| Recent advances in the synthesis of 2H-1, 4-benzoxazin-3-(4H)-ones and 3, 4-dihydro-2H-1, 4-benzoxazines J Ilaš, PŠ Anderluh, MS Dolenc, D Kikelj Tetrahedron 61 (31), 7325-7348, 2005 | 188 | 2005 |
| Dual inhibitors of human DNA topoisomerase II and other cancer-related targets Z Skok, N Zidar, D Kikelj, J Ilaš Journal of medicinal chemistry 63 (3), 884-904, 2019 | 166 | 2019 |
| Discovery of benzothiazole scaffold-based DNA gyrase B inhibitors M Gjorgjieva, T Tomasic, M Barancokova, S Katsamakas, J Ilas, ... Journal of medicinal chemistry 59 (19), 8941-8954, 2016 | 126 | 2016 |
| Discovery of 4,5,6,7-Tetrahydrobenzo[1,2-d]thiazoles as Novel DNA Gyrase Inhibitors Targeting the ATP-Binding Site T Tomasic, S Katsamakas, Z Hodnik, J Ilaš, M Brvar, T Solmajer, ... Journal of medicinal chemistry 58 (14), 5501-5521, 2015 | 126 | 2015 |
| A road map for prioritizing warheads for cysteine targeting covalent inhibitors P Abranyi-Balogh, L Petri, T Imre, P Szijj, A Scarpino, M Hrast, A Mitrović, ... European journal of medicinal chemistry 160, 94-107, 2018 | 113 | 2018 |
| Toward a Novel Class of Antithrombotic Compounds with Dual Function. Discovery of 1,4-Benzoxazin-3(4H)-one Derivatives Possessing Thrombin Inhibitory and … P Štefanič Anderluh, M Anderluh, J Ilaš, J Mravljak, M Sollner Dolenc, ... Journal of medicinal chemistry 48 (9), 3110-3113, 2005 | 77 | 2005 |
| Antimicrobial activity of the marine alkaloids, clathrodin and oroidin, and their synthetic analogues N Zidar, S Montalvão, Ž Hodnik, DA Nawrot, A Žula, J Ilaš, D Kikelj, ... Marine drugs 12 (2), 940-963, 2014 | 71 | 2014 |
| 3,4-Dihydro-2H-1,4-benzoxazine Derivatives Combining Thrombin Inhibitory and Glycoprotein IIb/IIIa Receptor Antagonistic Activity as a Novel Class of … J Ilaš, Z Jakopin, T Borštnar, M Stegnar, D Kikelj Journal of medicinal chemistry 51 (18), 5617-5629, 2008 | 69 | 2008 |
| N-Phenyl-4,5-dibromopyrrolamides and N-Phenylindolamides as ATP Competitive DNA Gyrase B Inhibitors: Design, Synthesis, and Evaluation N Zidar, H Macut, T Tomasic, M Brvar, S Montalvao, P Tammela, ... Journal of medicinal chemistry 58 (15), 6179-6194, 2015 | 65 | 2015 |
| Discovery of substituted oxadiazoles as a novel scaffold for DNA gyrase inhibitors Ž Jakopin, J Ilaš, M Barančoková, M Brvar, P Tammela, MS Dolenc, ... European Journal of Medicinal Chemistry 130, 171-184, 2017 | 64 | 2017 |
| Synthesis and Evaluation of N‐Phenylpyrrolamides as DNA Gyrase B Inhibitors M Durcik, P Tammela, M Barančoková, T Tomašič, J Ilaš, D Kikelj, N Zidar ChemMedChem 13 (2), 186-198, 2018 | 58 | 2018 |
| Influence of different classes of crosslinkers on alginate polyelectrolyte nanoparticle formation, thermodynamics and characteristics J Mirtič, J Ilaš, J Kristl Carbohydrate polymers 181, 93-102, 2018 | 57 | 2018 |
| ATP-competitive DNA gyrase and topoisomerase IV inhibitors as antibacterial agents M Durcik, T Tomašič, N Zidar, A Zega, D Kikelj, LP Mašič, J Ilaš Expert opinion on therapeutic patents 29 (3), 171-180, 2019 | 55 | 2019 |
| Recent progress in the discovery and development of DNA gyrase B inhibitors M Barančoková, D Kikelj, J Ilaš Future medicinal chemistry 10 (10), 1207-1227, 2018 | 51 | 2018 |
| Design, synthesis and biological evaluation of 4,5-dibromo-N-(thiazol-2-yl)-1H-pyrrole-2-carboxamide derivatives as novel DNA gyrase inhibitors T Tomašič, M Mirt, M Barančoková, J Ilaš, N Zidar, P Tammela, D Kikelj Bioorganic & medicinal chemistry 25 (1), 338-349, 2017 | 50 | 2017 |
| New N-phenylpyrrolamide DNA gyrase B inhibitors: Optimization of efficacy and antibacterial activity M Durcik, D Lovison, Ž Skok, CD Cruz, P Tammela, T Tomašič, DB Tiz, ... European journal of medicinal chemistry 154, 117-132, 2018 | 49 | 2018 |
| Structure-activity relationships and molecular docking studies of chromene and chromene based azo chromophores: A novel series of potent antimicrobial and anticancer agents TH Afifi, RM Okasha, HEA Ahmed, J Ilaš, T Saleh, AS Abd-El-Aziz EXCLI journal 16, 868, 2017 | 49 | 2017 |
| An optimised series of substituted N-phenylpyrrolamides as DNA gyrase B inhibitors DB Tiz, Ž Skok, M Durcik, T Tomašič, LP Mašič, J Ilaš, A Zega, ... European journal of medicinal chemistry 167, 269-290, 2019 | 40 | 2019 |
| Exploring protein hotspots by optimized fragment pharmacophores D Bajusz, WS Wade, G Satała, AJ Bojarski, J Ilaš, J Ebner, F Grebien, ... Nature Communications 12 (1), 3201, 2021 | 39 | 2021 |
| New N-phenyl-4, 5-dibromopyrrolamides and N-Phenylindolamides as ATPase inhibitors of DNA gyrase N Zidar, T Tomašič, H Macut, A Sirc, M Brvar, S Montalvao, P Tammela, ... European Journal of Medicinal Chemistry 117, 197-211, 2016 | 38 | 2016 |
