| Benzothiazole-containing hydroxamic acids as histone deacetylase inhibitors and antitumor agents DTK Oanh, H Van Hai, SH Park, HJ Kim, BW Han, HS Kim, JT Hong, ... Bioorganic & medicinal chemistry letters 21 (24), 7509-7512, 2011 | 75 | 2011 |
| C-terminal HSP90 inhibitor L80 elicits anti-metastatic effects in triple-negative breast cancer via STAT3 inhibition TM Cho, JY Kim, YJ Kim, D Sung, E Oh, S Jang, L Farrand, VH Hoang, ... Cancer letters 447, 141-153, 2019 | 45 | 2019 |
| Discovery of potent human glutaminyl cyclase inhibitors as anti-Alzheimer’s agents based on rational design VH Hoang, PT Tran, M Cui, VTH Ngo, J Ann, J Park, J Lee, K Choi, H Cho, ... Journal of medicinal chemistry 60 (6), 2573-2590, 2017 | 45 | 2017 |
| Structure–activity relationship of human glutaminyl cyclase inhibitors having an N-(5-methyl-1H-imidazol-1-yl)propyl thiourea template PT Tran, VH Hoang, SA Thorat, SE Kim, J Ann, YJ Chang, DW Nam, ... Bioorganic & medicinal chemistry 21 (13), 3821-3830, 2013 | 40 | 2013 |
| TRPV1 antagonist with high analgesic efficacy: 2-Thio pyridine C-region analogues of 2-(3-fluoro-4-methylsulfonylaminophenyl) propanamides TH Ha, HC Ryu, SE Kim, HS Kim, J Ann, PT Tran, VH Hoang, K Son, ... Bioorganic & medicinal chemistry 21 (21), 6657-6664, 2013 | 28 | 2013 |
| Potent human glutaminyl cyclase inhibitors as potential anti-Alzheimer’s agents: Structure-activity relationship study of Arg-mimetic region VTH Ngo, VH Hoang, PT Tran, J Ann, M Cui, G Park, S Choi, J Lee, H Kim, ... Bioorganic & medicinal chemistry 26 (5), 1035-1049, 2018 | 23 | 2018 |
| Investigation of B, C-ring truncated deguelin derivatives as heat shock protein 90 (HSP90) inhibitors for use as anti-breast cancer agents HS Kim, VH Hoang, M Hong, KC Kim, J Ann, CT Nguyen, JH Seo, H Choi, ... Bioorganic & Medicinal Chemistry 27 (7), 1370-1381, 2019 | 22 | 2019 |
| Discovery of conformationally restricted human glutaminyl cyclase inhibitors as potent anti-Alzheimer’s agents by structure-based design VH Hoang, VTH Ngo, M Cui, NV Manh, PT Tran, J Ann, HJ Ha, H Kim, ... Journal of medicinal chemistry 62 (17), 8011-8027, 2019 | 21 | 2019 |
| Structure-activity relationship investigation of Phe-Arg mimetic region of human glutaminyl cyclase inhibitors VTH Ngo, VH Hoang, PT Tran, N Van Manh, J Ann, E Kim, M Cui, S Choi, ... Bioorganic & Medicinal Chemistry 26 (12), 3133-3144, 2018 | 21 | 2018 |
| A novel HSP90 inhibitor SL-145 suppresses metastatic triple-negative breast cancer without triggering the heat shock response JY Kim, TM Cho, JM Park, S Park, M Park, KD Nam, D Ko, J Seo, S Kim, ... Oncogene 41 (23), 3289-3297, 2022 | 19 | 2022 |
| 2-Aryl substituted pyridine C-region analogues of 2-(3-fluoro-4-methylsulfonylaminophenyl) propanamides as highly potent TRPV1 antagonists HC Ryu, S Seo, MS Kim, MY Kim, HS Kim, J Ann, PT Tran, VH Hoang, ... Bioorganic & medicinal chemistry letters 24 (16), 4044-4047, 2014 | 19 | 2014 |
| In vitro and in silico determination of glutaminyl cyclase inhibitors PT Tran, VH Hoang, J Lee, TTT Hien, NT Tung, ST Ngo RSC advances 9 (51), 29619-29627, 2019 | 17 | 2019 |
| Identifying possible AChE inhibitors from drug-like molecules via machine learning and experimental studies TH Nguyen, PT Tran, NQA Pham, VH Hoang, DM Hiep, ST Ngo ACS omega 7 (24), 20673-20682, 2022 | 16 | 2022 |
| Inhibition of glutaminyl cyclase ameliorates amyloid pathology in an animal model of Alzheimer's disease via the modulation of γ-secretase activity H Song, YJ Chang, M Moon, SK Park, PT Tran, VH Hoang, J Lee, ... Journal of Alzheimer's Disease 43 (3), 797-807, 2015 | 16 | 2015 |
| Discovery of highly potent human glutaminyl cyclase (QC) inhibitors as anti-Alzheimer's agents by the combination of pharmacophore-based and structure-based design N Van Manh, VH Hoang, VTH Ngo, J Ann, TH Jang, JH Ha, JY Song, ... European Journal of Medicinal Chemistry 226, 113819, 2021 | 12 | 2021 |
| α-Substituted 2-(3-fluoro-4-methylsulfonamidophenyl)acetamides as potent TRPV1 antagonists PT Tran, HS Kim, J Ann, SE Kim, C Kim, M Hong, VH Hoang, VTH Ngo, ... Bioorganic & medicinal chemistry letters 25 (11), 2326-2330, 2015 | 12 | 2015 |
| Design, synthesis and bioevaluation of novel 6-substituted aminoindazole derivatives as anticancer agents NX Hoang, VH Hoang, HN Luu, T Ngo, D Van Hieu, NH Long, ST Ngo, ... RSC advances 10 (73), 45199-45206, 2020 | 9 | 2020 |
| α-Methylated simplified resiniferatoxin (sRTX) thiourea analogues as potent and stereospecific TRPV1 antagonists HS Kim, MK Jin, SU Kang, JO Lim, PT Tran, VH Hoang, J Ann, TH Ha, ... Bioorganic & medicinal chemistry letters 24 (12), 2685-2688, 2014 | 7 | 2014 |
| Discovery of potent indazole-based human glutaminyl cyclase (QC) inhibitors as Anti-Alzheimer's disease agents N Van Manh, VH Hoang, VTH Ngo, S Kang, JJ Jeong, HJ Ha, H Kim, ... European Journal of Medicinal Chemistry 244, 114837, 2022 | 6 | 2022 |
| Design, synthesis and evaluation the bioactivities of novel 1, 3-dimethyl-6-amino-1H-indazole derivatives as anticancer agents VH Hoang, NTK Trang, TC Minh, TH Lan, NT Hue, TX Nguyen, ... Bioorganic & Medicinal Chemistry 90, 117377, 2023 | 5 | 2023 |
