Design, preparation, and implementation of an imidazole-based chiral biaryl P, N-ligand for asymmetric catalysis FSP Cardoso, KA Abboud, A Aponick Journal of the American Chemical Society 135 (39), 14548-14551, 2013 | 138 | 2013 |
Enantioselective Copper‐Catalyzed Quinoline Alkynylation M Pappoppula, FSP Cardoso, BO Garrett, A Aponick Angewandte Chemie 127 (50), 15417-15421, 2015 | 128 | 2015 |
Heck arylation of styrenes with arenediazonium salts: short, efficient, and stereoselective synthesis of resveratrol, DMU-212, and analogues AV Moro, FSP Cardoso, CRD Correia Tetrahedron Letters 49 (39), 5668-5671, 2008 | 98 | 2008 |
Highly regio-and stereoselective Heck reaction of allylic esters with arenediazonium salts: application to the synthesis of kavalactones AV Moro, FSP Cardoso, CRD Correia Organic letters 11 (16), 3642-3645, 2009 | 77 | 2009 |
A concise route to MK-4482 (EIDD-2801) from cytidine N Vasudevan, GP Ahlqvist, CP McGeough, DJ Paymode, FSP Cardoso, ... Chemical Communications 56 (87), 13363-13364, 2020 | 56 | 2020 |
Toward a practical, two-step process for molnupiravir: Direct hydroxamination of cytidine followed by selective esterification DJ Paymode, N Vasudevan, S Ahmad, AL Kadam, FSP Cardoso, ... Organic Process Research & Development 25 (8), 1822-1830, 2021 | 43 | 2021 |
Expanding access to remdesivir via an improved pyrrolotriazine synthesis: supply centered synthesis DJ Paymode, FSP Cardoso, T Agrawal, JW Tomlin, DW Cook, JM Burns, ... Organic Letters 22 (19), 7656-7661, 2020 | 37 | 2020 |
An efficient synthesis of tenofovir (PMPA): A key intermediate leading to tenofovir-based HIV medicines BP Derstine, JW Tomlin, CL Peck, JP Dietz, BT Herrera, FSP Cardoso, ... Organic Process Research & Development 24 (8), 1420-1427, 2020 | 24 | 2020 |
Application of In Situ FTIR for the Preparation of 17-α-Estradiol via Mitsunobu Reaction FSP Cardoso, GE Mickle, MA da Silva, PT Baraldi, FB Ferreira Organic Process Research & Development 20 (2), 306-311, 2016 | 14 | 2016 |
Nitrogen Nucleophiles in Au‐Catalyzed Dehydrative Cyclization Reactions JM Ketcham, FSP Cardoso, B Biannic, H Piras, A Aponick Israel Journal of Chemistry 53 (11‐12), 923-931, 2013 | 11 | 2013 |
Short and Efficient Synthesis of the Antituberculosis Agent Pretomanid from (R)-Glycidol T Lucas, JP Dietz, FSP Cardoso, DR Snead, RC Nelson, KO Donsbach, ... Organic Process Research & Development 27 (9), 1641-1651, 2023 | 4 | 2023 |
Regioselective Addition of Quinoline Derivatives to Carbonyl Compounds via Palladium-Catalyzed Umpolung with Diethylzinc Y Matsumoto, K Yamamoto, M Kuriyama, K Nishida, O Onomura Synthesis 51 (08), 1795-1802, 2019 | 3 | 2019 |
Practical and Scalable Two-Step Process for 6-(2-Fluoro-4-nitrophenyl)-2-oxa-6-azaspiro [3.3] heptane: A Key Intermediate of the Potent Antibiotic Drug Candidate TBI-223 FSP Cardoso, AL Kadam, RC Nelson, JW Tomlin, D Dahal, CS Kuehner, ... Organic Process Research & Development 27 (7), 1390-1399, 2023 | 2 | 2023 |
A Practical and Economical Route to (S)-Glycidyl Pivalate JM Noble, L Chang, D Chen, B Wang, RN Dominey, DW Cook, JM Burns, ... SynOpen 6 (04), 258-262, 2022 | 2 | 2022 |
Toward Secure Supply of Remdesivir via a 2-Pot Triazine Synthesis: Supply Centered Synthesis DJ Paymode, FSP Cardoso, JD Sieber, JW Tomlin, DW Cook, J Burns, ... | 1 | 2020 |
Biaryl ligands A Aponick, FSP Cardoso US Patent 9,994,599, 2018 | 1 | 2018 |
A New Approach to Atropisomerism FSP Cardoso, A Aponick Blucher Chemistry Proceedings 1 (2), 157-157, 2013 | 1 | 2013 |
Biaryl ligands, methods of making biarlyl ligands, and methods of use thereof A Aponick, FSP Cardoso US Patent 11,198,701, 2021 | | 2021 |
A Concise Route to MK-4482 (EIDD-2801) N Vasudevan, GP Ahlqvist, CP McGeough, DJ Paymode, FSP Cardoso, ... | | 2020 |
Biaryl ligands, methods of making biaryl ligands, and methods of use thereof A Aponick, FSP Cardoso US Patent 10,618,922, 2020 | | 2020 |