Discovery of 3, 3′-diindolylmethanes as potent antileishmanial agents SB Bharate, JB Bharate, SI Khan, BL Tekwani, MR Jacob, R Mudududdla, ... European journal of medicinal chemistry 63, 435-443, 2013 | 107 | 2013 |
β-Glucuronidases of opportunistic bacteria are the major contributors to xenobiotic-induced toxicity in the gut P Dashnyam, R Mudududdla, TJ Hsieh, TC Lin, HY Lin, PY Chen, CY Hsu, ... Scientific reports 8 (1), 16372, 2018 | 90 | 2018 |
Tandem one-pot synthesis of flavans by recyclable silica–HClO 4 catalyzed Knoevenagel condensation and [4+ 2]-Diels–Alder cycloaddition SB Bharate, R Mudududdla, JB Bharate, N Battini, S Battula, RR Yadav, ... Organic & Biomolecular Chemistry 10 (26), 5143-5150, 2012 | 43 | 2012 |
Synthesis and biological evaluation of indoloquinoline alkaloid cryptolepine and its bromo-derivative as dual cholinesterase inhibitors VK Nuthakki, R Mudududdla, A Sharma, A Kumar, SB Bharate Bioorganic Chemistry 90, 103062, 2019 | 40 | 2019 |
Efficient synthesis of 2, 3-dihydroquinazolin-4 (1H)-ones using heterogeneous solid acid catalysts: unexpected formation of SB Bharate, N Mupparapu, S Manda, JB Bharate, R Mudududdla, ... Arkivoc 8, 308-318, 2012 | 38 | 2012 |
ortho-Amidoalkylation of Phenols via Tandem One-Pot Approach Involving Oxazine Intermediate R Mudududdla, SK Jain, JB Bharate, AP Gupta, B Singh, ... The Journal of Organic Chemistry 77 (19), 8821-8827, 2012 | 30 | 2012 |
3-(Benzo [d][1, 3] dioxol-5-ylamino)-N-(4-fluorophenyl) thiophene-2-carboxamide overcomes cancer chemoresistance via inhibition of angiogenesis and P-glycoprotein efflux pump … R Mudududdla, SK Guru, A Wani, S Sharma, P Joshi, RA Vishwakarma, ... Organic & Biomolecular Chemistry 13 (14), 4296-4309, 2015 | 23 | 2015 |
Discovery of benzoylsulfonohydrazides as potent inhibitors of the histone acetyltransferase KAT6A DJ Leaver, B Cleary, N Nguyen, DL Priebbenow, HR Lagiakos, ... Journal of medicinal chemistry 62 (15), 7146-7159, 2019 | 22 | 2019 |
Synthesis of 2-phenylnaphthalenes from styryl-2-methoxybenzenes R Mudududdla, R Sharma, S Abbat, PV Bharatam, RA Vishwakarma, ... Chemical Communications 50 (81), 12076-12079, 2014 | 21 | 2014 |
Deformylation of indole and azaindole-3-carboxaldehydes using anthranilamide and solid acid heterogeneous catalyst via quinazolinone intermediate RR Yadav, N Battini, R Mudududdla, JB Bharate, N Muparappu, ... Tetrahedron Letters 53 (17), 2222-2225, 2012 | 14 | 2012 |
Orally Effective Aminoalkyl 10H‐Indolo[3,2‐b]quinoline‐11‐carboxamide Kills the Malaria Parasite by Inhibiting Host Hemoglobin Uptake R Mudududdla, D Mohanakrishnan, SS Bharate, RA Vishwakarma, ... ChemMedChem 13 (23), 2581-2598, 2018 | 13 | 2018 |
Nonantioxidant tetramethoxystilbene abrogates α-synuclein-induced yeast cell death but not that triggered by the Bax or βA4 peptide A Derf, R Mudududdla, D Akintade, IS Williams, M Abdullaha, ... ACS omega 3 (8), 9513-9532, 2018 | 13 | 2018 |
Role of basic aminoalkyl chains in the lead optimization of Indoloquinoline alkaloids VK Nuthakki, R Mudududdla, SB Bharate European Journal of Medicinal Chemistry 227, 113938, 2022 | 10 | 2022 |
Discovery of acylsulfonohydrazide-derived inhibitors of the lysine acetyltransferase, KAT6A, as potent senescence-inducing anti-cancer agents DL Priebbenow, DJ Leaver, N Nguyen, B Cleary, HR Lagiakos, ... Journal of medicinal chemistry 63 (9), 4655-4684, 2020 | 10 | 2020 |
Tetramethoxystilbene inhibits NLRP3 inflammasome assembly via blocking the oligomerization of apoptosis-associated speck-like protein containing caspase recruitment domain: in … M Abdullaha, M Ali, D Kour, R Mudududdla, P Khajuria, A Kumar, ... ACS Pharmacology & Translational Science 4 (4), 1437-1448, 2021 | 9 | 2021 |
ortho-Quinone methides: TFA-mediated generation in water and trapping with lactams and styrenes R Sharma, S Abbat, R Mudududdla, RA Vishwakarma, PV Bharatam, ... Tetrahedron letters 56 (27), 4057-4059, 2015 | 8 | 2015 |
Trifluoroacetic acid catalyzed thiophenylmethylation and thioalkylmethylation of lactams and phenols via domino three-component reaction in water R Mudududdla, R Sharma, SK Guru, M Kushwaha, AP Gupta, SS Bharate, ... RSC Advances 4 (27), 14081-14088, 2014 | 8 | 2014 |
Development of [18F] MIPS15692, a radiotracer with in vitro proof-of-concept for the imaging of MER tyrosine kinase (MERTK) in neuroinflammatory disease SW Wong, L Vivash, R Mudududdla, N Nguyen, SJ Hermans, ... European Journal of Medicinal Chemistry 226, 113822, 2021 | 6 | 2021 |
The first method for C-devinylation of aromatic systems SB Bharate, R Mudududdla, R Sharma, RA Vishwakarma Tetrahedron Letters 54 (23), 2913-2915, 2013 | 5 | 2013 |
Design, development, and optimisation of smart linker chemistry for targeted colonic delivery—in vitro evaluation HS Abd-Ellah, R Mudududdla, GP Carter, JB Baell Pharmaceutics 15 (1), 303, 2023 | 2 | 2023 |