| Associating HIV-1 envelope glycoprotein structures with states on the virus observed by smFRET M Lu, X Ma, LR Castillo-Menendez, J Gorman, N Alsahafi, U Ermel, ... Nature 568 (7752), 415-419, 2019 | 178 | 2019 |
| Azithromycin, a 15-membered macrolide antibiotic, inhibits influenza A (H1N1) pdm09 virus infection by interfering with virus internalization process DH Tran, R Sugamata, T Hirose, S Suzuki, Y Noguchi, A Sugawara, F Ito, ... The Journal of antibiotics 72 (10), 759-768, 2019 | 166 | 2019 |
| Design, synthesis and biological evaluation of small molecule inhibitors of CD4-gp120 binding based on virtual screening JM LaLonde, MA Elban, JR Courter, A Sugawara, T Soeta, N Madani, ... Bioorganic & medicinal chemistry 19 (1), 91-101, 2011 | 89 | 2011 |
| Chitinase inhibitors: extraction of the active framework from natural argifin and use of in situ click chemistry T Hirose, T Sunazuka, A Sugawara, A Endo, K Iguchi, T Yamamoto, H Ui, ... The Journal of antibiotics 62 (5), 277-282, 2009 | 73 | 2009 |
| Novel 12-membered non-antibiotic macrolides from erythromycin A; EM900 series as novel leads for anti-inflammatory and/or immunomodulatory agents A Sugawara, A Sueki, T Hirose, K Nagai, H Gouda, S Hirono, H Shima, ... Bioorganic & medicinal chemistry letters 21 (11), 3373-3376, 2011 | 58 | 2011 |
| Macrolides sensitize EGFR-TKI-induced non-apoptotic cell death via blocking autophagy flux in pancreatic cancer cell lines S Mukai, S Moriya, M Hiramoto, H Kazama, H Kokuba, XF Che, ... International journal of oncology 48 (1), 45-54, 2016 | 57 | 2016 |
| Crystal structures of HIV-1 gp120 envelope glycoprotein in complex with NBD analogues that target the CD4-binding site YD Kwon, JM LaLonde, Y Yang, MA Elban, A Sugawara, JR Courter, ... PloS one 9 (1), e85940, 2014 | 52 | 2014 |
| Borrelidin analogues with antimalarial activity: design, synthesis and biological evaluation against Plasmodium falciparum parasites A Sugawara, T Tanaka, T Hirose, A Ishiyama, M Iwatsuki, Y Takahashi, ... Bioorganic & medicinal chemistry letters 23 (8), 2302-2305, 2013 | 51 | 2013 |
| Asymmetric total synthesis of neoxaline T Ideguchi, T Yamada, T Shirahata, T Hirose, A Sugawara, Y Kobayashi, ... Journal of the American Chemical Society 135 (34), 12568-12571, 2013 | 50 | 2013 |
| Design and synthesis via click chemistry of 8, 9-anhydroerythromycin A 6, 9-hemiketal analogues with anti-MRSA and-VRE activity A Sugawara, T Sunazuka, T Hirose, K Nagai, Y Yamaguchi, H Hanaki, ... Bioorganic & medicinal chemistry letters 17 (22), 6340-6344, 2007 | 47 | 2007 |
| An inducible cell-cell fusion system with integrated ability to measure the efficiency and specificity of HIV-1 entry inhibitors A Herschhorn, A Finzi, DM Jones, JR Courter, A Sugawara, AB Smith III, ... PloS one 6 (11), e26731, 2011 | 36 | 2011 |
| Observation of the controlled assembly of preclick components in the in situ click chemistry generation of a chitinase inhibitor T Hirose, N Maita, H Gouda, J Koseki, T Yamamoto, A Sugawara, ... Proceedings of the National Academy of Sciences 110 (40), 15892-15897, 2013 | 29 | 2013 |
| Macrolides with promotive activity of monocyte to macrophage differentiation K Yoshida, T Sunazuka, K Nagai, A Sugawara, A Cho, T Nagamitsu, ... The Journal of Antibiotics 58 (1), 79-81, 2005 | 29 | 2005 |
| Leucomycin A3, a 16-membered macrolide antibiotic, inhibits influenza A virus infection and disease progression R Sugamata, A Sugawara, T Nagao, K Suzuki, T Hirose, K Yamamoto, ... The Journal of antibiotics 67 (3), 213-222, 2014 | 28 | 2014 |
| Asymmetric total synthesis of indole alkaloids containing an indoline spiroaminal framework T Yamada, T Ideguchi‐Matsushita, T Hirose, T Shirahata, R Hokari, ... Chemistry–A European Journal 21 (33), 11855-11864, 2015 | 27 | 2015 |
| Solution-phase total synthesis of the hydrophilic natural product argifin using 3, 4, 5-tris (octadecyloxy) benzyl tag T Hirose, T Kasai, T Akimoto, A Endo, A Sugawara, K Nagasawa, ... Tetrahedron 67 (35), 6633-6643, 2011 | 25 | 2011 |
| Macrolides promote CCL2-mediated macrophage recruitment and clearance of nasopharyngeal pneumococcal colonization in mice N Iwanaga, S Nakamura, K Oshima, T Kajihara, T Takazono, T Miyazaki, ... The Journal of Infectious Diseases 212 (7), 1150-1159, 2015 | 24 | 2015 |
| Three-dimensional solution structure of bottromycin A2: a potent antibiotic active against methicillin-resistant Staphylococcus aureus and vancomycin-resistant Enterococci H Gouda, Y Kobayashi, T Yamada, T Ideguchi, A Sugawara, T Hirose, ... Chemical and Pharmaceutical Bulletin 60 (2), 169-171, 2012 | 23 | 2012 |
| Effects of a novel nonantibiotic macrolide, EM900, on cytokine and mucin gene expression in a human airway epithelial cell line K Otsu, H Ishinaga, S Suzuki, A Sugawara, T Sunazuka, S Omura, H Jono, ... Pharmacology 88 (5-6), 327-332, 2011 | 23 | 2011 |
| Argifin; efficient solid phase total synthesis and evalution of analogues of acyclic peptide T Sunazuka, A Sugawara, K Iguchi, T Hirose, K Nagai, Y Noguchi, Y Saito, ... Bioorganic & medicinal chemistry 17 (7), 2751-2758, 2009 | 23 | 2009 |
Takeshi Yamada (山田 健)神戸薬科大学在 kobepharma-u.ac.jp 的电子邮件经过验证
