/kainate receptor antagonists S Grasso, G De Sarro, A De Sarro, N Micale, M Zappalà, G Puia, ... Journal of medicinal chemistry 42 (21), 4414-4421, 1999 | 63 | 1999 |
| Chemoenzymic synthesis of the eight stereoisomeric muscarines M De Amici, C De Micheli, G Molteni, D Pitre, G Carrea, S Riva, S Spezia, ... The Journal of Organic Chemistry 56 (1), 67-72, 1991 | 62 | 1991 |
| Synthesis and functional characterization of novel derivatives related to oxotremorine and oxotremorine-M C Dallanoce, P Conti, M De Amici, C De Micheli, E Barocelli, M Chiavarini, ... Bioorganic & medicinal chemistry 7 (8), 1539-1547, 1999 | 58 | 1999 |
| Discovery of covalent inhibitors of glyceraldehyde-3-phosphate dehydrogenase, a target for the treatment of malaria S Bruno, A Pinto, G Paredi, L Tamborini, C De Micheli, V La Pietra, ... Journal of Medicinal Chemistry 57 (17), 7465-7471, 2014 | 57 | 2014 |
| Synthesis, binding affinity at glutamic acid receptors, neuroprotective effects, and molecular modeling investigation of novel dihydroisoxazole amino acids P Conti, M De Amici, G Grazioso, G Roda, A Pinto, KB Hansen, B Nielsen, ... Journal of medicinal chemistry 48 (20), 6315-6325, 2005 | 57 | 2005 |
| Design and synthesis of novel isoxazole-based HDAC inhibitors P Conti, L Tamborini, A Pinto, L Sola, R Ettari, C Mercurio, C De Micheli European journal of medicinal chemistry 45 (9), 4331-4338, 2010 | 51 | 2010 |
| Chemoenzymatic synthesis in flow reactors: A rapid and convenient preparation of Captopril V De Vitis, F Dall'Oglio, A Pinto, C De Micheli, F Molinari, P Conti, ... ChemistryOpen 6 (5), 668-673, 2017 | 50 | 2017 |
| Synthesis and enantiopharmacology of new AMPA-kainate receptor agonists P Conti, M De Amici, G De Sarro, M Rizzo, TB Stensbøl, ... Journal of medicinal chemistry 42 (20), 4099-4107, 1999 | 49 | 1999 |
| Development of rhodesain inhibitors with a 3‐bromoisoxazoline warhead R Ettari, L Tamborini, IC Angelo, S Grasso, T Schirmeister, L Lo Presti, ... ChemMedChem 8 (12), 2070-2076, 2013 | 47 | 2013 |
