Enhancement of solubility and dissolution rate of quercetin with solid dispersion system formation using hydroxypropyl methyl cellulose matrix

D Setyawan, AA Fadhil, D Juwita… - Thai Journal of …, 2017 - repository.unair.ac.id
Purpose: The aim of the present study was to obtain raw quercetin materials using solid
dispersion system with better solubility and dissolution rate than pure quercetin. Methods …

PEG 8000 increases solubility and dissolution rate of quercetin in solid dispersion system

D Setyawan, S Febrianti, A Zainul… - Marmara Journal of …, 2017 - repository.unair.ac.id
The aim of this study was to examine the physical characteristics, solubility, and in vitro
dissolution profile of quercetin-PEG 8000 solid dispersion prepared by melting method …

Improvement in vitro dissolution rate of quercetin using cocrystallization of quercetin-malonic acid

D Setyawan, SA Permata, A Zainul… - Indonesian Journal of …, 2018 - journal.ugm.ac.id
The aim of the study was to improve the in-vitro dissolution rate of quercetin (Qu) using
cocrystallization of quercetin. Cocrystals of quercetin (Co Qu) were produced with malonic …

[PDF][PDF] Preparation and characterization of quercetin-polyvinylpyrrolidone K-30 spray dried solid dispersion

PI Febriyenti, E Zaini, F Ismed… - Journal of Pharmacy & …, 2020 - academia.edu
Abstract Resumen Context: The use of quercetin as a potential active pharmaceutical
ingredient is limited by low aqueous solubility leading to low bioavailability. A spray-dried …

[HTML][HTML] Physicochemical characterization and in vitro dissolution test of quercetin-succinic acid co-crystals prepared using solvent evaporation

D Setyawan, IP Oktavia, R Farizka… - Turkish Journal of …, 2017 - ncbi.nlm.nih.gov
Objectives: Quercetin is one of the flavonoids with a polyhydroxyaromatic structure.
Quercetin has been proposed to exhibit a bioWactivity against oxidative stress. However …

The amorphous quercetin/hydroxypropylmethylcellulose acetate succinate solid dispersions prepared by co-precipitation method to enhance quercetin dissolution

Y Wang, Y Fang, F Zhou, Q Liang, Y Deng - Journal of Pharmaceutical …, 2021 - Elsevier
Abstract HPMCAS-HF, HPMCAS-MF and HPMCAS-LF were used as carriers to prepare the
amorphous solid dispersions (ASDs) of quercetin (Que) by co-precipitation. The Que ASD …

Solubility and dissolution enhancement of quercetin via preparation of spray dried microstructured solid dispersions

ASM Ghanem, H Saleh… - The Thai Journal of …, 2013 - digital.car.chula.ac.th
Solubility and dissolution enhancement of quercetin via preparation of spray dried
microstructured solid dispersions Page 1 The Thai Journal of Pharmaceutical Sciences Volume …

Novel formulation strategy to enhance solubility of quercetin

PN Kendre, VV Pande, KM Chavan - Pharmacophore, 2014 - pharmacophorejournal.com
The aim of present study to enhance the solubility of quercetin, a poorly water soluble drug,
quercetin containing blends (keeping total concentration 40% w/v, constant) was fabricated …

Preparation of quercetin nanorod/microcrystalline cellulose formulation via fluid bed coating crystallization for dissolution enhancement

F Sheng, PS Chow, J Hu, S Cheng, L Guo… - International journal of …, 2020 - Elsevier
This study reports a novel quercetin nanorod/microcrystalline cellulose (MCC) formulation
prepared by fluid bed coating crystallization technique. The process comprises fluidized bed …

Quercetin amorphous solid dispersions prepared by hot melt extrusion with enhanced solubility and intestinal absorption

X Shi, N Fan, G Zhang, J Sun, Z He… - Pharmaceutical …, 2020 - Taylor & Francis
The aim of this study was to investigate the effect of amorphous solid dispersions (ASDs) on
the dissolution rate and oral bioavailability of Quercetin (Que). First, we prepared the Que …