Ring Structure and Aromatic Substituent Effects on the pKa of the Benzoxaborole Pharmacophore JW Tomsho, A Pal, DG Hall, SJ Benkovic ACS medicinal chemistry letters 3 (1), 48-52, 2012 | 147 | 2012 |
The unique chemistry of benzoxaboroles: current and emerging applications in biotechnology and therapeutic treatments CT Liu, JW Tomsho, SJ Benkovic Bioorganic & medicinal chemistry 22 (16), 4462-4473, 2014 | 125 | 2014 |
Microtubule-assisted mechanism for functional metabolic macromolecular complex formation S An, Y Deng, JW Tomsho, M Kyoung, SJ Benkovic Proceedings of the National Academy of Sciences 107 (29), 12872-12876, 2010 | 118 | 2010 |
Elucidation of the mechanism of the reaction between phenylboronic acid and a model diol, Alizarin Red S JW Tomsho, SJ Benkovic The Journal of Organic Chemistry 77 (5), 2098-2106, 2012 | 112 | 2012 |
Discovery of antibacterial cyclic peptides that inhibit the ClpXP protease L Cheng, TA Naumann, AR Horswill, SJ Hong, BJ Venters, JW Tomsho, ... Protein Science 16 (8), 1535-1542, 2007 | 93 | 2007 |
Inhibition of HIV-1 reverse transcriptase-catalyzed DNA strand transfer reactions by 4-chlorophenylhydrazone of mesoxalic acid WR Davis, J Tomsho, S Nikam, EM Cook, D Somand, JA Peliska Biochemistry 39 (46), 14279-14291, 2000 | 68 | 2000 |
Examination of the Reactivity of Benzoxaboroles and Related Compounds with a cis-Diol JW Tomsho, SJ Benkovic The Journal of Organic Chemistry 77 (24), 11200-11209, 2012 | 37 | 2012 |
Vacuum matrix-assisted ionization source offering simplicity, sensitivity, and exceptional robustness in mass spectrometry S Trimpin, M Pophristic, A Adeniji-Adele, JW Tomsho, CN McEwen Analytical chemistry 90 (19), 11188-11192, 2018 | 27 | 2018 |
Identification of inhibitors of a bacterial sigma factor using a new high-throughput screening assay SA El-Mowafi, E Sineva, JN Alumasa, H Nicoloff, JW Tomsho, SE Ades, ... Antimicrobial agents and chemotherapy 59 (1), 193-205, 2015 | 26 | 2015 |
Concentration-dependent processivity of multiple glutamate ligations catalyzed by folylpoly-γ-glutamate synthetase JW Tomsho, RG Moran, JK Coward Biochemistry 47 (34), 9040-9050, 2008 | 20 | 2008 |
Synthesis of (6 R)-and (6 S)-5, 10-dideazatetrahydrofolate oligo-γ-glutamates: Kinetics of multiple glutamate ligations catalyzed by folylpoly-γ-glutamate synthetase JW Tomsho, JJ McGuire, JK Coward Organic & biomolecular chemistry 3 (18), 3388-3398, 2005 | 15 | 2005 |
Protection of the benzoxaborole moiety: Synthesis and functionalization of zwitterionic benzoxaborole complexes JM Gamrat, G Mancini, SJ Burke, RC Colandrea, NR Sadowski, BC Figula, ... The Journal of Organic Chemistry 83 (11), 6193-6201, 2018 | 13 | 2018 |
Potassium haloalkyltrifluoroborate salts: synthesis, application, and reversible ligand replacement with MIDA SJ Burke, JM Gamrat, JR Santhouse, DT Tomares, JW Tomsho Tetrahedron Letters 56 (41), 5500-5503, 2015 | 12 | 2015 |
Synthesis and Antimicrobial Evaluation of γ-Borono Phosphonate Compounds in Escherichia coli and Mycobacterium smegmatis G Mancini, M Bouda, JM Gamrat, JW Tomsho ACS omega 4 (11), 14551-14559, 2019 | 10 | 2019 |
Boronic and borinic acid compound as inhibitors of sulfenic acid-containing proteins S Benkovic, C Liu, JW Tomsho US Patent 9,309,508, 2016 | 8 | 2016 |
Inhibition of human folylpolyglutamate synthetase by diastereomeric phosphinic acid mimics of the tetrahedral intermediate JJ McGuire, DM Bartley, JW Tomsho, WH Haile, JK Coward Archives of biochemistry and biophysics 488 (2), 140-145, 2009 | 8 | 2009 |
Folylpoly-γ-glutamate synthetase: Kinetics of multiple glutamate ligations JW Tomsho University of Michigan, 2005 | 3 | 2005 |
Synthesis of Boron-Containing Nucleoside Analogs LM Alhthlol, CL Orme, BS Jefferis, SA Herter, HE Kemper, JW Tomsho The Journal of Organic Chemistry 89 (3), 1556-1566, 2024 | 2 | 2024 |
Boronic and borinic acid compounds as inhibitors of sulfenic acid-containing proteins S Benkovic, C Liu, JW Tomsho US Patent 8,980,544, 2015 | 2 | 2015 |
Protective groups and methods for protecting benzoxaboroles or oxaboroles JW Tomsho, JM Gamrat US Patent 11,427,603, 2022 | 1 | 2022 |